Benzoyl derivatives

ABSTRACT

Benzoyl derivatives of the formula I ##STR1## where the substituents L, M, X, Y and n have the meaning given in claim 1 and 
     Q for [sic] a cyclohexane-1,3-dione ring, which is linked in the 2-position, of the formula II, ##STR2## where R 15 , R 16 , R 18  and R 20  are hydrogen or C 1  -C 4  -alkyl, 
     R 19  is hydrogen, C 1  -C 4  -alkyl or a group --COOR 14 , 
     R 17  is hydrogen, C 1  -C 4  -alkyl, C 3  -C 4  -cycloalkyl, it being possible for these groups, if desired, to carry one to three of the following substituents: halogen, C 1  -C 4  -alkylthio or C 1  -C 4  -alkoxy, 
     or 
     R 17  is tetrahydropyran-3-yl, tetrahydropyran-4-yl or tetrahydrothiopyran-3-yl 
     or 
     R 17  and R 20  together form a bond or a three to six-membered carbocyclic ring, 
     where in the case where Y=C═O, X is not equal to NR 23 , 
     and agriculturally utilizable salts, a process for their preparation and their use as herbicides are described.

This application is a 371 of PCT/EP96/03800 filed Aug. 29, 1996.

The present invention relates to novel benzoyl derivatives having herbicidal action, processes for preparing the benzoyl derivatives, compositions which contain the latter and the use of these derivatives or compositions containing the latter for controlling weeds.

Herbicidally active 2-aroylcyclohexanediones are disclosed in the literature, for example in EP 283261, EP 90262, EP 135191, EP 186118, EP 186119, EP 186120, EP 319075, WO 9005712, WO 9404524, WO 9408988, JO3052862 and JO 3120202.

The herbicidal properties of the known compounds and the tolerability for crop plants, however, are only satisfactory to a limited extent.

It is an object of the present invention to find novel 2-aroylcyclohexanediones having improved properties.

We have found that this object is achieved by the benzoyl derivatives of the formula I ##STR3## where the substituents have the following meanings: L and M are hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, it being possible for these groups to be unsubstituted or substituted by one to five halogen atoms or C₁ -C₄ -alkoxy; halogen, cyano, nitro, a group --(A)_(m) --S(O)_(n) R¹ or a group --(A)_(m) --CO--R² ;

Y is C═O, C═N--R³, CR⁷ --NR⁵ R⁶, CR⁷ --OR⁸, CR¹⁰ R¹¹, CR⁷ --SR⁸ ; 1, 3-dioxanyl or 1,3-dioxolanyl substituted by hydrogen or C₁ -C₄ -alkyl; a heteroatom selected from the group oxygen, sulfur and nitrogen;

X is a chain (--CR¹² R¹³ --), (--CR¹² R¹³ --CR²¹ R²² --), (--CR¹² ═CR¹³ --), (--CR¹² R¹³ --CR¹² ═CR¹³ --); NR²³ the bond between X and Y can be saturated or unsaturated;

A is 0 or NR¹⁴ ;

m is zero or one;

n is zero, one or two;

R¹ is C₁ -C₄ -alkyl, C₁ -C₄ -haloalkyl or NR¹⁴ ;

R² is C₁ -C₄ -alkyl, C₁ -C₄ -haloalkyl, C₁ -C₄ -alkoxy or NR¹⁴ ;

R³ is hydrogen, --NR⁹ R⁴ ; C₁ -C₆ -alkyl, C₁ -C₆ -haloalkyl, C₁ -C₆ -alkoxy, C₁ -C₆ -haloalkoxy, C₂ -C₆ -alkenyl, C₂ -C₆ -haloalkenyl, C₂ -C₆ -alkynyl; monosubstituted to polysubstituted phenyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro; mono- to polysubstituted benzyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro; mono- to polysubstituted benzyloxy, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro;

R⁴ is hydrogen, C₁ -C₆ -alkyl, C₁ -C₆ -haloalkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C═O--NR¹⁴ ; monosubstituted to polysubstituted phenyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro; mono- to polysubstituted benzyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro;

R⁹ is hydrogen, C₁ -C₆ -alkyl, C₁ -C₆ -haloalkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C═O--NR¹⁴ ; monosubstituted to polysubstituted phenyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro; mono- to polysubstituted benzyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro;

R⁵ and R⁶ independently of one another are hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₁ -C₄ -haloalkyl, C₂ -C₆ -haloalkenyl, C₁ -C₆ -alkoxy, C₁ -C₆ -haloalkoxy; monosubstituted to polysubstituted phenyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro; mono- to polysubstituted benzyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro;

R⁷ is hydrogen, C₁ -C₆ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C_(l) -C₄ -haloalkoxy; substituted or unsubstituted phenyl, it being possible for the substituents to consist of one to three halogens, C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, nitro; R⁷ and R²¹ or R⁷ and R²³ or R⁷ and R¹² can form a bond;

R⁸ is hydrogen, C₁ -C₆ -alkyl, C₁ -C₄ -haloalkyl, substituted phenyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro; substituted benzyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro;

R¹⁰ and R¹¹ independently of one another are hydrogen, C₁ -C₆ -alkyl; phenyl which is unsubstituted or substituted by one to three halogens, C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, nitro; R¹⁰ and R¹² or R¹⁰ and R²³ or R¹⁰ and R²¹ can form a bond;

R¹² and R¹³ independently of one another are hydrogen, C₁ -C₆ -alkyl, C₁ -C₆ -haloalkyl, C₁ -C₆ -alkoxy, C₁ -C₆ -haloalkoxy; unsubstituted or substituted phenyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro;

R¹⁴ is C₁ -C₄ -alkyl;

R²¹ is hydrogen, C₁ -C₆ -alkyl, C₁ -C₆ -haloalkyl, C₁ -C₆ -alkoxy, C₁ -C₆ -haloalkoxy; unsubstituted or substituted phenyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro;

R²² is hydrogen, C₁ -C₆ -alkyl, C₁ -C₆ -haloalkyl, C₁ -C₆ -alkoxy, C₁ -C₆ -haloalkoxy; unsubstituted or substituted phenyl, it being possible for the substituents to consist of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro;

R²³ is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₁ -C₆ -alkoxy; phenyl or benzyl which is unsubstituted or substituted by C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano, nitro;

Q is a cyclohexane-1,3-dione ring, which is linked in the 2-position, of the formula II, ##STR4## where R¹⁵, R¹⁶, R¹⁸, and R²⁰ are hydrogen or C₁ -C₄ -alkyl,

R¹⁹ is hydrogen, C₁ -C₄ -alkyl or a group --COOR¹⁴,

R¹⁷ is hydrogen, C₁ -C₄ -alkyl, C₃ -C₄ -cycloalkyl, it being possible for these groups, if desired, to carry one to three of the following substituents: halogen, C₁ -C₄ -alkylthio or C₁ -C₄ -alkoxy,

or

R¹⁷ is tetrahydropyran-3-yl, tetrahydropyran-4-yl or tetrahydrothiopyran-3-yl,

or

R¹⁷ and R²⁰ together form a bond or a three to six-membered carbocyclic ring,

where in the case where Y=C═O, X is not equal to NR²³,

and agriculturally customary salts of the compound [sic] I.

Compounds of the formula Ia-Ie are obtained by reacting compounds of the formula II with a benzoic acid derivative of the formula III and rearranging to give benzoyl derivatives of the formula Ia-Ie. ##STR5##

In the above scheme 1, T in said formulae has the meaning halogen or OH and L, M, X, Y and n have the meanings given above.

The first step of the reaction sequence, the acylation, is carried out in a generally known manner, e.g. by adding an acid chloride of the formula III (T=Cl) or a carboxylic acids III (T=OH) activated, for example, with DCC (dicyclocarbodiimides or similar agents known from the literature, e.g. triphenylphosphine/DEAD=diethyl azodicarboxylate, 2-pyridine disulfide/triphenylphosphine to the solution or suspension of a cyclohexanedione II, if appropriate in the presence of an auxiliary base. The reactants and the auxiliary base are in this case expediently employed in equimolar amounts. A small excess, e.g. from 1.2 to 1.5 molar equivalents, based on II, of the auxiliary base can be advantageous under certain circumstances.

Suitable auxiliary bases are tertiary alkylamines, pyridine or alkali metal carbonates. The solvents used can be, e.g. methylene chloride, dioxane, diethyl ether, toluene, acetonitrile or ethyl acetate.

During the addition of the acid chloride, the reaction mixture is preferably cooled to from 0 to 10° C., then it is stirred at from 20 to 100° C., in particular 25 to 50° C., until the reaction is complete. working up is carried out in the customary manner, e.g. the reaction mixture is poured into water and the useful product is extracted, e.g. with methylene chloride. After drying the organic phase and removing the solvent, the crude enol ester can be employed without further purification for the rearrangement. Preparation examples for benzoyl enol esters of cyclohexane-1,3-diones are found, for example, EP-A 186 118 or U.S. Pat. No. 4,780,127.

The rearrangement of the enol esters to the compounds of the formula Ia-Ie is expediently carried out at from 20 to 40° C. in a solvent and in the presence of an auxiliary base and also with the aid of a cyano compound as a catalyst.

The solvents used can be, e.g. acetonitrile, methylene chloride, 1,2-dichloroethane, ethyl acetate or toluene. A preferred solvent is acetonitrile. Suitable auxiliary bases are tertiary alkylamines, pyridine or alkali metal carbonates, which are preferably employed in equimolar amounts or up to a four-fold excess, based on the benzoyl enol ester. A preferred auxiliary base is triethylamine in twice the amount.

Suitable catalysts are potassium cyanide, acetone cyanohydrin and trimethylsilyl cyanide, preferably in an amount of from 1 to 50 mol percent, based on the enol ester. Preferably, acetone cyanohydrin is added, e.g. in the amounts from 5 to 15, in particular 10 mol percent. Examples of the cyanide-catalyzed rearrangement of enol esters are found, for example, in EP-A 186118 or U.S. Pat. No. 4,780,127.

Working up is carried out in a manner known per se, e.g. the reaction mixture is acidified with dilute mineral acids such as 5% strength hydrochloric acid or sulfuric acid and extracted with an organic solvent such as methylene chloride or ethyl acetate. For purification, the extract is extracted with cold 5 to 10% strength alkali metal carbonate solution, the final product passing into the aqueous phase. By acidifying the aqueous solution, the product of the formula Ia-Ie is precipitated or extracted again with methylene chloride or ethyl acetate, dried and then freed from the solvent.

The 1,3-diketones of the formula II used as a starting material are known and can be prepared by processes known per se, such as are described, for example, in EP-A 71707, EP-A 142741, EP-A 243313, U.S. Pat. No. 4,249,937 and WO 92/13821. Cyclohexanedione and imedone are commercially available compounds.

Benzoic acids of the formula III can be prepared as follows:

Benzoyl halides, for example benzoyl chlorides of the formula III (T=Cl), are prepared in a known manner by reacting the benzoic acids of the formula III (T=OH) with thionyl chloride.

The benzoic acids of the formula III (T=OH) can be prepared in a known manner by acidic or basic hydrolysis of the corresponding esters of the formula III (T=C₁ -C₄ -alkoxy).

The intermediates of the formula III are known in some cases or can be prepared by processes known from the literature. ##STR6##

After this, for example, arylthio compounds IV as shown in scheme 2 can be reacted with substituted haloalkenyl as described in J. Med. Chem. 1984, 27, 1516, substituted alkynylcarboxylic acids as described in J. Org. Chem. 1980, 45, 4611 or J. Am. Chem. Soc. 1983, 105, 883, substituted haloalkylcarboxylic acids as desribed in Chem. Ber. 1925, 58, 1612 in the presence of a base such as alkali metal hydroxide, alkali metal hydride or alkali metal carbonate. The resulting compounds V are cyclized to VI under Friedel-Crafts conditions with addition of a Lewis acid 45 or a protic acid. Preferred Lewis acids are AlCl₃ or SnCl₄ and preferred protic acids are polyphoshoric acid and sulfuric acid as described in Can. J. Chem. 1981, 59, 199; Chem. Ber. 1925, 58, 1625; Chem. Ber. 1926, 59, 1074; Phosp. and Sulf. 1984, 19, 31.

Thiochromenone acids can furthermore be prepared by, for example, elimination of hydrogen halide from 3-halothiochromanone acids or, for example, by reaction of the substituted thiophenol acids with substituted α-alkylacetic esters in the presence of phosphorus pentoxide as described in Ann. Chem. 1964, 680, 40.

The arylthio compounds IV can be obtained, for example, by Sandmeyer reaction from corresponding anilines, which for their part are synthesized by reduction of suitable nitro compounds as described in Organicum 19th Edition 1992, 552 ff.

In the case where, for example, X is equal to (--CR¹² R¹³ --) or (--CR¹² R¹³ CR²¹ R²² --), Y is equal to C═O and T is equal to C₁ -C₄ -alkoxy, the thiochromonone ester or dihydrobenzothiophene ester as described in scheme 2 can be prepared by alkylation of the arylthio compound IV with halopropionic acid or haloacetic acid in solvent or water in the presence of one of the abovementioned bases and cyclized to VI.

The reactants and the base are in this case expediently employed in equimolar amounts. The reaction mixture is preferably stirred at 20-100° C., in particular at 20-40° C. Working-up is carried out, for example, in such a way that the reaction mixture is poured onto water, the aqueous phase is rendered acidic using mineral acids such as hydrochloric acid or sulfuric acid and the useful product is filtered off with suction or extracted by extraction with methylene chloride or ethyl acetate, and the extract is dried and freed from the solvent. The ester can be reacted without further purification.

By stirring V in, for example, polyphosphoric acid at 40-140° C., in particular at 70-100° C., or by activating the carboxylic acid by conversion into the acid chloride and stirring with 2-6, in particular 3.5 to 4.5, mol equivalents of a Lewis acid such as AlCl₃ or SnCl₄ in a solvent or by stirring with or in sulfuric acid, an intermediate of the formula III is obtained by working up in a manner known per se, ie. adding ice water and filtering off the useful product with suction or extracting the aqueous phase with ethyl acetate or methylene chloride, drying and removing the solvent.

In the case where, for example, X is equal to an ethylene group (--CR¹² ═CR¹³ --), Y is equal to C═O and T is equal to C₁ -C₄ -alkoxy, the thiochromenone ester can be converted by, for example, reaction of an arylthio compound with an acetylenecarboxylic acid derivative in water or solvent at 0-140° C. Working up is carried out in a manner known per se by adding water and dilute mineral acid, e.g. hydrochloric acid. The useful product is either filtered off with suction or obtained by extraction with methylene chloride or ethyl acetate, then drying and removing the solvent.

The intermediates of the formula III can be further functionalized by reactions known from the literature, such as reduction as described in Jerry March, Advanced Organic Chemistry, Fourth Ed., e.g. p.910ff, oximation as described in Jerry March, Advanced Organic Chemistry, Fourth Ed., e.g. p. 934, 935, 1039, 1226, 405ff, conversion into imines and amines as described in Jerry March, Advanced Organic Chemistry, Fourth Ed., ketalization, alkylation, halogenation, elimination and oxidation as described in Jerry March, Advanced Organic Chemistry, Fourth Ed.

The acids of the 3-alkoxy-1,2-benzisothiazole-1,1-dioxides or 3-alkoxy-1,2-benzisothiazoles can be obtained starting from corresponding saccharin derivatives or 1,2-benzisothiazoles by, for example, reaction with PCl₅, POCl₃ or chlorine and alcohol, if appropriate in the presence of an auxiliary base such as triethylamine, which is described, for example, in U.S. Pat. No. 4,571,429, Arch. Pharm. 1984, 317, 807, U.S. Pat. Nos. 4,461,901, 450,916, J. Med. Chem. 1986, 29, 359. Saccharincarboxylic acids can be obtained by processes known from the literature as described in Ann. Chem. 427, 231, 1922, Chem. Ber. 13, 1554, 1980, Chem. Ber. 25, 1740, 1892, German Offenlegungsschrift 3607343, German Patent Application P 44 27 995.7.

The derivatives of the benzo-1,4-oxathiin acids are known in some cases, e.g. from J. Org. Chem. 1968, 33, 456 or can be synthesized, for example, by reaction from the corresponding phenol derivatives as described in Chem. Comm., 1975, 451, J. Org. Chem. 1974, 39, 1811, J. Am. Chem. Soc. 1954, 76, 1068 or by combination of, for example, substitution reactions of halogen-substituted thiophenol derivatives and secondary reactions such as oxidation, reduction or addition as described in J. Het. Chem. 1983, 20, 867.

The benzoic acids of the formula III can also be obtained by reacting the corresponding bromo- or iodo-substituted compound of the formula VII ##STR7## T is OH, C₁ -C₄ -alkoxy Y,L,M,X, have the meanings described above

with carbon monoxide and water at elevated pressure in the presence of a palladium, nickel, cobalt or rhodium transition metal catalyst and a base.

The catalysts nickel, cobalt, rhodium and in particular palladium can be present in metallic form or in the form of customary salts, such as in the form of halogen compounds, e.g. PdCl₂, RhCl₃.H₂ O, acetates, e.g. Pd(OAc)₂, cyanides etc., in the known valency states. Metal complexes with tertiary phosphines, metal alkylcarbonyls, metal carbonyls, e.g. CO₂ (CO)₈, Ni(CO)₄, metal carbonyl complexes with tertiary phosphines, e.g. (PPh₃)₂ Ni(CO)₂, or transition metal salts complexed with tertiary phosphines can further be present. The last-mentioned embodiment is preferred, in particular, in the case of palladium as a catalyst. The nature of the phosphine ligands here is widely variable. For example, they can be represented by the following formulae: ##STR8## where n is the numbers 1, 2, 3 or 4 and the radicals R²⁴ to R²⁷ are low molecular weight alkyl, e.g. C₁ -C₆ -alkyl, aryl, C₁ -C₄ -alkylaryl, e.g. benzyl, phenethyl or aryloxy. Aryl is, for example, naphthyl, anthryl and preferably unsubstituted or substituted phenyl, where with respect to the substituents attention only has to be paid to their inertness to the carboxylation reaction, otherwise they can be widely varied and include all inert C-organic radicals such as C₁ -C₆ -alkyl radicals, e.g. methyl, carboxyl radicals such as COOH, COOM (M is, for example, an alkali metal, alkaline earth metal or ammonium salt or C-organic radicals bonded via oxygen, such as C₁ -C₆ -alkoxy radicals.

The phosphine complexes can be prepared in a manner known per se, e.g. as described in the documents mentioned at the outset. For example, the starting materials used are customary commercially available metal salts such as PdCl₂ or Pd(OCOCH₃)₂ and the phosphine for example P(C₆ H₅)₃, P(n-C₄ H₉)₃, PCH₃ (C₆ H₅)₂, 1,2-bis(diphenylphosphino)ethane is added.

The amount of phosphine, based on the transition metal, is customarily from 0 to 20, in particular 0.1 to 10, mol equivalents, particularly preferably 1 to 5 mol equivalents.

The amount of transition metal is not critical. Of course, for cost reasons, rather a small amount, e.g. from 0.1 to 10 mol %, in particular from 1 to 5 mol %, based on the starting substance II or III, is used.

For the preparation of the benzoic acids III (T=OH), the reaction is carried out with carbon monoxide and at least equimolar amounts of water, based on the starting substances VI. The reaction component water can simultaneously be used also as a solvent, ie. the maximum amount is not critical.

However, depending on the starting substances and the catalysts used, it can also be advantageous instead of the reaction component to use as the solvent another inert solvent or the base used for the carboxylation.

Suitable inert solvents are solvents customary for carboxylation reactions, such as hydrocarbons, e.g. toluene, xylene, hexane, pentane, cyclohexane, ethers, e.g. methyl tert-butyl ether, tetrahydrofuran, dioxane, dimethoxyethane, substituted amides such as dimethylformamide, persubstituted ureas such as tetra-C₁ -C₄ -alkylureas, or nitrites such as benzonitrile or acetonitrile.

In a preferred embodiment of the process, one of the reaction components, in particular the base, is used in an excess so that no additional solvent is necessary.

Bases suitable for the process are all inert bases which are able to bind the hydrogen iodide or hydrogen bromide liberated in the reaction. Examples which may be mentioned here are tertiary amines such as tert-alkylamines, e.g. trialkylamines such as triethylamine, cyclic amines such as N-methylpiperidine or N,N'-dimethylpiperazine, pyridine, alkali metal carbonates or hydrogen carbonates, or tetraalkyl-substituted urea derivatives such as tetra-C₁ -C₄ -alkylurea, e.g. tetramethylurea.

The amount of base is not critical, customarily from 1 to 10, in particular from 1 to 5, mol are used. When the base is simultaneously used as a solvent, the amount is generally proportioned such that the reaction components are dissolved, unnecessarily high excesses being avoided for practicability reasons, in order to save costs, to be able to employ small reaction vessels and to guarantee maximum contact of the reaction components.

During the reaction, the carbon monoxide pressure is adjusted such that an excess of CO, based on VI, is always present. Preferably, the carbon monoxide pressure at room temperature is from 1 to 250 bar, in particular from 5 to 150 bar of CO.

The carbonylation is generally carried out continuously or batchwise at from 20 to 250° C., in particular 30 to 150° C. In the case of batchwise operation, carbon monoxide is expediently injected into the reaction mixture continuously to maintain a constant pressure.

The arylhalogen compounds VII used as starting compounds are known or can easily be prepared by suitable combination of known syntheses and by reaction sequences described above.

With respect to the intended use of the benzoyl derivatives of the general formula I, suitable substituents are the following radicals:

L and M are hydrogen,

C₁ -C₆ -alkyl such as methyl, ethyl, propyl, 1-methylethyl, butyl, 1-methylpropyl, 2-methylpropyl, 1,1-dimethylethyl, pentyl, 1-methylbutyl, 2-methylbutyl, 3-methylbutyl, 1,1-dimethylpropyl, 1,2-dimethylpropyl, 2,2-dimethylpropyl, 1-ethylpropyl, hexyl, 1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1,1-dimethylbutyl, 1,2-dimethylbutyl, 1,3-dimethylbutyl, 2,2-dimethylbutyl, 2,3-dimethylbutyl, 3,3-dimethylbutyl, 1-ethylbutyl, 1,1,2-trimethylpropyl, 1,2,2-trimethylpropyl, 1-ethyl-1-methylpropyl or 1-ethyl-2-methylpropyl,

in particular methyl, ethyl, 1-methylethyl, 1-methylpropyl, 2-methylpropyl, 1, 1-dimethylethyl and 1, 1-dimethylpropyl;

C₂ -C₆ -alkenyl such as 2-propenyl, 2-butenyl, 3-butenyl, 1-methyl-2-propenyl, 2-methyl-2-propenyl, 2-pentenyl, 3-pentenyl, 4-pentenyl, 3-methyl-2-butenyl, 1-methyl-2-butenyl, 2-methyl-2-butenyl, 1-methyl-3-butenyl, 2-methyl-4-butenyl, 3-methyl-3-butenyl, 1,1-dimethyl-2-propenyl, 1,2-dimethyl-2-propenyl, 1-ethyl-2-propenyl, 2-hexenyl, 3-hexenyl, 4-hexenyl, 5-hexenyl, 1-methyl-2-pentenyl, 2-methyl-2-pentenyl, 3-methyl-2-pentenyl, 4-methyl-2-pentenyl, 1-methyl-3-pentenyl, 2-methyl-3-pentenyl, 3-methyl-3-pentenyl, 4-methyl-3-pentenyl, 1-methyl-4-pentenyl, 2-methyl-4-pentenyl, 3-methyl-4-pentenyl, 4-methyl-4-pentenyl, 1,1-dimethyl-2-butenyl, 1,1-dimethyl-3-butenyl, 1,2-dimethyl-2-butenyl, 1,3-dimethyl-3-butenyl, 2,2-dimethyl-3-butenyl, 2,3-dimethyl-2-butenyl, 2,3-dimethyl-3-butenyl, 1-ethyl-2-butenyl, 1-ethyl-3-butenyl, 2-ethyl-2-butenyl, 2-ethyl-3-butenyl, 1,1,2-trimethyl-2-propenyl, 1-ethyl-1-methyl-2-propenyl and ethyl-2-methyl-2-propenyl,

in particular 1-methyl-2-propenyl, 1-methyl-2-butenyl, 1,1-dimethyl-2-propenyl and 1,1-dimethyl-2-butenyl;

C₂ -C₆ -alkynyl such as propargyl, 2-butynyl, 3-butenyl, 2-pentynyl, 3-pentynyl, 4-pentynyl, 1-methyl-3-butynyl, 2-methyl-3-butynyl, 1-methyl-2-butynyl, 1,1-dimethyl-2-propynyl, 1-ethyl-2-propynyl, 2-hexynyl, 3-hexynyl, 4-hexynyl, 5-hexynyl, 1-methyl-2-pentynyl, 1-methyl-3-pentynyl, 1-methyl-4-pentynyl, 3-methyl-4-pentynyl, 4-methyl-2-pentynyl, 1,1-dimethyl-2-butynyl, 1,1-dimethyl-3-butynyl, 1,2-dimethyl-3-butynyl, 2,2-dimethyl-3-butynyl, 1-ethyl-2-butynyl, 1-ethyl-3-butynyl, 2-ethyl-3-butynyl and 1-ethyl-l-methyl-2-propynyl;

C₁ -C₄ -alkoxy such as methoxy, ethoxy, n-propoxy, 1-methylethoxy, n-butoxy, 1-methylpropoxy, 2-methylpropoxy and 1,1-dimethylethoxy,

in particular C₁ -C₃ -alkoxy such as methoxy, ethoxy or i-propoxy,

where these groups can be unsubstituted or substituted by one to five halogen atoms such as fluorine, chlorine, bromine and iodine, preferably fluorine and chlorine or C₁ -C₄ -alkoxy as mentioned above.

The group --(A)_(m) --S(O)_(n) R¹ defined above is, for example

C₁ -C₄ -alkylthio such as methylthio, ethylthio, n-propylthio, 1-methylethylthio, n-butylthio, 1-methylpropylthio, 2-methylpropylthio and 1,1-dimethylethylthio, in particular methylthio;

C₁ -C₄ -alkylsulfinyl such as methylsulfinyl, ethylsulfinyl, n-propylsulfinyl, 1-methylethylsulfinyl, n-butylsulfinyl, 1-methylpropylsulfinyl, 2-methylpropylsulfinyl and 1,1-dimethylethylsulfinyl, in particular methylsulfinyl;

C₁ -C₄ -alkylsulfonyl such as methylsulfonyl, ethylsulfonyl, n-propylsulfonyl, 1-methylethylsulfonyl, n-butylsulfonyl, 1-methylpropylsulfonyl, 2-methylpropylsulfonyl and 1,1-dimethylethylsulfonyl, in particular methylsulfonyl;

C₁ -C₄ -alkoxysulfonyl such as methoxysulfonyl, ethoxysulfonyl, n-propoxysulfonyl, 1-methylethoxysulfonyl, n-butoxysulfonyl, 1-methylpropoxysulfonyl, 2-methylpropoxysulfonyl and 1,1-dimethylethoxysulfonyl, in particular methoxysulfonyl;

N-C₁ -C₄ -alkylsulfamoyl such as N-methylsulfamoyl, N-ethylsulfamoyl, N-n-propylsulfamoyl, N-1-methylethylsulfamoyl, N-n-butylsulfamoyl, N-1,1-methylpropylsulfamoyl, N-2-methylpropylsulfamoyl and N-1,1-dimethylethylsulfamoyl, in particular N-methylsulfamoyl;

N-C₁ -C₄ -alkylsulfinamoyl such as N-methylsulfinamoyl, N-ethylsulfinamoyl, N-n-propylsulfinamoyl, N-1-methylethylsulfinamoyl, N-n-butylsulfinamoyl, N-1-methylpropylsulfinamoyl, N-2-methylpropylsulfinamoyl and N-1,1-dimethylethylsulfinamoyl, in particular N-methylsulfinamoyl;

di-C₁ -C₄ -alkylsulfamoyl such as dimethylsulfamoyl, diethylsulfamoyl, dipropylsulfamoyl, dibutylsulfamoyl, N-methyl-N-ethylsulfamoyl, N-methyl-N-propylsulfamoyl, N-methyl-N-1-methylethylsulfamoyl, N-methyl-N--C_(i), 1-dimethylethylsulfamoyl, di-1-methylethylsulfamoyl, N-ethyl-N-1-methylethylsulfamoyl and N-ethyl-N-1-dimethylethylsulfamoyl; in particular dimethylsulfamoyl;

di-C₁ -C₄ -alkylsulfinamoyl such as dimethylsulfinamoyl, diethylsulfinamoyl, dipropylsulfinamoyl, dibutylsulfinamoyl, N-methyl-N-ethylsulfinamoyl, N-methyl-N-propylsulfinamoyl, N-methyl-N-1-methylethylsulfinamoyl, N-methyl-N-1,1-dimethylethylsulfinamoyl, di-1-methylethylsulfinamoyl, N-ethyl-N-1-methylethylsulfinamoyl and N-ethyl-N-1,1-dimethylethylsulfinamoyl; in particular dimethylsulfinamoyl,

C₁ -C₄ -alkylsulfinyloxy such as methylsulfinyloxy, ethylsulfinyloxy, n-propylsulfinyloxy, 1-methylethylsulfinyloxy, n-butylsulfinyloxy, 1-methylpropylsulfinyloxy, 2-methylpropylsulfinyloxy and 1,1-dimethylethylsulfinyloxy, in particular methylsulfinyloxy;

C₁ -C₄ -alkylsulfonyloxy such as methylsulfonyloxy, ethylsulfonyloxy, n-propylsulfonyloxy, 1-methylethylsulfonyloxy, n-butylsulfonyloxy, 1-methylpropylsulfonyloxy, 2-methylpropylsulfonyloxy

and 1,1-dimethylethylsulfonyloxy, in particular methylsulfonyloxy;

C₁ -C₄ -alkylsulfinylamino such as methylsulfinylamino, ethyl sulfinylamino, n-propylsulfinylamino, 1-methylethylsulfinylamino, n-butylsulfinylamino, 1-methylpropylsulfinylamino, 2-methylpropylsulfinylamino and 1,1-dimethylethylsulfinylamino, in particular methylsulfinylamino;

C₁ -C₄ -alkylsulfonylamino such as methylsulfonylamino, ethylsulfonylamino, n-propylsulfonylamino, 1-methylethylsulfonylamino, n-butylsulfonylamino, 1-methylpropylsulfonylamino, 2-methylpropylsulfonylamino and 1,1-dimethylethylsulfonylamino, in particular methylsulfonylamino;

N-C₁ -C₄ -alkylsulfinyl-N-methylamino such as N-methylsulfinyl-N-methylamino, N-ethylsulfinyl-N-methylamino, N-n-propylsulfinyl-N-methylamino, N-1-methylethylsulfinyl-N-methylamino, N-n-butylsulfinyl-N-methylamino, N-1-methylpropylsulfinyl-N-methylamino, N-2-methylpropylsulfinyl-N-methylamino and N-1,1-dimethylethylsulfinyl-N-methylamino, in particular N-methylsulfinyl-N-methylamino;

N-C₁ -C₄ -alkylsulfinyl-N-ethylamino such as N-methylsulfinyl-N-ethylamino, N-ethylsulfinyl-N-ethylamino, N-n-propylsulfinyl-N-ethylamino, N-1-methylethylsulfinyl-N-ethylamino, N-n-butylsulfinyl-N-ethylamino, N-1-methylpropylsulfinyl-N-ethylamino, N-2-methylpropylsulfinyl-N-ethylamino and N-1,1-dimethylethylsulfinyl-N-ethylamino, in particular N-methylsulfinyl-N-ethylamino;

N-C₁ -C₄ -alkylsulfonyl-N-methylamino such as N-methylsulfonyl-N-methylamino, N-ethylsulfonyl-N-methylamino, N-n-propylsulfonyl-N-methylamino, N-1-methylethylsulfonyl-N-methylamino, N-n-butylsulfonyl-N-methyl-amino, N-1-methylpropylsulfonyl-N-methylamino, N-2-methylpropylsulfonyl-N-methylamino and N-1,1-dimethylethylsulfonyl-N-methylamino, in particular N-methylsulfonyl-N-methylamino;

N-C₁ -C₄ -alkylsulfonyl-N-ethylamino such as N-methylsulfonyl-N-ethylamino, N-ethylsulfonyl-N-ethylamino, N-n-propylsulfonyl-N-ethylamino, N-1-methylethylsulfonyl-N-ethylamino, N-n-butylsulfonyl-N-ethylamino, N-1-methylpropylsulfonyl-N-ethylamino, N-2-methylpropylsulfonyl-N-ethylamino and N-1,1-dimethylethylsulfonyl-N-ethylamino, in particular N-methylsulfonyl-N-ethylamino;

C₁ -C₄ -haloalkylthio such as chloromethylthio, dichloromethylthio, trichloromethylthio, fluoromethylthio, difluoromethylthio, trifluoromethylthio, chlorofluoromethylthio, chlorodifluoromethylthio, 1-fluoroethylthio, 2-fluoroethylthio, 2,2-difluoroethylthio, 2,2,2-trifluoroethylthio, 2-chloro-2,2-difluoroethylthio, 2,2-dichloro-2 fluoroethylthio, 2,2,2-trichloroethylthio and pentafluoroethylthio, in particular trifluoromethylthio.

The group --(A)_(m) --CO--R² defined above is, for example,

C₁ -C₄ -alkylcarbonyl such as methylcarbonyl, ethylcarbonyl, n-propylcarbonyl, 1-methylethylcarbonyl, n-butylcarbonyl, 1-methylpropylcarbonyl, 2-methylpropylcarbonyl and 1,1-dimethylethylcarbonyl, in particular methylcarbonyl;

C₁ -C₄ -alkoxycarbonyl such as methoxycarbonyl, ethoxycarbonyl, n-propoxycarbonyl, 1-methylethoxycarbonyl, n-butoxycarbonyl, 1-methylpropoxycarbonyl, 2-methylpropoxycarbonyl and 1,1-dimethylethoxycarbonyl, in particular methoxycarbonyl;

N-C₁ -C₄ -alkylcarbamoyl such as N-methylcarbamoyl, N-ethylcarbamoyl, N-n-propylcarbamoyl, N-1-methylethylcarbamoyl, N-n-butylcarbamoyl, N-1-methylpropylcarbamoyl, N-2-methylpropylcarbamoyl and N-1,1-dimethylethylcarbamoyl, in particular N-methylcarbamoyl;

di-C₁ -C₄ -alkylcarbamoyl such as dimethylcarbamoyl, diethylcarbamoyl, dipropylcarbamoyl, dibutylcarbamoyl, N-methyl-N-ethylcarbamoyl, N-methyl-N-propylcarbamoyl, N-methyl-N-1-methylethylcarbamoyl, N-methyl-N-1,1-dimethylethylcarbamoyl, di-1-methylethylcarbamoyl, N-ethyl-N-1-methylethylcarbamoyl and N-ethyl-N-1,1-dimethylethylcarbamoyl; in particular dimethylcarbamoyl;

C₁ -C₄ -alkylcarbonyloxy such as methylcarbonyloxy, ethylcarbonyloxy, n-propylcarbonyloxy, 1-methylethylcarbonyloxy, n-butylcarbonyloxy, 1-methylpropylcarbonyloxy, 2-methylpropylcarbonyloxy and 1,1-dimethylethylcarbonyloxy, in particular methylcarbonyloxy;

C₁ -C₄ -alkylcarbonylamino such as methylcarbonylamino, ethylcarbonylamino, n-propylcarbonylamino, 1-methylethylcarbonylamino, n-butylcarbonylamino, 1-methylpropylcarbonylamino, 2-methylpropylcarbonylamino and 1,1-dimethylethylcarbonylamino, in particular methylcarbonylamino;

N-C₁ -C₄ -alkylcarbonyl-N-methylamino such as N-methylcarbonyl-N-methylamino, N-ethylcarbonyl-N-methylamino, N-n-propylcarbonyl-N-methylamino, N-1-methylethylcarbonyl-N-methylamino, N-n-butylcarbonyl-N-methylamino, N-1-methylpropylcarbonyl-N-methylamino, N-2-methylpropylcarbonyl-N-methylamino and N-1,1-dimethylethylcarbonyl-N-methyl-amino, in particular N-methylcarbonyl-N-methylamino.

X is, for example: CH₂, CH(CH₃), C((CH₃)₂), CH(C₂ H₅), C((C₂ H₅)₂), CH(C₆ H₅), CH₂ --CH₂, CH₂ --CH(CH₃), CH₂ --C((CH₃)₂), CH(CH₃)--CH(CH₃), CH(CH₃)--C((CH₃)₂), C((CH₃)₂)--C((CH₃)₂), CH₂ --CH(C₂ H₅), CH₂ --C((C₂ H₅)₂), CH(C₂ H₅)--CH(C₂ H₅), CH(C₂ H₅)--C((C₂ H₅)₂), C((C₂ H₅)₂)--C((C₂ H₅)₂), CH₂ --CH(C₃ H₇), CH₂ --CH(iC₃ H₇), CH₂ --CH(C₄ H₉), CH₂ --CH(iC₄ H₉), CH₂ --CH(Br), CH₂ --C((Br)₂), CH(Br)--CH(Br), C((Br)₂)--C((Br)₂), CH₂ --CH(Cl), CH₂ --C((Cl)₂), CH(Cl)--C((Cl₂), C((Cl)₂)--C((Cl)₂), CH₂ --CH(C₆ H₅), CH(C₆ H₅)--CH(C₆ H₅), CH₂ --CH(p-NO₂ C₆ H₅)]CH═CH, C(CH₃)═CH, C(CH₃)═CCH₃, CH═CBr, CH═CCl, CBr═CBr, CCl═CCl, CH═C(OCH₃), CH═C(C₆ H₅), C(C₆ H₅)═C(C₆ H₅), C(C₂ H₅)═CH, C(C₂ H₅)═C(C₂ H₅), CH═C(C₃ H₅), CH═C(C₄ H₇), CH₂ --CH═CH, CH(CH₃)--C═CH, C((CH₃)₂)--CH═CH, CH₂ --CH═C(CH₃), CH₂ --C(CH₃)═CH, CH₂ --C(CH₃)═C(CH₃), CH(CH₃)--C(CH₃)═C(CH₃), C((CH₃)₂)--C(CH₃)═C(CH₃), N--H, N--CH₃, N--C₂ H₅, N--C₃ H₇, N--C₄ H₉, N-iCH₃ H₇, N--OCH₃, N--OC₂ H₅, N--CH₂ C₆ H₅, N--C₆ H₅ ;

Y is, for example:

C═O, CH--OH, CH--OCH₃, CH--OC₂ H₅, CH--OC₃ H₇, CH--OiPr, CH--OC₄ H₉, CH--OiBu, CH--OC₅ H₁₁, CH--OC₆ H₁₃, CH--OC₆ H₅, C(CH₃)--OCH₃, C(CH₃)--OC₂ H₅, C(CH₃)--OC₃ H₇, C(CH₃)--OC₄ H₉, C(CH₃)--OiPr, C(CH₃)--OiBu, C(CH₃)--OtBu, C(CH₃)--OPh, CH₂, CH(CH₃), C((CH₃)₂), C═N--CH₃, C═N--C₂ H₅, C═N-C₃ H₇, C═N-C₄ H₉, C═N-iC₄ H₉, C═N-tC₄ H₉, C═N-iPr, C═N--OCH₃, C═N-OC₂ H₅, C═N--OC₃ H₇, C═N--OC₄ H₉, C═N--OiC₄ H₉, C═N--OtC₄ H₉, C═N--OCH₂ CH═CH₂, C═N--OCH(CH₃)CH═CH₂, C═N--OCH₂ CH═CHCH₃, C═N--OCH₂ CH═C(CH₃)₂, C═N--OCH₂ CH═CHBr, C═N--OCH₂ CH═CHCl, C═N--OCH₂ CH═CHC₂ H₅, C═N--OCH₂ C.tbd.CH, C═N--OCH₂ C.tbd.CCH3, C═N--OCH₂ C₆ H₅, CH--NH(OCH₃), CH--NH(OC₂ H₅), CH--NH(OiPr), CH--NH(OnPr), CH--NH(OC₆ H₅), CH--NCH₃ (OCH₃), CH--NCH₃ (OC₂ H₅), CH--NCH₃ (OiPr), CH--NCH₃ (OnPr), CH--NCH₃ (OC₆ H₅), CH--NH(CH₃), CH--NH(C₂ H₅), CH--NH(C₃ H₇), CH--NH(C₄ H₉), CH--NH(iPr), CH--NH(iBu), CH--NH(tBu), CH--NH(C₆ H₅), CH--N(CH₃)₂, CH--NCH₃ (C₂ H₅), CH--NCH₃ (C₃ H₇), CH--NCH₃ (C₄ H₉), CH--NCH₃ (iPr), CH--NCH₃ (iBu), C═N--NH₂, C═N--NHCH₃, C═N--((CH₃)₂), C═N--NH(C₂ H₅), C═N--NCH₃ (C₂ H₅), C═N--N((C₂ H₅)₂), CH--SCH₃, CH--SC₂ H₅, CH--SC₃ H₇, CH--SC₄ H₉, CH--SPr, CH--SiBu, CH--SH, C(CH₃)--SCH₃, C(CH₃)--SC₂ H₅, C(CH₃)--SC₃ H₇, 1,3-dioxanyl, 1,3-dioxolanyl, 5,5-dimethyl-1,3-dioxanyl

Preferred benzoyl derivatives are those of the formula Ia, ##STR9## where L is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -alkylthio, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkylthio, C₁ -C₄ -alkylsulfonyl, halogen, nitro or cyano and M is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -alkylthio, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkylthio, C₁ -C₄ -alkylsulfonyl, halogen, nitro or cyano and Q, X, n and Y have the meanings given in claim 1, where in the case where Y=C═O, X is not equal to NR²³.

Furthermore preferred benzoyl derivatives are those of the formula Ib, ##STR10## where L is C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C_(-C) ₁ -C₄ -haloalkoxy, halogen, nitro or cyano and M is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano and Q, X, n and Y have the meanings given in claim 1, where in the case where Y=C═O, X is not equal to NR²³.

Preferred benzoyl derivatives are also those of the formula I as claimed in claim 1, where the radicals L and M are hydrogen, methyl, methoxy, chlorine, cyano, nitro or trifluoromethyl.

Preferred benzoyl derivatives are those of the formula Ic, ##STR11## where L is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano and M is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano and Q, n, Y and also R²², R²¹, R¹² and R¹³ have the meanings given in claim 1.

Likewise preferred benzoyl derivatives are those of the formula Id, ##STR12## where L is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano and M is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano and Q, n, Y and also R¹² and R¹³ have the meanings given in claim 1.

Also preferred benzoyl derivatives are those of the formula Ie, ##STR13## where L is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano and M is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano and Q, n, Y and also R¹² and R¹³ have the meanings given in claim 1.

Preferred benzoyl derivatives are likewise those of the formula I as claimed in claim 1, where n is 1 or 2 and Y is CR⁷ --OR⁸, where R⁷ and R⁸ have the meanings given in claim 1.

                                      TABLE 1                                      __________________________________________________________________________     Compounds of the formula                                                        ##STR14##                                                                     No.                                                                               R.sup.17                                                                          R.sup.18                                                                          R.sup.19                                                                          n R.sup.12                                                                          R.sup.13                                                                          Y          L M                                             __________________________________________________________________________     1.1                                                                               H  H  H  0 H  H  C═O    H H                                             1.2                                                                               H  H  H  2 H  H  C═O    H H                                             1.3                                                                               H  H  H  0 H  H  CHOCH.sub.3                                                                               H H                                             1.4                                                                               H  H  H  2 H  H  CHOCH.sub.3                                                                               H H                                             1.5                                                                               H  H  H  0 H  H  CHOC.sub.2 H.sub.5                                                                        H H                                             1.6                                                                               H  H  H  2 H  H  CHOC.sub.2 H.sub.5                                                                        H H                                             1.7                                                                               H  H  H  0 H  H  CHOiPr     H H                                             1.8                                                                               H  H  H  2 H  H  CHOiPr     H H                                             1.9                                                                               H  H  H  0 H  H  CHOH       H H                                             1.10                                                                              H  H  H  2 H  H  CHOH       H H                                             1.11                                                                              H  H  H  0 H  H  C═NOCH.sub.3                                                                          H H                                             1.12                                                                              H  H  H  2 H  H  C═NOCH.sub.3                                                                          H H                                             1.13                                                                              H  H  H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   H H                                             1.14                                                                              H  H  H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   H H                                             1.15                                                                              H  H  H  0 H  H  C═NOiPr                                                                               H H                                             1.16                                                                              H  H  H  2 H  H  C═NOiPr                                                                               H H                                             1.17                                                                              H  H  H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              H H                                             1.18                                                                              H  H  H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              H H                                             1.19                                                                              H  H  H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H H                                             1.20                                                                              H  H  H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H H                                             1.21                                                                              H  H  H  0 H  H  C(CH.sub.3).sub.2                                                                         H H                                             1.22                                                                              H  H  H  2 H  H  C(CH.sub.3).sub.2                                                                         H H                                             1.23                                                                              CH.sub.3                                                                          H  H  0 H  H  C═O    H H                                             1.24                                                                              CH.sub.3                                                                          H  H  2 H  H  C═O    H H                                             1.25                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOCH.sub.3                                                                               H H                                             1.26                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOCH.sub.3                                                                               H H                                             1.27                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOC.sub.2 H.sub.5                                                                        H H                                             1.28                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOC.sub.2 H.sub.5                                                                        H H                                             1.29                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOiPr     H H                                             1.30                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOiPr     H H                                             1.31                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOH       H H                                             1.32                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOH       H H                                             1.33                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.3                                                                          H H                                             1.34                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.3                                                                          H H                                             1.35                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   H H                                             1.36                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   H H                                             1.37                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOiPr                                                                               H H                                             1.38                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOiPr                                                                               H H                                             1.39                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              H H                                             1.40                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              H H                                             1.41                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H H                                             1.42                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H H                                             1.43                                                                              CH.sub.3                                                                          H  H  0 H  H  C(CH.sub.3).sub.2                                                                         H H                                             1.44                                                                              CH.sub.3                                                                          H  H  2 H  H  C(CH.sub.3).sub.2                                                                         H H                                             1.45                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═O    H H                                             1.46                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═O    H H                                             1.47                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOCH.sub.3                                                                               H H                                             1.48                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOCH.sub.3                                                                               H H                                             1.49                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOC.sub.2 H.sub.5                                                                        H H                                             1.50                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOC.sub.2 H.sub.5                                                                        H H                                             1.51                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOiPr     H H                                             1.52                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOiPr     H H                                             1.53                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.3                                                                          H H                                             1.54                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.3                                                                          H H                                             1.55                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   H H                                             1.56                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   H H                                             1.57                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOiPr                                                                               H H                                             1.58                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOiPr                                                                               H H                                             1.59                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              H H                                             1.60                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              H H                                             1.61                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H H                                             1.62                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H H                                             1.63                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C(CH.sub.3).sub.2                                                                         H H                                             1.64                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C(CH.sub.3).sub.2                                                                         H H                                             1.65                                                                              H  H  H  0 H  H  C═O    H CH.sub.3                                      1.66                                                                              H  H  H  2 H  H  C═O    H CH.sub.3                                      1.67                                                                              H  H  H  0 H  H  CHOCH.sub.3                                                                               H CH.sub.3                                      1.68                                                                              H  H  H  2 H  H  CHOCH.sub.3                                                                               H CH.sub.3                                      1.69                                                                              H  H  H  0 H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                      1.70                                                                              H  H  H  2 H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                      1.71                                                                              H  H  H  0 H  H  CHOiPr     H CH.sub.3                                      1.72                                                                              H  H  H  2 H  H  CHOiPr     H CH.sub.3                                      1.73                                                                              H  H  H  0 H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                      1.74                                                                              H  H  H  2 H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                      1.75                                                                              H  H  H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                      1 76                                                                              H  H  H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                      1.77                                                                              H  H  H  0 H  H  C═NOiPr                                                                               H CH.sub.3                                      1.78                                                                              H  H  H  2 H  H  C═NOiPr                                                                               H CH.sub.3                                      1.79                                                                              H  H  H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                      1.80                                                                              H  H  H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                      1.81                                                                              H  H  H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                      1.82                                                                              H  H  H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                      1.83                                                                              H  H  H  0 H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                      1.84                                                                              H  H  H  2 H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                      1.85                                                                              CH.sub.3                                                                          H  H  0 H  H  C═O    H CH.sub.3                                      1.86                                                                              CH.sub.3                                                                          H  H  2 H  H  C═O    H CH.sub.3                                      1.87                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOCH.sub.3                                                                               H CH.sub.3                                      1.88                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOCH.sub.3                                                                               H CH.sub.3                                      1.89                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                      1.90                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                      1.91                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOiPr     H CH.sub.3                                      1.92                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOiPr     H CH.sub.3                                      1.93                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                      1.94                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                      1.95                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                      1.96                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                      1.97                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOiPr                                                                               H CH.sub.3                                      1.98                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOiPr                                                                               H CH.sub.3                                      1.99                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                      1.100                                                                             CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                      1.101                                                                             CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                      1.102                                                                             CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                      1.103                                                                             CH.sub.3                                                                          H  H  0 H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                      1.104                                                                             CH.sub.3                                                                          H  H  2 H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                      1.105                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═O    H CH.sub.3                                      1.106                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═O    H CH.sub.3                                      1.107                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOCH.sub.3                                                                               H CH.sub.3                                      1.108                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOCH.sub.3                                                                               H CH.sub.3                                      1.109                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                      1.110                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                      1.111                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOiPr     H CH.sub.3                                      1.112                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOiPr     H CH.sub.3                                      1.113                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOH       H CH.sub.3                                      1.114                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOH       H CH.sub.3                                      1.115                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                      1.116                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                      1.117                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                      1.118                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                      1.119                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOiPr                                                                               H CH.sub.3                                      1.120                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOiPr                                                                               H CH.sub.3                                      1.121                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                      1.122                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                      1.123                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                      1.124                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                      1.125                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                      1.126                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                      1.127                                                                             H  H  H  0 H  H  C═O    H Cl                                            1.128                                                                             H  H  H  2 H  H  C═O    H Cl                                            1.129                                                                             H  H  H  0 H  H  CHOCH.sub.3                                                                               H Cl                                            1.130                                                                             H  H  H  2 H  H  CHOCH.sub.3                                                                               H Cl                                            1.131                                                                             H  H  H  0 H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                            1.132                                                                             H  H  H  2 H  H  CHOC2 H.sub.5                                                                             H Cl                                            1.133                                                                             H  H  H  0 H  H  CHOiPr     H Cl                                            1.134                                                                             H  H  H  2 H  H  CHOiPr     H Cl                                            1.135                                                                             H  H  H  0 H  H  C═NOCH.sub.3                                                                          H Cl                                            1.136                                                                             H  H  H  2 H  H  C═NOCH.sub.3                                                                          H Cl                                            1.137                                                                             H  H  H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                            1.138                                                                             H  H  H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                            1.139                                                                             H  H  H  0 H  H  C═NOiPr                                                                               H Cl                                            1.140                                                                             H  H  H  2 H  H  C═NOiPr                                                                               H Cl                                            1.141                                                                             H  H  H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                            1.142                                                                             H  H  H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                            1.143                                                                             H  H  H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                            1.144                                                                             H  H  H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                            1.145                                                                             H  H  H  0 H  H  C(CH.sub.3).sub.2                                                                         H Cl                                            1.146                                                                             H  H  H  2 H  H  C(CH.sub.3).sub.2                                                                         H Cl                                            1.147                                                                             CH.sub.3                                                                          H  H  0 H  H  C═O    H Cl                                            1.148                                                                             CH.sub.3                                                                          H  H  2 H  H  C═O    H Cl                                            1.149                                                                             CH.sub.3                                                                          H  H  0 H  H  CHOCH.sub.3                                                                               H Cl                                            1.150                                                                             CH.sub.3                                                                          H  H  2 H  H  CHOCH.sub.3                                                                               H Cl                                            1.151                                                                             CH.sub.3                                                                          H  H  0 H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                            1.152                                                                             CH.sub.3                                                                          H  H  2 H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                            1.153                                                                             CH.sub.3                                                                          H  H  0 H  H  CHOiPr     H Cl                                            1.154                                                                             CH.sub.3                                                                          H  H  2 H  H  CHOiPr     H Cl                                            1.155                                                                             CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.3                                                                          H Cl                                            1.156                                                                             CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.3                                                                          H Cl                                            1.157                                                                             CH.sub.3                                                                          H  H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                            1158                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                            1.159                                                                             CH.sub.3                                                                          H  H  0 H  H  C═NOiPr                                                                               H Cl                                            1.160                                                                             CH.sub.3                                                                          H  H  2 H  H  C═NOiPr                                                                               H Cl                                            1.161                                                                             CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                            1.162                                                                             CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                            1.163                                                                             CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                            1.164                                                                             CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                            1.165                                                                             CH.sub.3                                                                          H  H  0 H  H  C(CH.sub.3).sub.2                                                                         H Cl                                            1.166                                                                             CH.sub.3                                                                          H  H  2 H  H  C(CH.sub.3).sub.2                                                                         H Cl                                            1.167                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═O    H Cl                                            1.168                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═O    H Cl                                            1.169                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOCH.sub.3                                                                               H Cl                                            1.170                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOCH.sub.3                                                                               H Cl                                            1.171                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                            1.172                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                            1.173                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOiPr     H Cl                                            1.174                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOiPr     H Cl                                            1.175                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.3                                                                          H Cl                                            1.176                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.3                                                                          H Cl                                            1.177                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                            1.178                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                            1.179                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOiPr                                                                               H Cl                                            1.180                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOiPr                                                                               H Cl                                            1.181                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                            1.182                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                            1.183                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                            1.184                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                            1.185                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C(CH.sub.3).sub.2                                                                         H Cl                                            1.186                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C(CH.sub.3).sub.2                                                                         H Cl                                            __________________________________________________________________________

                  TABLE 2                                                          ______________________________________                                         Compounds of the formula                                                        ##STR15##                                                                     The radicals R.sup.12 of X and R.sup.7 of Y form a bond                        No.  R.sup.17                                                                              R.sup.18                                                                               R.sup.19                                                                            n    R.sup.13                                                                            Y       L   M                               ______________________________________                                         2.1  H      H       H    0    H    COCH.sub.3                                                                             H   H                               2.2  H      H       H    2    H    COCH.sub.3                                                                             H   H                               2.3  H      H       H    0    H    COC.sub.2 H.sub.5                                                                      H   H                               2.4  H      H       H    2    H    COC.sub.2 H.sub.5                                                                      H   H                               2.5  H      H       H    0    H    COiPr   H   H                               2.6  H      H       H    2    H    COiPr   H   H                               2.7  CH.sub.3                                                                              H       H    0    H    COCH.sub.3                                                                             H   H                               2.8  CH.sub.3                                                                              H       H    2    H    COCH.sub.3                                                                             H   H                               2.9  CH.sub.3                                                                              H       H    0    H    COC.sub.2 H.sub.5                                                                      H   H                               2.10 CH.sub.3                                                                              H       H    2    H    COC.sub.2 H.sub.5                                                                      H   H                               2.11 CH.sub.3                                                                              H       H    0    H    COiPr   H   H                               2.12 CH.sub.3                                                                              H       H    2    H    COiPr   H   H                               2.13 CH.sub.3                                                                              CH.sub.3                                                                               H    0    H    COCH.sub.3                                                                             H   H                               2.14 CH.sub.3                                                                              CH.sub.3                                                                               H    2    H    COCH.sub.3                                                                             H   H                               2.15 CH.sub.3                                                                              CH.sub.3                                                                               H    0    H    COC.sub.2 H.sub.5                                                                      H   H                               2.16 CH.sub.3                                                                              CH.sub.3                                                                               H    2    H    COC.sub.2 H.sub.5                                                                      H   H                               2.17 CH.sub.3                                                                              CH.sub.3                                                                               H    0    H    COiPr   H   H                               2.18 CH.sub.3                                                                              CH.sub.3                                                                               H    2    H    COiPr   H   H                               2.19 H      H       H    0    H    COCH.sub.3                                                                             H   CH.sub.3                        2.20 H      H       H    2    H    COCH.sub.3                                                                             H   CH.sub.3                        2.21 H      H       H    0    H    COC.sub.2 H.sub.5                                                                      H   CH.sub.3                        2.22 H      H       H    2    H    COC.sub.2 H.sub.5                                                                      H   CH.sub.3                        2.23 H      H       H    0    H    COiPr   H   CH.sub.3                        2.24 H      H       H    2    H    COiPr   H   CH.sub.3                        2.25 CH.sub.3                                                                              H       H    0    H    COCH.sub.3                                                                             H   CH.sub.3                        2.26 CH.sub.3                                                                              H       H    2    H    COCH.sub.3                                                                             H   CH.sub.3                        2.27 CH.sub.3                                                                              H       H    0    H    COC.sub.2 H.sub.5                                                                      H   CH.sub.3                        2.28 CH.sub.3                                                                              H       H    2    H    COC.sub.2 H.sub.5                                                                      H   CH.sub.3                        2.29 CH.sub.3                                                                              H       H    0    H    COiPr   H   CH.sub.3                        2.30 CH.sub.3                                                                              H       H    2    H    COiPr   H   CH.sub.3                        2.31 CH.sub.3                                                                              CH.sub.3                                                                               H    0    H    COCH.sub.3                                                                             H   CH.sub.3                        2.32 CH.sub.3                                                                              CH.sub.3                                                                               H    2    H    COCH.sub.3                                                                             H   CH.sub.3                        2.33 CH.sub.3                                                                              CH.sub.3                                                                               H    0    H    COC.sub.2 H.sub.5                                                                      H   CH.sub.3                        2.34 CH.sub.3                                                                              CH.sub.3                                                                               H    2    H    COC.sub.2 H.sub.5                                                                      H   CH.sub.3                        2.35 CH.sub.3                                                                              CH.sub.3                                                                               H    0    H    COiPr   H   CH.sub.3                        2.36 CH.sub.3                                                                              CH.sub.3                                                                               H    2    H    COiPr   H   CH.sub.3                        2.37 H      H       H    0    H    COCH.sub.3                                                                             H   Cl                              2.38 H      H       H    2    H    COCH.sub.3                                                                             H   Cl                              2.39 H      H       H    0    H    COC.sub.2 H.sub.5                                                                      H   Cl                              2.40 H      H       H    2    H    COC.sub.2 H.sub.5                                                                      H   Cl                              2.41 H      H       H    0    H    COiPr   H   Cl                              2.42 H      H       H    2    H    COiPr   H   Cl                              2.43 CH.sub.3                                                                              H       H    0    H    COCH.sub.3                                                                             H   Cl                              2.44 CH.sub.3                                                                              H       H    2    H    COCH.sub.3                                                                             H   Cl                              2.45 CH.sub.3                                                                              H       H    0    H    COC.sub.2 H.sub.5                                                                      H   Cl                              2.46 CH.sub.3                                                                              H       H    2    H    COC.sub.2 H.sub.5                                                                      H   Cl                              2.47 CH.sub.3                                                                              H       H    0    H    COiPr   H   Cl                              2.48 CH.sub.3                                                                              H       H    2    H    COiPr   H   Cl                              2.49 CH.sub.3                                                                              CH.sub.3                                                                               H    0    H    COCH.sub.3                                                                             H   Cl                              2.50 CH.sub.3                                                                              CH.sub.3                                                                               H    2    H    COCH.sub.3                                                                             H   Cl                              2.51 CH.sub.3                                                                              CH.sub.3                                                                               H    0    H    COC.sub.2 H.sub.5                                                                      H   Cl                              2.52 CH.sub.3                                                                              CH.sub.3                                                                               H    2    H    COC.sub.2 H.sub.5                                                                      H   Cl                              2.53 CH.sub.3                                                                              CH.sub.3                                                                               H    0    H    COiPr   H   Cl                              2.54 CH.sub.3                                                                              CH.sub.3                                                                               H    2    H    COiPr   H   Cl                              ______________________________________                                    

                                      TABLE 3                                      __________________________________________________________________________     Compounds of the formula                                                        ##STR16##                                                                     No.                                                                               R.sup.17                                                                          R.sup.18                                                                          R.sup.19                                                                          n R.sup.12                                                                          R.sup.13                                                                          Y          L  M                                            __________________________________________________________________________     3.1                                                                               H  H  H  0 H  H  C═O    CH.sub.3                                                                          H                                            3.2                                                                               H  H  H  2 H  H  C═O    CH.sub.3                                                                          H                                            3.3                                                                               H  H  H  0 H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.4                                                                               H  H  H  2 H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.5                                                                               H  H  H  0 H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.6                                                                               H  H  H  2 H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.7                                                                               H  H  H  0 H  H  CHOiPr     CH.sub.3                                                                          H                                            3.8                                                                               H  H  H  2 H  H  CHOiPr     CH.sub.3                                                                          H                                            3.9                                                                               H  H  H  0 H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.10                                                                              H  H  H  2 H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.11                                                                              H  H  H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.12                                                                              H  H  H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.13                                                                              H  H  H  D H  H  C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.14                                                                              H  H  H  2 H  H  C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.15                                                                              H  H  H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.16                                                                              H  H  H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.17                                                                              H  H  H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.18                                                                              H  H  H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.19                                                                              H  H  H  0 H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.20                                                                              H  H  H  2 H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.21                                                                              CH.sub.3                                                                          H  H  0 H  H  C═O    CH.sub.3                                                                          H                                            3.22                                                                              CH.sub.3                                                                          H  H  2 H  H  C═O    CH.sub.3                                                                          H                                            3.23                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.24                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.25                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.26                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.27                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOiPr     CH.sub.3                                                                          H                                            3.28                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOiPr     CH.sub.3                                                                          H                                            3.29                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.30                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.31                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.32                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.33                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.34                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.35                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.36                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.37                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.38                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.39                                                                              CH.sub.3                                                                          H  H  0 H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.40                                                                              CH.sub.3                                                                          H  H  2 H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.41                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═O    CH.sub.3                                                                          H                                            3.42                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═O    CH.sub.3                                                                          H                                            3.43                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.44                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.45                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.46                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.47                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOiPr     CH.sub.3                                                                          H                                            3.48                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOiPr     CH.sub.3                                                                          H                                            3.49                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.50                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.51                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.52                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.53                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.54                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.55                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.56                                                                              CH.sub.3                                                                          CH.sub.3                                                                          W  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.57                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.58                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.59                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.60                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.61                                                                              H  H  H  0 H  H  C═O    Cl H                                            3.62                                                                              H  H  H  2 H  H  C═O    Cl H                                            3.63                                                                              H  H  H  0 H  H  CHOCH.sub.3                                                                               Cl H                                            3.64                                                                              H  H  H  2 H  H  CHOCH.sub.3                                                                               Cl H                                            3.65                                                                              H  H  H  0 H  H  CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.66                                                                              H  H  H  2 H  H  CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.67                                                                              H  H  H  0 H  H  CHOiPr     Cl H                                            3.68                                                                              H  H  H  2 H  H  CHOiPr     Cl H                                            3.69                                                                              H  H  H  0 H  H  C═NOCH.sub.3                                                                          Cl H                                            3.70                                                                              H  H  H  2 H  H  C═NOCH.sub.3                                                                          Cl H                                            3.71                                                                              H  H  H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.72                                                                              H  H  H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.73                                                                              H  H  H  0 H  H  C═NOiPr                                                                               Cl H                                            3.74                                                                              H  H  H  2 H  H  C═NOiPr                                                                               Cl H                                            3.75                                                                              H  H  H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.76                                                                              H  H  H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3 77                                                                              H  H  H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.78                                                                              H  H  H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.79                                                                              H  H  H  0 H  H  C(CH.sub.3).sub.2                                                                         Cl H                                            3.80                                                                              H  H  H  2 H  H  C(CH.sub.3).sub.2                                                                         Cl H                                            3.81                                                                              CH.sub.3                                                                          H  H  0 H  H  C═O    Cl H                                            3.82                                                                              CH.sub.3                                                                          H  H  2 H  H  C═O    Cl H                                            3.83                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOCH.sub.3                                                                               Cl H                                            3.84                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOCH.sub.3                                                                               Cl H                                            3.85                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.86                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.87                                                                              CH.sub.3                                                                          H  H  0 H  H  CHOiPr     Cl H                                            3.88                                                                              CH.sub.3                                                                          H  H  2 H  H  CHOiPr     Cl H                                            3.89                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.3                                                                          Cl H                                            3.90                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.3                                                                          Cl H                                            3.91                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.92                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.93                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOiPr                                                                               Cl H                                            3.94                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOiPr                                                                               Cl H                                            3.95                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.96                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.97                                                                              CH.sub.3                                                                          H  H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.98                                                                              CH.sub.3                                                                          H  H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.99                                                                              CH.sub.3                                                                          H  H  0 H  H  C(CH.sub.3).sub.2                                                                         Cl H                                            3.100                                                                             CH.sub.3                                                                          H  H  2 H  H  C(CH.sub.3).sub.2                                                                         Cl H                                            3.101                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═O    Cl H                                            3.102                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═O    Cl H                                            3.103                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOCH.sub.3                                                                               Cl H                                            3.104                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOCH.sub.3                                                                               Cl H                                            3.105                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.106                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.107                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  CHOiPr     Cl H                                            3.108                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  CHOiPr     Cl H                                            3.109                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═N--OCH.sub.3                                                                        Cl H                                            3.110                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.3                                                                          Cl H                                            3.111                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.112                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.113                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOiPr                                                                               Cl H                                            3.114                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOiPr                                                                               Cl H                                            3.115                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.116                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.117                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.118                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.119                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  C(CH.sub.3).sub.2                                                                         Cl H                                            3.120                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  C(CH.sub.3).sub.2                                                                         Cl H                                            3.121                                                                             H  H  H  0 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          H                                            3.122                                                                             H  H  H  2 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          H                                            3.123                                                                             H  H  H  0 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.124                                                                             H  H  H  2 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.125                                                                             H  H  H  0 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.126                                                                             H  H  H  2 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.127                                                                             H  H  H  0 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          H                                            3.128                                                                             H  H  H  2 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          H                                            3.129                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.130                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.131                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.132                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.133                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.134                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.135                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.136                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.137                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.138                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.139                                                                             H  H  H  0 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.140                                                                             H  H  H  2 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.141                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          H                                            3.142                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          H                                            3.143                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.144                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.145                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.146                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.147                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          H                                            3.148                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          H                                            3.149                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.150                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.151                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.152                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.153                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.154                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.155                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.156                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.157                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.158                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.159                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.160                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.161                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          H                                            3.162                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          H                                            3.163                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.164                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          H                                            3.165                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.166                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          H                                            3.167                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          H                                            3.168                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          H                                            3.169                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.170                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          H                                            3.171                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.172                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          H                                            3.173                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.174                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          H                                            3.175                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.176                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          H                                            3.177                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.178                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          H                                            3.179                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.180                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          H                                            3.181                                                                             H  H  H  0 H  CH.sub.3                                                                          C═O    Cl H                                            3.182                                                                             H  H  H  2 H  CH.sub.3                                                                          C═O    Cl H                                            3.183                                                                             H  H  H  0 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               Cl H                                            3.184                                                                             H  H  H  2 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               Cl H                                            3.185                                                                             H  H  H  0 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.186                                                                             H  H  H  2 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.187                                                                             H  H  H  0 H  CH.sub.3                                                                          CHOiPr     Cl H                                            3.188                                                                             H  H  H  2 H  CH.sub.3                                                                          CHOiPr     Cl H                                            3.189                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          Cl H                                            3.190                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          Cl H                                            3.191                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.192                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.193                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOiPr                                                                               Cl H                                            3.194                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOiPr                                                                               Cl H                                            3.195                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.196                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.197                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.198                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.199                                                                             H  H  H  0 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         Cl H                                            3.200                                                                             H  H  H  2 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         Cl H                                            3.201                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═O    Cl H                                            3.202                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═O    Cl H                                            3.203                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               Cl H                                            3.204                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               Cl H                                            3.205                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.206                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.207                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          CHOiPr     Cl H                                            3.208                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          CHOiPr     Cl H                                            3.209                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          Cl H                                            3.210                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          Cl H                                            3.211                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.212                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.213                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOiPr                                                                               Cl H                                            3.214                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOiPr                                                                               Cl H                                            3.215                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.216                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.217                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.218                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.219                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         Cl H                                            3.220                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         Cl H                                            3.221                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═O    Cl H                                            3.222                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═O    Cl H                                            3.223                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               Cl H                                            3.224                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               Cl H                                            3.225                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.226                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        Cl H                                            3.227                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          CHOiPr     Cl H                                            3.228                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          CHOiPr     Cl H                                            3.229                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          Cl H                                            3.230                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          Cl H                                            3.231                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.232                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   Cl H                                            3.233                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOiPr                                                                               Cl H                                            3.234                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOiPr                                                                               Cl H                                            3.235                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.236                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              Cl H                                            3.237                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.238                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl H                                            3.239                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          (CH.sub.3).sub.2                                                                          Cl H                                            3.240                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         Cl H                                            3.241                                                                             H  H  H  0 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          CH.sub.3                                     3.242                                                                             H  H  H  2 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          CH.sub.3                                     3.243                                                                             H  H  H  0 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                                     3.244                                                                             H  H  H  2 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                                     3.245                                                                             H  H  H  0 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                                     3.246                                                                             H  H  H  2 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                                     3.247                                                                             H  H  H  0 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          CH.sub.3                                     3.248                                                                             H  H  H  2 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          CH.sub.3                                     3.249                                                                             H  H  H  0 H  CH.sub.3                                                                          COCH.sub.3 CH.sub.3                                                                          CH.sub.3                                     3.250                                                                             H  H  H  2 H  CH.sub.3                                                                          COCH.sub.3 CH.sub.3                                                                          CH.sub.3                                     3.251                                                                             H  H  H  0 H  CH.sub.3                                                                          COC.sub.2 H.sub.5                                                                         CH.sub.3                                                                          CH.sub.3                                     3.252                                                                             H  H  H  2 H  CH.sub.3                                                                          COC.sub.2 H.sub.5                                                                         CH.sub.3                                                                          CH.sub.3                                     3.253                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                                     3.254                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                                     3.255                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                                     3.256                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                                     3.257                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                                     3.258                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                                     3.259                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                                     3.260                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                                     3.261                                                                             H  H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                                     3.262                                                                             H  H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                                     3.263                                                                             H  H  H  0 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                                     3.264                                                                             H  H  H  2 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                                     3.265                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          CH.sub.3                                     3.266                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          CH.sub.3                                     3.267                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                                     3.268                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                                     3.269                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                                     3.270                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                                     3.271                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          CH.sub.3                                     3.272                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          CH.sub.3                                     3.273                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                                     3.274                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                                     3.275                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                                     3.276                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                                     3.277                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                                     3.278                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                                     3.279                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                                     3.280                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                                     3.281                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                                     3.282                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                                     3.283                                                                             CH.sub.3                                                                          H  H  0 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                                     3.284                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                                     3.285                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          CH.sub.3                                     3.286                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═O    CH.sub.3                                                                          CH.sub.3                                     3.287                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                                     3.288                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                                     3.289                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                                     3.290                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                                     3.291                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          CH.sub.3                                     3.292                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          CHOiPr     CH.sub.3                                                                          CH.sub.3                                     3.293                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                                     3.294                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                                     3.295                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                                     3.296                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                                     3.297                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                                     3.298                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                                     3.299                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                                     3.300                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                                     3.301                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                                     3.302                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                                     3.303                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                                     3.304                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                          C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                                     __________________________________________________________________________

                                      TABLE 4                                      __________________________________________________________________________     Compounds of the formula                                                        ##STR17##                                                                     No. R.sup.17                                                                          R.sup.18                                                                           R.sup.19                                                                          n R.sup.12                                                                          R.sup.13                                                                          R.sup.21                                                                          R.sup.22                                                                          Y          L  M                                    __________________________________________________________________________     4.1 H  H   H  0 H  H  H  H  C═O    H  H                                    4.2 H  H   H  1 H  H  H  H  C═O    H  H                                    4.3 H  H   H  2 H  H  H  H  C═O    H  H                                    4.4 H  H   H  0 H  H  H  H  CHOH       H  H                                    4.5 H  H   H  1 H  H  H  H  CHOH       H  H                                    4.6 H  H   H  2 H  H  H  H  CHOH       H  H                                    4.7 H  H   H  0 H  H  H  H  CHOCH.sub.3                                                                               H  H                                    4.8 H  H   H  1 H  H  H  H  CHOCH.sub.3                                                                               H  H                                    4.9 H  H   H  2 H  H  H  H  CHOCH.sub.3                                                                               H  H                                    4.10                                                                               H  H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  H                                    4.11                                                                               H  H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  H                                    4.12                                                                               H  H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  H                                    4.13                                                                               H  H   H  0 H  H  H  H  CHOiPr     H  H                                    4.14                                                                               H  H   H  1 H  H  H  H  CHOiPr     H  H                                    4.15                                                                               H  H   H  2 H  H  H  H  CHOiPr     H  H                                    4.16                                                                               H  H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  H                                    4.17                                                                               H  H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  H                                    4.18                                                                               H  H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  H                                    4.19                                                                               H  H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  H                                    4.20                                                                               H  H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  H                                    4.21                                                                               H  H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  H                                    4.22                                                                               H  H   H  0 H  H  H  H  C═NOiPr                                                                               H  H                                    4.23                                                                               H  H   H  1 H  H  H  H  C═NOiPr                                                                               H  H                                    4.24                                                                               H  H   H  2 H  H  H  H  C═NOiPr                                                                               H  H                                    4.25                                                                               H  H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  H                                    4.26                                                                               H  H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  H                                    4.27                                                                               H  H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  H                                    4.28                                                                               H  H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  H                                    4.29                                                                               H  H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  H                                    4.30                                                                               H  H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  H                                    4.31                                                                               H  H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  H                                    4.32                                                                               H  H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  H                                    4.33                                                                               H  H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  H                                    4.34                                                                               H  H   H  0 H  H  H  H                                                                                  ##STR18## H  H                                    4.35                                                                               H  H   H  1 H  H  H  H                                                                                  ##STR19## H  H                                    4.36                                                                               H  H   H  2 H  H  H  H                                                                                  ##STR20## H  H                                    4.37                                                                               H  H   H  0 H  H  H  H                                                                                  ##STR21## H  H                                    4.38                                                                               H  H   H  1 H  H  H  H                                                                                  ##STR22## H  H                                    4.39                                                                               H  H   H  2 H  H  H  H                                                                                  ##STR23## H  H                                    4.40                                                                               H  H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  H                                    4.41                                                                               H  H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  H                                    4.42                                                                               H  H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  H                                    4.43                                                                               H  H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  H                                    4.44                                                                               H  H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  H                                    4.45                                                                               H  H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  H                                    4.46                                                                               H  H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  H                                    4.47                                                                               H  H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  H                                    4.48                                                                               H  H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  H                                    4.49                                                                               H  H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  H                                    4.50                                                                               H  H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  H                                    4.51                                                                               H  H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  H                                    4.52                                                                               H  H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  H                                    4.53                                                                               H  H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  H                                    4.54                                                                               H  H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  H                                    4.55                                                                               H  H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  H                                    4.56                                                                               H  H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  H                                    4.57                                                                               H  H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  H                                    4.58                                                                               H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  H                                    4.59                                                                               H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  H                                    4.60                                                                               H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  H                                    4.61                                                                               H  H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  H                                    4.62                                                                               H  H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  H                                    4.63                                                                               H  H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  H                                    4.64                                                                               H  H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  H                                    4.65                                                                               H  H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  H                                    4.66                                                                               H  H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  H                                    4.67                                                                               H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  H                                    4.68                                                                               H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  H                                    4.69                                                                               H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  H                                    4.70                                                                               H  H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  H                                    4.71                                                                               H  H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  H                                    4.72                                                                               H  H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  H                                    4.73                                                                               H  H   H  0 H  H  H  H  O          H  H                                    4.74                                                                               H  H   H  1 H  H  H  H  O          H  H                                    4.75                                                                               H  H   H  2 H  H  H  H  O          H  H                                    4.76                                                                               CH.sub.3                                                                          H   H  0 H  H  H  H  C═O    H  H                                    4.77                                                                               CH.sub.3                                                                          H   H  1 H  H  H  H  C═O    H  H                                    4.78                                                                               CH.sub.3                                                                          H   H  2 H  H  H  H  C═O    H  H                                    4.79                                                                               CH.sub.3                                                                          H   H  0 H  H  H  H  CHOH       H  H                                    4.80                                                                               CH.sub.3                                                                          H   H  1 H  H  H  H  CHOH       H  H                                    4.81                                                                               CH.sub.3                                                                          H   H  2 H  H  H  H  CHOH       H  H                                    4.82                                                                               CH.sub.3                                                                          H   H  0 H  H  H  H  CHOCH.sub.3                                                                               H  H                                    4.83                                                                               CH.sub.3                                                                          H   H  1 H  H  H  H  CHOCH.sub.3                                                                               H  H                                    4.84                                                                               CH.sub.3                                                                          H   H  2 H  H  H  H  CHOCH.sub.3                                                                               H  H                                    4.85                                                                               CH.sub.3                                                                          H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  H                                    4.86                                                                               CH.sub.3                                                                          H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  H                                    4.87                                                                               CH.sub.3                                                                          H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  H                                    4.88                                                                               CH.sub.3                                                                          H   H  0 H  H  H  H  CHOiPr     H  H                                    4.89                                                                               CH.sub.3                                                                          H   H  1 H  H  H  H  CHOiPr     H  H                                    4.90                                                                               CH.sub.3                                                                          H   H  2 H  H  H  H  CHOiPr     H  H                                    4.91                                                                               CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  H                                    4.92                                                                               CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  H                                    4.93                                                                               CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  H                                    4.94                                                                               CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  H                                    4.95                                                                               CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  H                                    4.96                                                                               CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  H                                    4.97                                                                               CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOiPr                                                                               H  H                                    4.98                                                                               CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOiPr                                                                               H  H                                    4.99                                                                               CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOiPr                                                                               H  H                                    4.100                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  H                                    4.101                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  H                                    4.102                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  H                                    4.103                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  H                                    4.104                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  H                                    4.105                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  H                                    4.106                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  H                                    4.107                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  H                                    4.108                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  H                                    4.109                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR24## H  H                                    4.110                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR25## H  H                                    4.111                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR26## H  H                                    4.112                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR27## H  H                                    4.113                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR28## H  H                                    4.114                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR29## H  H                                    4.115                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  H                                    4.116                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  H                                    4.117                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  H                                    4.118                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  H                                    4.119                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  H                                    4.120                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  H                                    4.121                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  H                                    4.122                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  H                                    4.123                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  H                                    4.124                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  H                                    4.125                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  H                                    4.126                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  H                                    4.127                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  H                                    4.128                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  H                                    4.129                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  H                                    4.130                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  H                                    4.131                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  H                                    4.132                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  H                                    4.133                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  H                                    4.134                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  H                                    4.135                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  H                                    4.136                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  H                                    4.137                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  H                                    4.138                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  H                                    4.139                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  H                                    4.140                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  H                                    4.141                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  H                                    4.142                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  H                                    4.143                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  H                                    4.144                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  H                                    4.145                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  H                                    4.146                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  H                                    4.147                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  H                                    4.148                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  O          H  H                                    4.149                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  O          H  H                                    4.150                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  O          H  H                                    4.151                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═O    H  H                                    4.152                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═O    H  H                                    4.153                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═O    H  H                                    4.154                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOH       H  H                                    4.155                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOH       H  H                                    4.156                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOH       H  H                                    4.157                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOCH.sub.3                                                                               H  H                                    4.158                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOCH.sub.3                                                                               H  H                                    4.159                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOCH.sub.3                                                                               H  H                                    4.160                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  H                                    4.161                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  H                                    4.162                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  H                                    4.163                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOiPr     H  H                                    4.164                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOiPr     H  H                                    4.165                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOiPr     H  H                                    4.166                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  H                                    4.167                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  H                                    4.168                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  H                                    4.169                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  H                                    4.170                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  H                                    4.171                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  H                                    4.172                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOiPr                                                                               H  H                                    4.173                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOiPr                                                                               H  H                                    4.174                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOiPr                                                                               H  H                                    4.175                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  H                                    4.176                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  H                                    4.177                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  H                                    4.178                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  H                                    4.179                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  H                                    4.180                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  H                                    4.181                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  H                                    4.182                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  H                                    4.183                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  H                                    4.184                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR30## H  H                                    4.185                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR31## H  H                                    4.186                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR32## H  H                                    4.187                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR33## H  H                                    4.188                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR34## H  H                                    4.189                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR35## H  H                                    4.190                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  H                                    4.191                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  H                                    4.192                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  H                                    4.193                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  H                                    4.194                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  H                                    4.195                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  H                                    4.196                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  H                                    4.197                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  H                                    4.198                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  H                                    4.199                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  H                                    4.200                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  H                                    4.201                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  H                                    4.202                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  H                                    4.203                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  H                                    4.204                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  H                                    4.205                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  H                                    4.206                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  H                                    4.207                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  H                                    4.208                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  H                                    4.209                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  H                                    4.210                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  H                                    4.211                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  H                                    4.212                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  H                                    4.213                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  H                                    4.214                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  H                                    4.215                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  H                                    4.216                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  H                                    4.217                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  H                                    4.218                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  H                                    4.219                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  H                                    4.220                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  H                                    4.221                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  H                                    4.222                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  H                                    4.223                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  O          H  H                                    4.224                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  O          H  H                                    4.225                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  O          H  H                                    4.226                                                                              H  H   H  0 H  H  H  H  C═O    H  CH.sub.3                             4.227                                                                              H  H   H  1 H  H  H  H  C═O    H  CH.sub.3                             4.228                                                                              H  H   H  2 H  H  H  H  C═O    H  CH.sub.3                             4.229                                                                              H  H   H  0 H  H  H  H  CHOH       H  CH.sub.3                             4.230                                                                              H  H   H  1 H  H  H  H  CHOH       H  CH.sub.3                             4.231                                                                              H  H   H  2 H  H  H  H  CHOH       H  CH.sub.3                             4.232                                                                              H  H   H  0 H  H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.233                                                                              H  H   H  1 H  H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.234                                                                              H  H   H  2 H  H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.235                                                                              H  H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.236                                                                              H  H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.237                                                                              H  H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.238                                                                              H  H   H  0 H  H  H  H  CHOiPr     H  CH.sub.3                             4.239                                                                              H  H   H  1 H  H  H  H  CHOiPr     H  CH.sub.3                             4.240                                                                              H  H   H  2 H  H  H  H  CHOiPr     H  CH.sub.3                             4.241                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.242                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.243                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.244                                                                              H  H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.245                                                                              H  H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.246                                                                              H  H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.247                                                                              H  H   H  0 H  H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.248                                                                              H  H   H  1 H  H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.249                                                                              H  H   H  2 H  H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.250                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.251                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.252                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.253                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.254                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.255                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.256                                                                              H  H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.257                                                                              H  H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.258                                                                              H  H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.259                                                                              H  H   H  0 H  H  H  H                                                                                  ##STR36## H  CH.sub.3                             4.260                                                                              H  H   H  1 H  H  H  H                                                                                  ##STR37## H  CH.sub.3                             4.261                                                                              H  H   H  2 H  H  H  H                                                                                  ##STR38## H  CH.sub.3                             4.262                                                                              H  H   H  0 H  H  H  H                                                                                  ##STR39## H  CH.sub.3                             4.263                                                                              H  H   H  1 H  H  H  H                                                                                  ##STR40## H  CH.sub.3                             4.264                                                                              H  H   H  2 H  H  H  H                                                                                  ##STR41## H  CH.sub.3                             4.265                                                                              H  H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.266                                                                              H  H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.267                                                                              H  H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.268                                                                              H  H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.269                                                                              H  H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.270                                                                              H  H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.271                                                                              H  H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.272                                                                              H  H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.273                                                                              H  H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.274                                                                              H  H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.275                                                                              H  H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.276                                                                              H  H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.277                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.278                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.279                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.280                                                                              H  H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.281                                                                              H  H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.282                                                                              H  H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.283                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.284                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.285                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.286                                                                              H  H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.287                                                                              H  H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.288                                                                              H  H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.289                                                                              H  H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.290                                                                              H  H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.291                                                                              H  H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.292                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.293                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.294                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.295                                                                              H  H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.296                                                                              H  H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.297                                                                              H  H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.298                                                                              H  H   H  0 H  H  H  H  O          H  CH.sub.3                             4.299                                                                              H  H   H  1 H  H  H  H  O          H  CH.sub.3                             4.300                                                                              H  H   H  2 H  H  H  H  O          H  CH.sub.3                             4.301                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═O    H  CH.sub.3                             4.302                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═O    H  CH.sub.3                             4.303                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═O    H  CH.sub.3                             4.304                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOH       H  CH.sub.3                             4.305                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOH       H  CH.sub.3                             4.306                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOH       H  CH.sub.3                             4.307                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.308                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.309                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.310                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.311                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.312                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.313                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOiPr     H  CH.sub.3                             4.314                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOiPr     H  CH.sub.3                             4.315                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOiPr     H  CH.sub.3                             4.316                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.317                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.318                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.319                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.320                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.321                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.322                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.323                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.324                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.325                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.326                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.327                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.328                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.329                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.330                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.331                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.332                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.333                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.334                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR42## H  CH.sub.3                             4.335                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR43## H  CH.sub.3                             4.336                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR44## H  CH.sub.3                             4.337                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR45## H  CH.sub.3                             4.338                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR46## H  CH.sub.3                             4.339                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR47## H  CH.sub.3                             4.340                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.341                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.342                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.343                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.344                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.345                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.346                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.347                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.348                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.349                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.350                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.351                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.352                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.353                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.354                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.355                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.356                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.357                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.358                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.359                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.360                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.361                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.362                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.363                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.364                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.365                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.366                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.367                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.368                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.369                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.370                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.371                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.372                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.373                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  O          H  CH.sub.3                             4.374                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  O          H  CH.sub.3                             4.375                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  O          H  CH.sub.3                             4.376                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═O    H  CH.sub.3                             4.377                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═O    H  CH.sub.3                             4.378                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═O    H  CH.sub.3                             4.379                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOH       H  CH.sub.3                             4.380                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOH       H  CH.sub.3                             4.381                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOH       H  CH.sub.3                             4.382                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.383                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.384                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.385                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.386                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.387                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.388                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOiPr     H  CH.sub.3                             4.389                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOiPr     H  CH.sub.3                             4.390                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOiPr     H  CH.sub.3                             4.391                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.392                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.393                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.394                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.395                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.396                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.397                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.398                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.399                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.400                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.401                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.402                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.403                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.404                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.405                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.406                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.407                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.408                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.409                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR48## H  CH.sub.3                             4.410                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR49## H  CH.sub.3                             4.411                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR50## H  CH.sub.3                             4.412                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR51## H  CH.sub.3                             4.413                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR52## H  CH.sub.3                             4.414                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR53## H  CH.sub.3                             4.415                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.416                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.417                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.418                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.419                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.420                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.421                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.422                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.423                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.424                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.425                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.426                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.427                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.428                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.429                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.430                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.431                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.432                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.433                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.434                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.435                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.436                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.437                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.438                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.439                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.440                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.441                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.442                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.443                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.444                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.445                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.446                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.447                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.448                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  O          H  CH.sub.3                             4.449                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  O          H  CH.sub.3                             4.450                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  O          H  CH.sub.3                             4.451                                                                              H  H   H  0 H  H  H  H  C═O    H  Cl                                   4.452                                                                              H  H   H  1 H  H  H  H  C═O    H  Cl                                   4.453                                                                              H  H   H  2 H  H  H  H  C═O    H  Cl                                   4.454                                                                              H  H   H  0 H  H  H  H  CHOH       H  Cl                                   4.455                                                                              H  H   H  1 H  H  H  H  CHOH       H  Cl                                   4.456                                                                              H  H   H  2 H  H  H  H  CHOH       H  Cl                                   4.457                                                                              H  H   H  0 H  H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.458                                                                              H  H   H  1 H  H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.459                                                                              H  H   H  2 H  H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.460                                                                              H  H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.461                                                                              H  H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.462                                                                              H  H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.463                                                                              H  H   H  0 H  H  H  H  CHOiPr     H  Cl                                   4.464                                                                              H  H   H  1 H  H  H  H  CHOiPr     H  Cl                                   4.465                                                                              H  H   H  2 H  H  H  H  CHOiPr     H  Cl                                   4.466                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.467                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.468                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.469                                                                              H  H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.470                                                                              H  H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.471                                                                              H  H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.472                                                                              H  H   H  0 H  H  H  H  C═NOiPr                                                                               H  Cl                                   4.473                                                                              H  H   H  1 H  H  H  H  C═NOiPr                                                                               H  Cl                                   4.474                                                                              H  H   H  2 H  H  H  H  C═NOiPr                                                                               H  Cl                                   4.475                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.476                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.477                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.478                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.479                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.480                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.481                                                                              H  H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.482                                                                              H  H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.483                                                                              H  H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.484                                                                              H  H   H  0 H  H  H  H                                                                                  ##STR54## H  Cl                                   4.485                                                                              H  H   H  1 H  H  H  H                                                                                  ##STR55## H  Cl                                   4.486                                                                              H  H   H  2 H  H  H  H                                                                                  ##STR56## H  Cl                                   4.487                                                                              H  H   H  0 H  H  H  H                                                                                  ##STR57## H  Cl                                   4.488                                                                              H  H   H  1 H  H  H  H                                                                                  ##STR58## H  Cl                                   4.489                                                                              H  H   H  2 H  H  H  H                                                                                  ##STR59## H  Cl                                   4.490                                                                              H  H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.491                                                                              H  H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.492                                                                              H  H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.493                                                                              H  H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.494                                                                              H  H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.495                                                                              H  H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.496                                                                              H  H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.497                                                                              H  H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.498                                                                              H  H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.499                                                                              H  H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.500                                                                              H  H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.501                                                                              H  H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.502                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.503                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.504                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.505                                                                              H  H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.506                                                                              H  H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.507                                                                              H  H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.508                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.509                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.510                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.511                                                                              H  H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.512                                                                              H  H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.513                                                                              H  H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.514                                                                              H  H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.515                                                                              H  H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.516                                                                              H  H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.517                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.518                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.519                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.520                                                                              H  H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.521                                                                              H  H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.522                                                                              H  H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.523                                                                              H  H   H  0 H  H  H  H  O          H  Cl                                   4.524                                                                              H  H   H  1 H  H  H  H  O          H  Cl                                   4.525                                                                              H  H   H  2 H  H  H  H  O          H  Cl                                   4.526                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═O    H  Cl                                   4.527                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═O    H  Cl                                   4.528                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═O    H  Cl                                   4.529                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOH       H  Cl                                   4.530                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOH       H  Cl                                   4.531                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOH       H  Cl                                   4.532                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.533                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.534                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.535                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.536                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.537                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.538                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOiPr     H  Cl                                   4.539                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOiPr     H  Cl                                   4.540                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOiPr     H  Cl                                   4.541                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.542                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.543                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.544                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.545                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.546                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.547                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOiPr                                                                               H  Cl                                   4.548                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOiPr                                                                               H  Cl                                   4.549                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOiPr                                                                               H  Cl                                   4.550                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.551                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.552                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.553                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.554                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.555                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.556                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.557                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.558                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.559                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR60## H  Cl                                   4.560                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR61## H  Cl                                   4.561                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR62## H  Cl                                   4.562                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR63## H  Cl                                   4.563                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR64## H  Cl                                   4.564                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR65## H  Cl                                   4.565                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.566                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.567                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.568                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.569                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.570                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.571                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.572                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.573                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.574                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.575                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.576                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.577                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.578                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.579                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.580                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.581                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.582                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.583                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.584                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.585                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.586                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.587                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.588                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.589                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.590                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.591                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.592                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.593                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.594                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.595                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.596                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.597                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.598                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  O          H  Cl                                   4.599                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  O          H  Cl                                   4.600                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  O          H  Cl                                   4.601                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═O    H  Cl                                   4.602                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═O    H  Cl                                   4.603                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═O    H  Cl                                   4.604                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOH       H  Cl                                   4.605                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOH       H  Cl                                   4.606                                                                              CH.sub.3                                                                          CH.sub.3 C                                                                         H  2 H  H  H  H  CHOH       H  Cl                                   4.607                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.608                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.609                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.610                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.611                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.612                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.613                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOiPr     H  Cl                                   4.614                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOiPr     H  Cl                                   4.615                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOiPr     H  Cl                                   4.616                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.617                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.618                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.619                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.620                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.621                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.622                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOiPr                                                                               H  Cl                                   4.623                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOiPr                                                                               H  Cl                                   4.624                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOiPr                                                                               H  Cl                                   4.625                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.626                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.627                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.628                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.629                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.630                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.631                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.632                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.633                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.634                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR66## H  Cl                                   4.635                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR67## H  Cl                                   4.636                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR68## H  Cl                                   4.637                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR69## H  Cl                                   4.638                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR70## H  Cl                                   4.639                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR71## H  Cl                                   4.640                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.641                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.642                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.643                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.644                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.645                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.646                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.647                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.648                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.649                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.650                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.651                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.652                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.653                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.654                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.655                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.656                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.657                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.658                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.659                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.660                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.661                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.662                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.663                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.664                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.665                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.666                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.667                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.668                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.669                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.670                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.671                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.672                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.673                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  O          H  Cl                                   4.674                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  O          H  Cl                                   4.675                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  O          H  Cl                                   4.676                                                                              H  H   H  0 H  H  H  H  C═O    H  NO.sub.2                             4.677                                                                              H  H   H  1 H  H  H  H  C═O    H  NO.sub.2                             4.678                                                                              H  H   H  2 H  H  H  H  C═O    H  NO.sub.2                             4.679                                                                              H  H   H  0 H  H  H  H  CHOCH.sub.3                                                                               H  NO.sub.2                             4.680                                                                              H  H   H  1 H  H  H  H  CHOCH.sub.3                                                                               H  NO.sub.2                             4.681                                                                              H  H   H  2 H  H  H  H  CHOCH.sub.3                                                                               H  NO.sub.2                             4.682                                                                              H  H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  NO.sub.2                             4.683                                                                              H  H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  NO.sub.2                             4.684                                                                              H  H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  NO.sub.2                             4.685                                                                              H  H   H  0 H  H  H  H  CHOiPr     H  NO.sub.2                             4.686                                                                              H  H   H  1 H  H  H  H  CHOiPr     H  NO.sub.2                             4.687                                                                              H  H   H  2 H  H  H  H  CHOiPr     H  NO.sub.2                             4.688                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  NO.sub.2                             4.689                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  NO.sub.2                             4.690                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  NO.sub.2                             4.691                                                                              H  H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  NO.sub.2                             4.692                                                                              H  H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  NO.sub.2                             4.693                                                                              H  H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  NO.sub.2                             4.694                                                                              H  H   H  0 H  H  H  H  C═NOiPr                                                                               H  NO.sub.2                             4.695                                                                              H  H   H  1 H  H  H  H  C═NOiPr                                                                               H  NO.sub.2                             4.696                                                                              H  H   H  2 H  H  H  H  C═NOiPr                                                                               H  NO.sub.2                             4.697                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  NO.sub.2                             4.698                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  NO.sub.2                             4.699                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  NO.sub.2                             4.700                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  NO.sub.2                             4.701                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  NO.sub.2                             4.702                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  NO.sub.2                             4.703                                                                              H  H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  NO.sub.2                             4.704                                                                              H  H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  NO.sub.2                             4.705                                                                              H  H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  NO.sub.2                             4.706                                                                              H  H   H  0 H  H  H  H                                                                                  ##STR72## H  NO.sub.2                             4.707                                                                              H  H   H  1 H  H  H  H                                                                                  ##STR73## H  NO.sub.2                             4.708                                                                              H  H   H  2 H  H  H  H                                                                                  ##STR74## H  NO.sub.2                             4.709                                                                              H  H   H  0 H  H  H  H                                                                                  ##STR75## H  NO.sub.2                             4.710                                                                              H  H   H  1 H  H  H  H                                                                                  ##STR76## H  NO.sub.2                             4.711                                                                              H  H   H  2 H  H  H  H                                                                                  ##STR77## H  NO.sub.2                             4.712                                                                              H  H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  NO.sub.2                             4.713                                                                              H  H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  NO.sub.2                             4.714                                                                              H  H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  NO.sub.2                             4.715                                                                              H  H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.716                                                                              H  H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.717                                                                              H  H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.718                                                                              H  H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  NO.sub.2                             4.719                                                                              H  H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  NO.sub.2                             4.720                                                                              H  H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  NO.sub.2                             4.721                                                                              H  H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  NO.sub.2                             4.722                                                                              H  H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  NO.sub.2                             4.723                                                                              H  H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  NO.sub.2                             4.724                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  NO.sub.2                             4.725                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  NO.sub.2                             4.726                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  NO.sub.2                             4.727                                                                              H  H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.728                                                                              H  H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.729                                                                              H  H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.730                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  NO.sub.2                             4.731                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  NO.sub.2                             4.732                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  NO.sub.2                             4.733                                                                              H  H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  NO.sub.2                             4.734                                                                              H  H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  NO.sub.2                             4.735                                                                              H  H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  NO.sub.2                             4.736                                                                              H  H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  NO.sub.2                             4.737                                                                              H  H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  NO.sub.2                             4.738                                                                              H  H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  NO.sub.2                             4.739                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  NO.sub.2                             4.740                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  NO.sub.2                             4.741                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  NO.sub.2                             4.742                                                                              H  H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  NO.sub.2                             4.743                                                                              H  H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  NO.sub.2                             4.744                                                                              H  H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  NO.sub.2                             4.745                                                                              H  H   H  0 H  H  H  H  O          H  NO.sub.2                             4.746                                                                              H  H   H  1 H  H  H  H  O          H  NO.sub.2                             4.747                                                                              H  H   H  2 H  H  H  H  O          H  NO.sub.2                             4.748                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═O    H  NO.sub.2                             4.749                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═O    H  NO.sub.2                             4.750                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═O    H  NO.sub.2                             4.751                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOCH.sub.3                                                                               H  NO.sub.2                             4.752                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOCH.sub.3                                                                               H  NO.sub.2                             4.753                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOCH.sub.3                                                                               H  NO.sub.2                             4.754                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  NO.sub.2                             4.755                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  NO.sub.2                             4.756                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  NO.sub.2                             4.757                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOiPr     H  NO.sub.2                             4.758                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOiPr     H  NO.sub.2                             4.759                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOiPr     H  NO.sub.2                             4.760                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  NO.sub.2                             4.761                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  NO.sub.2                             4.762                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  NO.sub.2                             4.763                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  NO.sub.2                             4.764                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  NO.sub.2                             4.765                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  NO.sub.2                             4.766                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOiPr                                                                               H  NO.sub.2                             4.767                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOiPr                                                                               H  NO.sub.2                             4.768                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOiPr                                                                               H  NO.sub.2                             4.769                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  NO.sub.2                             4.770                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  NO.sub.2                             4.771                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  NO.sub.2                             4.772                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  NO.sub.2                             4.773                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  NO.sub.2                             4.774                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  NO.sub.2                             4.775                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  NO.sub.2                             4.776                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  NO.sub.2                             4.777                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  NO.sub.2                             4.778                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR78## H  NO.sub.2                             4.779                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR79## H  NO.sub.2                             4.780                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR80## H  NO.sub.2                             4.781                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR81## H  NO.sub.2                             4.782                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR82## H  NO.sub.2                             4.783                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR83## H  NO.sub.2                             4.784                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  NO.sub.2                             4.785                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  NO.sub.2                             4.786                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  NO.sub.2                             4.787                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.788                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.789                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.790                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  NO.sub.2                             4.791                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  NO.sub.2                             4.792                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  NO.sub.2                             4.793                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  NO.sub.2                             4.794                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  NO.sub.2                             4.795                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  NO.sub.2                             4.796                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  NO.sub.2                             4.797                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  NO.sub.2                             4.798                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  NO.sub.2                             4.799                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.800                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.801                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.802                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  NO.sub.2                             4.803                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  NO.sub.2                             4.804                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  NO.sub.2                             4.805                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  NO.sub.2                             4.806                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  NO.sub.2                             4.807                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  NO.sub.2                             4.808                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  NO.sub.2                             4.809                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  NO.sub.2                             4.810                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  NO.sub.2                             4.811                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  NO.sub.2                             4.812                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  NO.sub.2                             4.813                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  NO.sub.2                             4.814                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  NO.sub.2                             4.815                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  NO.sub.2                             4.816                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  NO.sub.2                             4.817                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  O          H  NO.sub.2                             4.818                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  O          H  NO.sub.2                             4.819                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  O          H  NO.sub.2                             4.820                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═O    H  NO.sub.2                             4.821                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═O    H  NO.sub.2                             4.822                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═O    H  NO.sub.2                             4.823                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOCH.sub.3                                                                               H  NO.sub.2                             4.824                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOCH.sub.3                                                                               H  NO.sub.2                             4.825                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOCH.sub.3                                                                               H  NO.sub.2                             4.826                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  NO.sub.2                             4.827                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  NO.sub.2                             4.828                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H  NO.sub.2                             4.829                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOiPr     H  NO.sub.2                             4.830                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOiPr     H  NO.sub.2                             4.831                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOiPr     H  NO.sub.2                             4.832                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.3                                                                          H  NO.sub.2                             4.833                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.3                                                                          H  NO.sub.2                             4.834                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.3                                                                          H  NO.sub.2                             4.835                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  NO.sub.2                             4.836                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  NO.sub.2                             4.837                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  NO.sub.2                             4.838                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOiPr                                                                               H  NO.sub.2                             4.839                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOiPr                                                                               H  NO.sub.2                             4.840                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOiPr                                                                               H  NO.sub.2                             4.841                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  NO.sub.2                             4.842                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  NO.sub.2                             4.843                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  NO.sub.2                             4.844                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  NO.sub.2                             4.845                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  NO.sub.2                             4.846                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  NO.sub.2                             4.847                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  NO.sub.2                             4.848                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  NO.sub.2                             4.849                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H  NO.sub.2                             4.850                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR84## H  NO.sub.2                             4.851                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR85## H  NO.sub.2                             4.852                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR86## H  NO.sub.2                             4.853                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR87## H  NO.sub.2                             4.854                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR88## H  NO.sub.2                             4.855                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR89## H  NO.sub.2                             4.856                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--CH.sub.3                                                                         H  NO.sub.2                             4.857                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--CH.sub.3                                                                         H  NO.sub.2                             4.858                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--CH.sub.3                                                                         H  NO.sub.2                             4.859                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.860                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.861                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.862                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H  NO.sub.2                             4.863                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H  NO.sub.2                             4.864                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H  NO.sub.2                             4.865                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  NO.sub.2                             4.866                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  NO.sub.2                             4.867                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  NO.sub.2                             4.868                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  NO.sub.2                             4.869                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  NO.sub.2                             4.870                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  NO.sub.2                             4.871                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.872                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.873                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  NO.sub.2                             4.874                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  NO.sub.2                             4.875                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  NO.sub.2                             4.876                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  NO.sub.2                             4.877                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--NH.sub.2                                                                         H  NO.sub.2                             4.878                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--NH.sub.2                                                                         H  NO.sub.2                             4.879                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--NH.sub.2                                                                         H  NO.sub.2                             4.880                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  NO.sub.2                             4.881                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  NO.sub.2                             4.882                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  NO.sub.2                             4.883                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  NO.sub.2                             4.884                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  NO.sub.2                             4.885                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  NO.sub.2                             4.886                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  NO.sub.2                             4.887                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  NO.sub.2                             4.888                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  NO.sub.2                             4.889                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  O          H  NO.sub.2                             4.890                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  O          H  NO.sub.2                             4.891                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  O          H  NO.sub.2                             4.892                                                                              H  H   H  0 H  H  H  H  C═O    CH.sub.3                                                                          CH.sub.3                             4.893                                                                              H  H   H  1 H  H  H  H  C═O    CH.sub.3                                                                          CH.sub.3                             4.894                                                                              H  H   H  2 H  H  H  H  C═O    CH.sub.3                                                                          CH.sub.3                             4.895                                                                              H  H   H  0 H  H  H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                             4.896                                                                              H  H   H  1 H  H  H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                             4.897                                                                              H  H   H  2 H  H  H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                             4.898                                                                              H  H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                             4.899                                                                              H  H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                             4.900                                                                              H  H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                             4.901                                                                              H  H   H  0 H  H  H  H  CHOiPr     CH.sub.3                                                                          CH.sub.3                             4.902                                                                              H  H   H  1 H  H  H  H  CHOiPr     CH.sub.3                                                                          CH.sub.3                             4.903                                                                              H  H   H  2 H  H  H  H  CHOiPr     CH.sub.3                                                                          CH.sub.3                             4.904                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                             4.905                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                             4.906                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                             4.907                                                                              H  H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                             4.908                                                                              H  H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                             4.909                                                                              H  H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                             4.910                                                                              H  H   H  0 H  H  H  H  C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                             4.911                                                                              H  H   H  1 H  H  H  H  C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                             4.912                                                                              H  H   H  2 H  H  H  H  C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                             4.913                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                             4.914                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                             4.915                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                             4.916                                                                              H  H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                             4.917                                                                              H  H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                             4.918                                                                              H  H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                             4.919                                                                              H  H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.920                                                                              H  H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.921                                                                              H  H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.922                                                                              H  H   H  0 H  H  H  H                                                                                  ##STR90## CH.sub.3                                                                          CH.sub.3                             4.923                                                                              H  H   H  1 H  H  H  H                                                                                  ##STR91## CH.sub.3                                                                          CH.sub.3                             4.924                                                                              H  H   H  2 H  H  H  H                                                                                  ##STR92## CH.sub.3                                                                          CH.sub.3                             4.925                                                                              H  H   H  0 H  H  H  H                                                                                  ##STR93## CH.sub.3                                                                          CH.sub.3                             4.926                                                                              H  H   H  1 H  H  H  H                                                                                  ##STR94## CH.sub.3                                                                          CH.sub.3                             4.927                                                                              H  H   H  2 H  H  H  H                                                                                  ##STR95## CH.sub.3                                                                          CH.sub.3                             4.928                                                                              H  H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                             4.929                                                                              H  H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                             4.930                                                                              H  H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                             4.931                                                                              H  H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.932                                                                              H  H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.933                                                                              H  H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.934                                                                              H  H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            CH.sub.3                                                                          CH.sub.3                             4.935                                                                              H  H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            CH.sub.3                                                                          CH.sub.3                             4.936                                                                              H  H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            CH.sub.3                                                                          CH.sub.3                             4.937                                                                              H  H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     CH.sub.3                                                                          CH.sub.3                             4.938                                                                              H  H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     CH.sub.3                                                                          CH.sub.3                             4.939                                                                              H  H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     CH.sub.3                                                                          CH.sub.3                             4.940                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     CH.sub.3                                                                          CH.sub.3                             4.941                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     CH.sub.3                                                                          CH.sub.3                             4.942                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     CH.sub.3                                                                          CH.sub.3                             4.943                                                                              H  H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.944                                                                              H  H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.945                                                                              H  H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.946                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           CH.sub.3                                                                          CH.sub.3                             4.947                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           CH.sub.3                                                                          CH.sub.3                             4.948                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           CH.sub.3                                                                          CH.sub.3                             4.949                                                                              H  H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.950                                                                              H  H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.951                                                                              H  H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.952                                                                              H  H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                             4.953                                                                              H  H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                             4.954                                                                              H  H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                             4.955                                                                              H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  CH.sub.3                                                                          CH.sub.3                             4.956                                                                              H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  CH.sub.3                                                                          CH.sub.3                             4.957                                                                              H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  CH.sub.3                                                                          CH.sub.3                             4.958                                                                              H  H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    CH.sub.3                                                                          CH.sub.3                             4.959                                                                              H  H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    CH.sub.3                                                                          CH.sub.3                             4.960                                                                              H  H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    CH.sub.3                                                                          CH.sub.3                             4.961                                                                              H  H   H  0 H  H  H  H  O          CH.sub.3                                                                          CH.sub.3                             4.962                                                                              H  H   H  1 H  H  H  H  O          CH.sub.3                                                                          CH.sub.3                             4.963                                                                              H  H   H  2 H  H  H  H  O          CH.sub.3                                                                          CH.sub.3                             4.964                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═O    CH.sub.3                                                                          CH.sub.3                             4.965                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═O    CH.sub.3                                                                          CH.sub.3                             4.966                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═O    CH.sub.3                                                                          CH.sub.3                             4.967                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                             4.968                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                             4.969                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                             4.970                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                             4.971                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                             4.972                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                             4.973                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  CHOiPr     CH.sub.3                                                                          CH.sub.3                             4.974                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  CHOiPr     CH.sub.3                                                                          CH.sub.3                             4.975                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  CHOiPr     CH.sub.3                                                                          CH.sub.3                             4.976                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                             4.977                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                             4.978                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                             4.979                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                             4.980                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                             4.981                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                             4.982                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                             4.983                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                             4.984                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                             4.985                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                             4.986                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                             4.987                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                             4.988                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                             4.989                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                             4.990                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                             4.991                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.992                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.993                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.994                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR96## CH.sub.3                                                                          CH.sub.3                             4.995                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR97## CH.sub.3                                                                          CH.sub.3                             4.996                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR98## CH.sub.3                                                                          CH.sub.3                             4.997                                                                              CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR99## CH.sub.3                                                                          CH.sub.3                             4.998                                                                              CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR100##                                                                               CH.sub.3                                                                          CH.sub.3                             4.999                                                                              CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR101##                                                                               CH.sub.3                                                                          CH.sub.3                             4.1000                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                             4.1001                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                             4.1002                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                             4.1003                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1004                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1005                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1006                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            CH.sub.3                                                                          CH.sub.3                             4.1007                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            CH.sub.3                                                                          CH.sub.3                             4.1008                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            CH.sub.3                                                                          CH.sub.3                             4.1009                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     CH.sub.3                                                                          CH.sub.3                             4.1010                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     CH.sub.3                                                                          CH.sub.3                             4.1011                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     CH.sub.3                                                                          CH.sub.3                             4.1012                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     CH.sub.3                                                                          CH.sub.3                             4.1013                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     CH.sub.3                                                                          CH.sub.3                             4.1014                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     CH.sub.3                                                                          CH.sub.3                             4.1015                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1016                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1017                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1018                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           CH.sub.3                                                                          CH.sub.3                             4.1019                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           CH.sub.3                                                                          CH.sub.3                             4.1020                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           CH.sub.3                                                                          CH.sub.3                             4.1021                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.1022                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.1023                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.1024                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                             4.1025                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                             4.1026                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                             4.1027                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  CH.sub.3                                                                          CH.sub.3                             4.1028                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  CH.sub.3                                                                          CH.sub.3                             4.1029                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  CH.sub.3                                                                          CH.sub.3                             4.1030                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    CH.sub.3                                                                          CH.sub.3                             4.1031                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    CH.sub.3                                                                          CH.sub.3                             4.1032                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    CH.sub.3                                                                          CH.sub.3                             4.1033                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  O          CH.sub.3                                                                          CH.sub.3                             4.1034                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  O          CH.sub.3                                                                          CH.sub.3                             4.1035                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  O          CH.sub.3                                                                          CH.sub.3                             4.1036                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═O    CH.sub.3                                                                          CH.sub.3                             4.1037                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═O    CH.sub.3                                                                          CH.sub.3                             4.1038                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═O    CH.sub.3                                                                          CH.sub.3                             4.1039                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                             4.1040                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                             4.1041                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOCH.sub.3                                                                               CH.sub.3                                                                          CH.sub.3                             4.1042                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                             4.1043                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                             4.1044                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        CH.sub.3                                                                          CH.sub.3                             4.1045                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOiPr     CH.sub.3                                                                          CH.sub.3                             4.1046                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOiPr     CH.sub.3                                                                          CH.sub.3                             4.1047                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOiPr     CH.sub.3                                                                          CH.sub.3                             4.1048                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                             4.1049                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                             4.1050                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.3                                                                          CH.sub.3                                                                          CH.sub.3                             4.1051                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                             4.1052                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                             4.1053                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   CH.sub.3                                                                          CH.sub.3                             4.1054                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                             4.1055                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                             4.1056                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOiPr                                                                               CH.sub.3                                                                          CH.sub.3                             4.1057                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                             4.1058                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                             4.1059                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              CH.sub.3                                                                          CH.sub.3                             4.1060                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                             4.1061                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                             4.1062                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          CH.sub.3                                                                          CH.sub.3                             4.1063                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.1064                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.1065                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.1066                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR102##                                                                               CH.sub.3                                                                          CH.sub.3                             4.1067                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR103##                                                                               CH.sub.3                                                                          CH.sub.3                             4.1068                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR104##                                                                               CH.sub.3                                                                          CH.sub.3                             4.1069                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR105##                                                                               CH.sub.3                                                                          CH.sub.3                             4.1070                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR106##                                                                               CH.sub.3                                                                          CH.sub.3                             4.1071                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR107##                                                                               CH.sub.3                                                                          CH.sub.3                             4.1072                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                             4.1073                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                             4.1074                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--CH.sub.3                                                                         CH.sub.3                                                                          CH.sub.3                             4.1075                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1076                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1077                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1078                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHCH.sub.3                                                                            CH.sub.3                                                                          CH.sub.3                             4.1079                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHCH.sub.3                                                                            CH.sub.3                                                                          CH.sub.3                             4.1080                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHCH.sub.3                                                                            CH.sub.3                                                                          CH.sub.3                             4.1081                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     CH.sub.3                                                                          CH.sub.3                             4.1082                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     CH.sub.3                                                                          CH.sub.3                             4.1083                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     CH.sub.3                                                                          CH.sub.3                             4.1084                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     CH.sub.3                                                                          CH.sub.3                             4.1085                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     CH.sub.3                                                                          CH.sub.3                             4.1086                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     CH.sub.3                                                                          CH.sub.3                             4.1087                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1088                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1089                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    CH.sub.3                                                                          CH.sub.3                             4.1090                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           CH.sub.3                                                                          CH.sub.3                             4.1091                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           CH.sub.3                                                                          CH.sub.3                             4.1092                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           CH.sub.3                                                                          CH.sub.3                             4.1093                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--NH.sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.1094                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--NH.sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.1095                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--NH.sub.2                                                                         CH.sub.3                                                                          CH.sub.3                             4.1096                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                             4.1097                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                             4.1098                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                CH.sub.3                                                                          CH.sub.3                             4.1099                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  CH.sub.3                                                                          CH.sub.3                             4.1100                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  CH.sub.3                                                                          CH.sub.3                             4.1101                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  CH.sub.3                                                                          CH.sub.3                             4.1102                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    CH.sub.3                                                                          CH.sub.3                             4.1103                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    CH.sub.3                                                                          CH.sub.3                             4.1104                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    CH.sub.3                                                                          CH.sub.3                             4.1105                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  O          CH.sub.3                                                                          CH.sub.3                             4.1106                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  O          CH.sub.3                                                                          CH.sub.3                             4.1107                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  O          CH.sub.3                                                                          CH.sub.3                             4.1108                                                                             H  H   H  0 H  H  H  H  C═O    Cl Cl                                   4.1109                                                                             H  H   H  1 H  H  H  H  C═O    Cl Cl                                   4.1110                                                                             H  H   H  2 H  H  H  H  C═O    Cl Cl                                   4.1111                                                                             H  H   H  0 H  H  H  H  CHOCH.sub.3                                                                               Cl Cl                                   4.1112                                                                             H  H   H  1 H  H  H  H  CHOCH.sub.3                                                                               Cl Cl                                   4.1113                                                                             H  H   H  2 H  H  H  H  CHOCH.sub.3                                                                               Cl Cl                                   4.1114                                                                             H  H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        Cl Cl                                   4.1115                                                                             H  H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        Cl Cl                                   4.1116                                                                             H  H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        Cl Cl                                   4.1117                                                                             H  H   H  0 H  H  H  H  CHOiPr     Cl Cl                                   4.1118                                                                             H  H   H  1 H  H  H  H  CHOiPr     Cl Cl                                   4.1119                                                                             H  H   H  2 H  H  H  H  CHOiPr     Cl Cl                                   4.1120                                                                             H  H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          Cl Cl                                   4.1121                                                                             H  H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          Cl Cl                                   4.1122                                                                             H  H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          Cl Cl                                   4.1123                                                                             H  H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   Cl Cl                                   4.1124                                                                             H  H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   Cl Cl                                   4.1125                                                                             H  H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   Cl Cl                                   4.1126                                                                             H  H   H  0 H  H  H  H  C═NOiPr                                                                               Cl Cl                                   4.1127                                                                             H  H   H  1 H  H  H  H  C═NOiPr                                                                               Cl Cl                                   4.1128                                                                             H  H   H  2 H  H  H  H  C═NOiPr                                                                               Cl Cl                                   4.1129                                                                             H  H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl Cl                                   4.1130                                                                             H  H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl Cl                                   4.1131                                                                             H  H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl Cl                                   4.1132                                                                             H  H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl Cl                                   4.1133                                                                             H  H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl Cl                                   4.1134                                                                             H  H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl Cl                                   4.1135                                                                             H  H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         Cl Cl                                   4.1136                                                                             H  H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         Cl Cl                                   4.1137                                                                             H  H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         Cl Cl                                   4.1138                                                                             H  H   H  0 H  H  H  H                                                                                  ##STR108##                                                                               Cl Cl                                   4.1139                                                                             H  H   H  1 H  H  H  H                                                                                  ##STR109##                                                                               Cl Cl                                   4.1140                                                                             H  H   H  2 H  H  H  H                                                                                  ##STR110##                                                                               Cl Cl                                   4.1141                                                                             H  H   H  0 H  H  H  H                                                                                  ##STR111##                                                                               Cl Cl                                   4.1142                                                                             H  H   H  1 H  H  H  H                                                                                  ##STR112##                                                                               Cl Cl                                   4.1143                                                                             H  H   H  2 H  H  H  H                                                                                  ##STR113##                                                                               Cl Cl                                   4.1144                                                                             H  H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         Cl Cl                                   4.1145                                                                             H  H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         Cl Cl                                   4.1146                                                                             H  H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         Cl Cl                                   4.1147                                                                             H  H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1148                                                                             H  H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1149                                                                             H  H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1150                                                                             H  H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            Cl Cl                                   4.1151                                                                             H  H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            Cl Cl                                   4.1152                                                                             H  H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            Cl Cl                                   4.1153                                                                             H  H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     Cl Cl                                   4.1154                                                                             H  H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     Cl Cl                                   4.1155                                                                             H  H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     Cl Cl                                   4.1156                                                                             H  H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     Cl Cl                                   4.1157                                                                             H  H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     Ci Cl                                   4.1158                                                                             H  H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     Cl Cl                                   4.1159                                                                             H  H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1160                                                                             H  H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1161                                                                             H  H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1162                                                                             H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           Cl Cl                                   4.1163                                                                             H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           Cl Cl                                   4.1164                                                                             H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           Cl Cl                                   4.1165                                                                             H  H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         Cl Cl                                   4.1166                                                                             H  H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         Cl Cl                                   4.1167                                                                             H  H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         Cl Cl                                   4.1168                                                                             H  H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                Cl Cl                                   4.1169                                                                             H  H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                Cl Cl                                   4.1170                                                                             H  H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                Cl Cl                                   4.1171                                                                             H  H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  Cl Cl                                   4.1172                                                                             H  H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  Cl Cl                                   4.1173                                                                             H  H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  Cl Cl                                   4.1174                                                                             H  H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    Cl Cl                                   4.1175                                                                             H  H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    Cl Cl                                   4.1176                                                                             H  H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    Cl Cl                                   4.1177                                                                             H  H   H  0 H  H  H  H  O          Cl Cl                                   4.1178                                                                             H  H   H  1 H  H  H  H  O          Cl Cl                                   4.1179                                                                             H  H   H  2 H  H  H  H  O          Cl Cl                                   4.1180                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═O    Cl Cl                                   4.1181                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═O    Cl Cl                                   4.1182                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═O    Cl Cl                                   4.1183                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CHOCH.sub.3                                                                               Cl Cl                                   4.1184                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CHOCH.sub.3                                                                               Cl Cl                                   4.1185                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CHOCH.sub.3                                                                               Cl Cl                                   4.1186                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        Cl Cl                                   4.1187                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        Cl Cl                                   4.1188                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        Cl Cl                                   4.1189                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CHOiPr     Cl Cl                                   4.1190                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CHOiPr     Cl Cl                                   4.1191                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CHOiPr     Cl Cl                                   4.1192                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.3                                                                          Cl Cl                                   4.1193                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.3                                                                          Cl Cl                                   4.1194                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.3                                                                          Cl Cl                                   4.1195                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   Cl Cl                                   4.1196                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   Cl Cl                                   4.1197                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   Cl Cl                                   4.1198                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOiPr                                                                               Cl Cl                                   4.1199                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOiPr                                                                               Cl Cl                                   4.1200                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOiPr                                                                               Cl Cl                                   4.1201                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl Cl                                   4.1202                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl Cl                                   4.1203                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl Cl                                   4.1204                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl Cl                                   4.1205                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl Cl                                   4.1206                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl Cl                                   4.1207                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         Cl Cl                                   4.1208                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         Cl Cl                                   4.1209                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         Cl Cl                                   4.1210                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR114##                                                                               Cl Cl                                   4.1211                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR115##                                                                               Cl Cl                                   4.1212                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR116##                                                                               Cl Cl                                   4.1213                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H                                                                                  ##STR117##                                                                               Cl Cl                                   4.1214                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H                                                                                  ##STR118##                                                                               Cl Cl                                   4.1215                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H                                                                                  ##STR119##                                                                               Cl Cl                                   4.1216                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--CH.sub.3                                                                         Cl Cl                                   4.1217                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--CH.sub.3                                                                         Cl Cl                                   4.1218                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--CH.sub.3                                                                         Cl Cl                                   4.1219                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1220                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1221                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1222                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHCH.sub.3                                                                            Cl Cl                                   4.1223                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHCH.sub.3                                                                            Cl Cl                                   4.1224                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHCH.sub.3                                                                            Cl Cl                                   4.1225                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     Cl Cl                                   4.1226                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     Cl Cl                                   4.1227                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     Cl Cl                                   4.1228                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     Cl Cl                                   4.1229                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     Cl Cl                                   4.1230                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     Cl Cl                                   4.1231                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1232                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1233                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1234                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           Cl Cl                                   4.1235                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           Cl Cl                                   4.1236                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           Cl Cl                                   4.1237                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--NH.sub.2                                                                         Cl Cl                                   4.1238                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--NH.sub.2                                                                         Cl Cl                                   4.1239                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--NH.sub.2                                                                         Cl Cl                                   4.1240                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                Cl Cl                                   4.1241                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                Cl Cl                                   4.1242                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                Cl Cl                                   4.1243                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  Cl Cl                                   4.1244                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  Cl Cl                                   4.1245                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  Cl Cl                                   4.1246                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    Cl Cl                                   4.1247                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    Cl Cl                                   4.1248                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    Cl Cl                                   4.1249                                                                             CH.sub.3                                                                          H   H  0 H  H  H  H  O          Cl Cl                                   4.1250                                                                             CH.sub.3                                                                          H   H  1 H  H  H  H  O          Cl Cl                                   4.1251                                                                             CH.sub.3                                                                          H   H  2 H  H  H  H  O          Cl Cl                                   4.1252                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═O    Cl Cl                                   4.1253                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═O    Cl Cl                                   4.1254                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═O    Cl Cl                                   4.1255                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOCH.sub.3                                                                               Cl Cl                                   4.1256                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOCH.sub.3                                                                               Cl Cl                                   4.1257                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOCH.sub.3                                                                               Cl Cl                                   4.1258                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        Cl Cl                                   4.1259                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        Cl Cl                                   4.1260                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        Cl Cl                                   4.1261                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CHOiPr     Cl Cl                                   4.1262                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CHOiPr     Cl Cl                                   4.1263                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CHOiPr     Cl Cl                                   4.1264                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.3                                                                          Cl Cl                                   4.1265                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.3                                                                          Cl Cl                                   4.1266                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.3                                                                          Cl Cl                                   4.1267                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   Cl Cl                                   4.1268                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   Cl Cl                                   4.1269                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   Cl Cl                                   4.1270                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOiPr                                                                               Cl Cl                                   4.1271                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOiPr                                                                               Cl Cl                                   4.1272                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOiPr                                                                               Cl Cl                                   4.1273                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl Cl                                   4.1274                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl Cl                                   4.1275                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              Cl Cl                                   4.1276                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl Cl                                   4.1277                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl Cl                                   4.1278                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          Cl Cl                                   4.1279                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         Cl Cl                                   4.1280                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         Cl Cl                                   4.1281                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         Cl Cl                                   4.1282                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR120##                                                                               Cl Cl                                   4.1283                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR121##                                                                               Cl Cl                                   4.1284                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR122##                                                                               Cl Cl                                   4.1285                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H                                                                                  ##STR123##                                                                               Cl Cl                                   4.1286                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H                                                                                  ##STR124##                                                                               Cl Cl                                   4.1287                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H                                                                                  ##STR125##                                                                               Cl Cl                                   4.1288                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--CH.sub.3                                                                         Cl Cl                                   4.1289                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--CH.sub.3                                                                         Cl Cl                                   4.1290                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--CH.sub.3                                                                         Cl Cl                                   4.1291                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1292                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1293                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1294                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHCH.sub.3                                                                            Cl Cl                                   4.1295                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHCH.sub.3                                                                            Cl Cl                                   4.1296                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHCH.sub.3                                                                            Cl Cl                                   4.1297                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     Cl Cl                                   4.1298                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     Cl Cl                                   4.1299                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     Cl Cl                                   4.1300                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     Cl Cl                                   4.1301                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     Cl Cl                                   4.1302                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     Cl Cl                                   4.1303                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1304                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1305                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    Cl Cl                                   4.1306                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           Cl Cl                                   4.1307                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           Cl Cl                                   4.1308                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           Cl Cl                                   4.1309                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--NH.sub.2                                                                         Cl Cl                                   4.1310                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--NH.sub.2                                                                         Cl Cl                                   4.1311                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--NH.sub.2                                                                         Cl Cl                                   4.1312                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                Cl Cl                                   4.1313                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                Cl Cl                                   4.1314                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                Cl Cl                                   4.1315                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  Cl Cl                                   4.1316                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  Cl Cl                                   4.1317                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  Cl Cl                                   4.1 CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    Cl Cl                                   4.2 CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    Cl Cl                                   4.3 CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    Cl Cl                                   4.4 CH.sub.3                                                                          CH.sub.3                                                                           H  0 H  H  H  H  O          Cl Cl                                   4.5 CH.sub.3                                                                          CH.sub.3                                                                           H  1 H  H  H  H  O          Cl Cl                                   4.6 CH.sub.3                                                                          CH.sub.3                                                                           H  2 H  H  H  H  O          Cl Cl                                   4.7 H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  CH.sub.3                             4.8 H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  CH.sub.3                             4.9 H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  CH.sub.3                             4.10                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--OCH.sub.3                                                                             H  CH.sub.3                             4.11                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--OCH.sub.3                                                                             H  CH.sub.3                             4.12                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--OCH.sub.3                                                                             H  CH.sub.3                             4.13                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.14                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.15                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.16                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  CH.sub.3                             4.17                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  CH.sub.3                             4.18                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  CH.sub.3                             4.19                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.20                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.21                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.22                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.23                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.24                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.25                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  CH.sub.3                             4.26                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  CH.sub.3                             4.27                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  CH.sub.3                             4.28                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.29                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.30                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.31                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.32                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.33                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.34                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.35                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.36                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.37                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR126##                                                                               H  CH.sub.3                             4.38                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR127##                                                                               H  CH.sub.3                             4.39                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR128##                                                                               H  CH.sub.3                             4.40                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR129##                                                                               H  CH.sub.3                             4.41                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR130##                                                                               H  CH.sub.3                             4.42                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR131##                                                                               H  CH.sub.3                             4.43                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.44                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.45                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.46                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.47                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.48                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.49                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.50                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.51                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.52                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.53                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.54                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.55                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.56                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.57                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.58                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.59                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.60                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.61                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.62                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.63                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.64                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.65                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.66                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.67                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.68                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.69                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.70                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.71                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.72                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.73                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.74                                                                               H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.75                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.76                                                                               H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  CH.sub.3                             4.77                                                                               H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  CH.sub.3                             4.78                                                                               CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  CH.sub.3                             4.79                                                                               CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  CH.sub.3                             4.80                                                                               CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  CH.sub.3                             4.81                                                                               CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.82                                                                               CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.83                                                                               CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.84                                                                               CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.85                                                                               CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.86                                                                               CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.87                                                                               CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  CH.sub.3                             4.88                                                                               CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  CH.sub.3                             4.89                                                                               CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  CH.sub.3                             4.90                                                                               CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.91                                                                               CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.92                                                                               CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.93                                                                               CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.94                                                                               CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.95                                                                               CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.96                                                                               CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  CH.sub.3                             4.97                                                                               CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  CH.sub.3                             4.98                                                                               CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  CH.sub.3                             4.99                                                                               CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.100                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.101                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.102                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.103                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.104                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.105                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.106                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.107                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.108                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR132##                                                                               H  CH.sub.3                             4.109                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR133##                                                                               H  CH.sub.3                             4.110                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR134##                                                                               H  CH.sub.3                             4.111                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR135##                                                                               H  CH.sub.3                             4.112                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR136##                                                                               H  CH.sub.3                             4.113                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR137##                                                                               H  CH.sub.3                             4.114                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.115                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.116                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.117                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.118                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.119                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.120                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.121                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.122                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.123                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.124                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.125                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.126                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.127                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.128                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.129                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.130                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.131                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.132                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.133                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.134                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.135                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.136                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.137                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.138                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.139                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.140                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.141                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.142                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.143                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.144                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.145                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.146                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.147                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  CH.sub.3                             4.148                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  CH.sub.3                             4.149                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  CH.sub.3                             4.150                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  CH.sub.3                             4.151                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  CH.sub.3                             4.152                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.153                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.154                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.155                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.156                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.157                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.158                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  CH.sub.3                             4.159                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  CH.sub.3                             4.160                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  CH.sub.3                             4.161                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.162                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.163                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.164                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.165                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.166                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.167                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  CH.sub.3                             4.168                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  CH.sub.3                             4.169                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  CH.sub.3                             4.170                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.171                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.172                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.173                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.174                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.175                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.176                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.177                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.178                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.179                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR138##                                                                               H  CH.sub.3                             4.180                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR139##                                                                               H  CH.sub.3                             4.181                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR140##                                                                               H  CH.sub.3                             4.182                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR141##                                                                               H  CH.sub.3                             4.183                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR142##                                                                               H  CH.sub.3                             4.184                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR143##                                                                               H  CH.sub.3                             4.185                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.186                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.187                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.188                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.189                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.190                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.191                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.192                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.193                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.194                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.195                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.196                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.197                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.198                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.199                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.200                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.201                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.202                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.203                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.204                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.205                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.206                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.207                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.208                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.209                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.210                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.211                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.212                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.213                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.214                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.215                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.216                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.217                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.218                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  CH.sub.3                             4.219                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  CH.sub.3                             4.220                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═O    H  Cl                                   4.221                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═O    H  Cl                                   4.222                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═O    H  Cl                                   4.223                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.224                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.225                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.226                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.227                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.228                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.229                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CHOiPr     H  Cl                                   4.230                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CHOiPr     H  Cl                                   4.231                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CHOiPr     H  Cl                                   4.232                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.233                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.234                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.235                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.236                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.237                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.238                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  Cl                                   4.239                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  Cl                                   4.240                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  Cl                                   4.241                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.242                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.243                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.244                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.245                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.246                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.247                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.248                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.249                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.250                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR144##                                                                               H  Cl                                   4.251                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR145##                                                                               H  Cl                                   4.252                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR146##                                                                               H  Cl                                   4.253                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR147##                                                                               H  Cl                                   4.254                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR148##                                                                               H  Cl                                   4.255                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR149##                                                                               H  Cl                                   4.256                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.257                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.258                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.259                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.260                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.261                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.262                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.263                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.264                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.265                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.266                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.267                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.268                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.269                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.270                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.271                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.272                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.273                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.274                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.275                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.276                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.277                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.278                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.279                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.280                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.281                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.282                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.283                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.284                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.285                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.286                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.287                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.288                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.289                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  O          H  Cl                                   4.290                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  O          H  Cl                                   4.291                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═O    H  Cl                                   4.292                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═O    H  Cl                                   4.293                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═O    H  Cl                                   4.294                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.295                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.296                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.297                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.298                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.299                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.300                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CHOiPr     H  Cl                                   4.301                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CHOiPr     H  Cl                                   4.302                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CHOiPr     H  Cl                                   4.303                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.304                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.305                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.306                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.307                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.308                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.309                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  Cl                                   4.310                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  Cl                                   4.311                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  Cl                                   4.312                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.313                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.314                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.315                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.316                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.317                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.318                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.319                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.320                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.321                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR150##                                                                               H  Cl                                   4.322                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR151##                                                                               H  Cl                                   4.323                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR152##                                                                               H  Cl                                   4.324                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR153##                                                                               H  Cl                                   4.325                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR154##                                                                               H  Cl                                   4.326                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR155##                                                                               H  Cl                                   4.327                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.328                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.329                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.330                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.331                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.332                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.333                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.334                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.335                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.336                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.337                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.338                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.339                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.340                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.341                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.342                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.343                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.344                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.345                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.346                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.347                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.348                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.349                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.350                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.351                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.352                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.353                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.354                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.355                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.356                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.357                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.358                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.359                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.360                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  O          H  Cl                                   4.361                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  O          H  Cl                                   4.362                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═O    H  Cl                                   4.363                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═O    H  Cl                                   4.364                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═O    H  Cl                                   4.365                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.366                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.367                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  Cl                                   4.368                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.369                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.370                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.371                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CHOiPr     H  Cl                                   4.372                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CHOiPr     H  Cl                                   4.373                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CHOiPr     H  Cl                                   4.374                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.375                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.376                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.377                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.378                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.379                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.380                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  Cl                                   4.381                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  Cl                                   4.382                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  Cl                                   4.383                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.384                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.385                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.386                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.387                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.388                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.389                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.390                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.391                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.392                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR156##                                                                               H  Cl                                   4.393                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR157##                                                                               H  Cl                                   4.394                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR158##                                                                               H  Cl                                   4.395                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR159##                                                                               H  Cl                                   4.396                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR160##                                                                               H  Cl                                   4.397                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR161##                                                                               H  Cl                                   4.398                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.399                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.400                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.401                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.402                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.403                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.404                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.405                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.406                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.407                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.408                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.409                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.410                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.411                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.412                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.413                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.414                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.415                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.416                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.417                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.418                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.419                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.420                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.421                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.422                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.423                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.424                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.425                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.426                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.427                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.428                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.429                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.430                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.431                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  O          H  Cl                                   4.432                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  O          H  Cl                                   4.433                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  CH.sub.3                             4.434                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  CH.sub.3                             4.435                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  CH.sub.3                             4.436                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--OCH.sub.3                                                                             H  CH.sub.3                             4.437                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--OCH.sub.3                                                                             H  CH.sub.3                             4.438                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--OCH.sub.3                                                                             H  CH.sub.3                             4.439                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.440                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.441                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.442                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  CH.sub.3                             4.443                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  CH.sub.3                             4.444                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  CH.sub.3                             4.445                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.446                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.447                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.448                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.449                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.450                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.451                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  CH.sub.3                             4.452                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.453                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  CH.sub.3                             4.454                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.455                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.456                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.457                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.458                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.459                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.460                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.461                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.462                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.463                                                                              H  H   H  0 CH.sub.3                                                                          H     H                                                                                  ##STR162##                                                                               H  CH.sub.3                             4.464                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR163##                                                                               H  CH.sub.3                             4.465                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR164##                                                                               H  CH.sub.3                             4.466                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR165##                                                                               H  CH.sub.3                             4.467                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR166##                                                                               H  CH.sub.3                             4.468                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR167##                                                                               H  CH.sub.3                             4.469                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.470                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.471                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.472                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.473                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.474                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.475                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.476                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.477                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.478                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.479                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.480                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.481                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.482                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.483                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.484                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.485                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.486                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.487                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.488                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.489                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.490                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.491                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.492                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.493                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.494                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.495                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.496                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.497                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.498                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.499                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.500                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.501                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.502                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  CH.sub.3                             4.503                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  CH.sub.3                             4.504                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  CH.sub.3                             4.505                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  CH.sub.3                             4.506                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  CH.sub.3                             4.507                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.508                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.509                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.510                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.511                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.512                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.513                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  CH.sub.3                             4.514                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  CH.sub.3                             4.515                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  CH.sub.3                             4.516                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.517                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.518                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.519                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.520                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.521                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.522                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  CH.sub.3                             4.523                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  CH.sub.3                             4.524                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  CH.sub.3                             4.525                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.526                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.527                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.528                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.529                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.530                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.531                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.532                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.533                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.534                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR168##                                                                               H  CH.sub.3                             4.535                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR169##                                                                               H  CH.sub.3                             4.536                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR170##                                                                               H  CH.sub.3                             4.537                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR171##                                                                               H  CH.sub.3                             4.538                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR172##                                                                               H  CH.sub.3                             4.539                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR173##                                                                               H  CH.sub.3                             4.540                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.541                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.542                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.543                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.544                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.545                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.546                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.547                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.548                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.549                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.550                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.551                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.552                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.553                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.554                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.555                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.556                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.557                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.558                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.559                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.560                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.561                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.562                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.563                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.564                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.565                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.566                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.567                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.568                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.569                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.570                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.571                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.572                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.573                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  CH.sub.3                             4.574                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  CH.sub.3                             4.575                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  CH.sub.3                             4.576                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  CH.sub.3                             4.577                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  CH.sub.3                             4.578                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.579                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.580                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.581                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.582                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.583                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.584                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  CH.sub.3                             4.585                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  CH.sub.3                             4.586                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  CH.sub.3                             4.587                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.588                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.589                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.590                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.591                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.592                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.593                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  CH.sub.3                             4.594                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  CH.sub.3                             4.595                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  CH.sub.3                             4.596                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.597                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.598                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.599                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.600                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.601                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.602                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.603                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.604                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.605                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR174##                                                                               H  CH.sub.3                             4.606                                                                              CH.sub.3                                                                          CH.sub.3 C                                                                         H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR175##                                                                               H  CH.sub.3                             4.607                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR176##                                                                               H  CH.sub.3                             4.608                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR177##                                                                               H  CH.sub.3                             4.609                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR178##                                                                               H  CH.sub.3                             4.610                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR179##                                                                               H  CH.sub.3                             4.611                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.612                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.613                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.614                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.615                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.616                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.617                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.618                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.619                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.620                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.621                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.622                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.623                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.624                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.625                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.626                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.627                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.628                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.629                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.630                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.631                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.632                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.633                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.634                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.635                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.636                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.637                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.638                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.639                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.640                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.641                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.642                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.643                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.644                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  CH.sub.3                             4.645                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  CH.sub.3                             4.646                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  Cl                                   4.647                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  Cl                                   4.648                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  Cl                                   4.649                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  Cl                                   4.650                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  Cl                                   4.651                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  Cl                                   4.652                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.653                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.654                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.655                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  Cl                                   4.656                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  Cl                                   4.657                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  Cl                                   4.658                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  Cl                                   4.659                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  Cl                                   4.660                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  Cl                                   4.661                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.662                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.663                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.664                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  Cl                                   4.665                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  Cl                                   4.666                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  Cl                                   4.667                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.668                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.669                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.670                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.671                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.672                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.673                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.674                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.675                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.676                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR180##                                                                               H  Cl                                   4.677                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR181##                                                                               H  Cl                                   4.678                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR182##                                                                               H  Cl                                   4.679                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR183##                                                                               H  Cl                                   4.680                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR184##                                                                               H  Cl                                   4.681                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR185##                                                                               H  Cl                                   4.682                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  Cl                                   4.683                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  Cl                                   4.684                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  Cl                                   4.685                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.686                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.687                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.688                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  Cl                                   4.689                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  Cl                                   4.690                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  Cl                                   4.691                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.692                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.693                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.694                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.695                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.696                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.697                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.698                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.699                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.700                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.701                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.702                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.703                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  Cl                                   4.704                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  Cl                                   4.705                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  Cl                                   4.706                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.707                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.708                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.709                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.710                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.711                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.712                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.713                                                                              H  H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.714                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.715                                                                              H  H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  Cl                                   4.716                                                                              H  H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  Cl                                   4.717                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  Cl                                   4.718                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  Cl                                   4.719                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  Cl                                   4.720                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  Cl                                   4.721                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  Cl                                   4.722                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  Cl                                   4.723                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.724                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.725                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.726                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  Cl                                   4.727                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  Cl                                   4.728                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  Cl                                   4.729                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  Cl                                   4.730                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  Cl                                   4.731                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  Cl                                   4.732                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.733                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.734                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.735                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  Cl                                   4.736                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  Cl                                   4.737                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  Cl                                   4.738                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.739                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.740                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.741                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.742                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.743                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.744                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.745                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.746                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.747                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR186##                                                                               H  Cl                                   4.748                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR187##                                                                               H  Cl                                   4.749                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR188##                                                                               H  Cl                                   4.750                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR189##                                                                               H  Cl                                   4.751                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR190##                                                                               H  Cl                                   4.752                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR191##                                                                               H  Cl                                   4.753                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  Cl                                   4.754                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  Cl                                   4.755                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  Cl                                   4.756                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.757                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.758                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.759                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  Cl                                   4.760                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  Cl                                   4.761                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  Cl                                   4.762                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.763                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.764                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.765                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.766                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.767                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.768                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.769                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.770                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.771                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.772                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.773                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.774                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  Cl                                   4.775                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  Cl                                   4.776                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  Cl                                   4.777                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.778                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.779                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.780                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.781                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.782                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.783                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.784                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.785                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.786                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  Cl                                   4.787                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  Cl                                   4.788                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  Cl                                   4.789                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  Cl                                   4.790                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═O    H  Cl                                   4.791                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  Cl                                   4.792                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  Cl                                   4.793                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                               H  Cl                                   4.794                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.795                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.796                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.797                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  Cl                                   4.798                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  Cl                                   4.799                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CHOiPr     H  Cl                                   4.800                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  Cl                                   4.801                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  Cl                                   4.802                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.3                                                                          H  Cl                                   4.803                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.804                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.805                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.806                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  Cl                                   4.807                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  Cl                                   4.808                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOiPr                                                                               H  Cl                                   4.809                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.810                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.811                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.812                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.813                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.814                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.815                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.816                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.817                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.818                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR192##                                                                               H  Cl                                   4.819                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR193##                                                                               H  Cl                                   4.820                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR194##                                                                               H  Cl                                   4.821                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR195##                                                                               H  Cl                                   4.822                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR196##                                                                               H  Cl                                   4.823                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H                                                                                  ##STR197##                                                                               H  Cl                                   4.824                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  Cl                                   4.825                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  Cl                                   4.826                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--CH.sub.3                                                                         H  Cl                                   4.827                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.828                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.829                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.830                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  Cl                                   4.831                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  Cl                                   4.832                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHCH.sub.3                                                                            H  Cl                                   4.833                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.834                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.835                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.836                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.837                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.838                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.839                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.840                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.841                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.842                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.843                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.844                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.845                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  Cl                                   4.846                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  Cl                                   4.847                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--NH.sub.2                                                                         H  Cl                                   4.848                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.849                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.850                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.851                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.852                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.853                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.854                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.855                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.856                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.857                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  Cl                                   4.858                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  CH.sub.3                                                                          H  O          H  Cl                                   4.859                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═O    H  CH.sub.3                             4.860                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═O    H  CH.sub.3                             4.861                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═O    H  CH.sub.3                             4.862                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--OCH.sub.3                                                                             H  CH.sub.3                             4.863                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--OCH.sub.3                                                                             H  CH.sub.3                             4.864                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--OCH.sub.3                                                                             H  CH.sub.3                             4.865                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.866                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.867                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.868                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CHOiPr     H  CH.sub.3                             4.869                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CHOiPr     H  CH.sub.3                             4.870                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CHOiPr     H  CH.sub.3                             4.871                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.872                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.873                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.874                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.875                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.876                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.877                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.878                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.879                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.880                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.881                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.882                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.883                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.884                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.885                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.886                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.887                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.888                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.889                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR198##                                                                               H  CH.sub.3                             4.890                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR199##                                                                               H  CH.sub.3                             4.891                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR200##                                                                               H  CH.sub.3                             4.892                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR201##                                                                               H  CH.sub.3                             4.893                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR202##                                                                               H  CH.sub.3                             4.894                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR203##                                                                               H  CH.sub.3                             4.895                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.896                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.897                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.898                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.899                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.900                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.901                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.902                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.903                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.904                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.905                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.906                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.907                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.908                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.909                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.910                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.911                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.912                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.913                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.914                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.915                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.916                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.917                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.918                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.919                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.920                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.921                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.922                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.923                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.924                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.925                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.926                                                                              H  H   H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.927                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.928                                                                              H  H   H  0 CH.sub.3                                                                          H  H  H  O          H  CH.sub.3                             4.929                                                                              H  H   H  2 CH.sub.3                                                                          H  H  H  O          H  CH.sub.3                             4.930                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═O    H  CH.sub.3                             4.931                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═O    H  CH.sub.3                             4.932                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═O    H  CH.sub.3                             4.933                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.934                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.935                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.936                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.937                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.938                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.939                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CHOiPr     H  CH.sub.3                             4.940                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CHOiPr     H  CH.sub.3                             4.941                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CHOiPr     H  CH.sub.3                             4.942                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.943                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.944                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.945                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.946                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.947                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.948                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.949                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.950                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.951                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.952                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.953                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.954                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.955                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.956                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.957                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.958                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.959                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.960                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR204##                                                                               H  CH.sub.3                             4.961                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR205##                                                                               H  CH.sub.3                             4.962                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR206##                                                                               H  CH.sub.3                             4.963                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR207##                                                                               H  CH.sub.3                             4.964                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR208##                                                                               H  CH.sub.3                             4.965                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR209##                                                                               H  CH.sub.3                             4.966                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.967                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.968                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.969                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.970                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.971                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.972                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.973                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.974                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.975                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.976                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.977                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.978                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.979                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.980                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.981                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.982                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.983                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.984                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.985                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.986                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.987                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.988                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.989                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.990                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.991                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.992                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.993                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.994                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.995                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.996                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.997                                                                              CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.998                                                                              CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.999                                                                              CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          H  H  H  O          H  CH.sub.3                             4.1000                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          H  H  H  O          H  CH.sub.3                             4.1001                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═O    H  CH.sub.3                             4.1002                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═O    H  CH.sub.3                             4.1003                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═O    H  CH.sub.3                             4.1004                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.1005                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.1006                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CHOCH.sub.3                                                                               H  CH.sub.3                             4.1007                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.1008                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.1009                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                             4.1010                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CHOiPr     H  CH.sub.3                             4.1011                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CHOiPr     H  CH.sub.3                             4.1012                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CHOiPr     H  CH.sub.3                             4.1013                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.1014                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.1015                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.3                                                                          H  CH.sub.3                             4.1016                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.1017                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.1018                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                             4.1019                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.1020                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.1021                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NOiPr                                                                               H  CH.sub.3                             4.1022                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.1023                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.1024                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                             4.1025                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.1026                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.1027                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                             4.1028                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.1029                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.1030                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3).sub.2                                                                         H  CH.sub.3                             4.1031                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR210##                                                                               H  CH.sub.3                             4.1032                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR211##                                                                               H  CH.sub.3                             4.1033                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR212##                                                                               H  CH.sub.3                             4.1034                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H                                                                                  ##STR213##                                                                               H  CH.sub.3                             4.1035                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H                                                                                  ##STR214##                                                                               H  CH.sub.3                             4.1036                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H                                                                                  ##STR215##                                                                               H  CH.sub.3                             4.1037                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.1038                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.1039                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═N--CH.sub.3                                                                         H  CH.sub.3                             4.1040                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.1041                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.1042                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═NC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.1043                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.1044                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.1045                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--NHCH.sub.3                                                                            H  CH.sub.3                             4.1046                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.1047                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.1048                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H  CH.sub.3                             4.1049                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.1050                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.1051                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3).sub.2                                                                     H  CH.sub.3                             4.1052                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.1053                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.1054                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  CH.sub.3                             4.1055                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.1056                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.1057                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  CH.sub.3                             4.1058                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.1059                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.1060                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═N--NH.sub.2                                                                         H  CH.sub.3                             4.1061                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.1062                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.1063                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C═N--N(CH.sub.3).sub.2                                                                H  CH.sub.3                             4.1064                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.1065                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.1066                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  CH.sub.3                             4.1067                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.1068                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.1069                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  CH.sub.3                             4.1070                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          H  H  H  O          H  CH.sub.3                             4.1071                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          H  H  H  O          H  CH.sub.3                             4.1072                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  Cl                                   4.1073                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  Cl                                   4.1074                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  Cl                                   4.1075                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  Cl                                   4.1076                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  Cl                                   4.1077                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  Cl                                   4.1078                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.1079                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.1080                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.1081                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  Cl                                   4.1082                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  Cl                                   4.1083                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  Cl                                   4.1084                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.1085                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.1086                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.1087                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.1088                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.1089                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.1090                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  Cl                                   4.1091                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  Cl                                   4.1092                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  Cl                                   4.1093                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.1094                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.1095                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.1096                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.1097                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.1098                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.1099                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.1100                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.1101                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.1102                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR216##                                                                               H  Cl                                   4.1103                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR217##                                                                               H  Cl                                   4.1104                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR218##                                                                               H  Cl                                   4.1105                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR219##                                                                               H  Cl                                   4.1106                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR220##                                                                               H  Cl                                   4.1107                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR221##                                                                               H  Cl                                   4.1108                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.1109                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.1110                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.1111                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.1112                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.1113                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.1114                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.1115                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.1116                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.1117                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.1118                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.1119                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.1120                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.1121                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.1122                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.1123                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.1124                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.1125                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.1126                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.1127                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.1128                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.1129                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.1130                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.1131                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.1132                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.1133                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.1134                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.1135                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.1136                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.1137                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.1138                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.1139                                                                             H  H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.1140                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.1141                                                                             H  H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  Cl                                   4.1142                                                                             H  H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  Cl                                   4.1143                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  Cl                                   4.1144                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  Cl                                   4.1145                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  Cl                                   4.1146                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  Cl                                   4.1147                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  Cl                                   4.1148                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  Cl                                   4.1149                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.1150                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.1151                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.1152                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  Cl                                   4.1153                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  Cl                                   4.1154                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  Cl                                   4.1155                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.1156                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.1157                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.1158                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.1159                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.1160                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.1161                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  Cl                                   4.1162                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  Cl                                   4.1163                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  Cl                                   4.1164                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.1165                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.1166                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.1167                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.1168                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.1169                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.1170                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.1171                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.1172                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.1173                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR222##                                                                               H  Cl                                   4.1174                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR223##                                                                               H  Cl                                   4.1175                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR224##                                                                               H  Cl                                   4.1176                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR225##                                                                               H  Cl                                   4.1177                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR226##                                                                               H  Cl                                   4.1178                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR227##                                                                               H  Cl                                   4.1179                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.1180                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.1181                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.1182                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.1183                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.1184                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.1185                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.1186                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.1187                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.1188                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.1189                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.1190                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.1191                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.1192                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.1193                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.1194                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.1195                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.1196                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.1197                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.1198                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.1199                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.1200                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.1201                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.1202                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.1203                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.1204                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.1205                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.1206                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.1207                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.1208                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.1209                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.1210                                                                             CH.sub.3                                                                          H   H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.1211                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.1212                                                                             CH.sub.3                                                                          H   H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  Cl                                   4.1213                                                                             CH.sub.3                                                                          H   H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  Cl                                   4.1214                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  Cl                                   4.1215                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  Cl                                   4.1216                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O    H  Cl                                   4.1217                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  Cl                                   4.1218                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  Cl                                   4.1219                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                               H  Cl                                   4.1220                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.1221                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.1222                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOC.sub.2 H.sub.5                                                                        H  Cl                                   4.1223                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  Cl                                   4.1224                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  Cl                                   4.1225                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOiPr     H  Cl                                   4.1226                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.1227                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.1228                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.3                                                                          H  Cl                                   4.1229                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.1230                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.1231                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOC.sub.2 H.sub.5                                                                   H  Cl                                   4.1232                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  Cl                                   4.1233                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  Cl                                   4.1234                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOiPr                                                                               H  Cl                                   4.1235                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.1236                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.1237                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 CH═CHCl                                                              H  Cl                                   4.1238                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.1239                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.1240                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  Cl                                   4.1241                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.1242                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.1243                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3).sub.2                                                                         H  Cl                                   4.1244                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR228##                                                                               H  ClCl                                 4.1245                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR229##                                                                               H  Cl                                   4.1246                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR230##                                                                               H  Cl                                   4.1247                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR231##                                                                               H  Cl                                   4.1248                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR232##                                                                               H  Cl                                   4.1249                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H                                                                                  ##STR233##                                                                               H  Cl                                   4.1250                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.1251                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.1252                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--CH.sub.3                                                                         H  Cl                                   4.1253                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.1254                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.1255                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═NC.sub.2 H.sub.5                                                                    H  Cl                                   4.1256                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.1257                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.1258                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHCH.sub.3                                                                            H  Cl                                   4.1259                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.1260                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.1261                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHC.sub.2 H.sub.5                                                                     H  Cl                                   4.1262                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.1263                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.1264                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3).sub.2                                                                     H  Cl                                   4.1265                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.1266                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.1267                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--NHOC.sub.2 H.sub.5                                                                    H  Cl                                   4.1268                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.1269                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.1270                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H  Cl                                   4.1271                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.1272                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.1273                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--NH.sub.2                                                                         H  Cl                                   4.1274                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.1275                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.1276                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═N--N(CH.sub.3).sub.2                                                                H  Cl                                   4.1277                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.1278                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.1279                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H  Cl                                   4.1280                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.1281                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  1 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.1282                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C(CH.sub.3)--OCH.sub.3                                                                    H  Cl                                   4.1283                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  Cl                                   4.1284                                                                             CH.sub.3                                                                          CH.sub.3                                                                           H  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  O          H  Cl                                   __________________________________________________________________________

                                      TABLE 5                                      __________________________________________________________________________     Compounds of the formula                                                        ##STR234##                                                                    The radicals R.sup.12 of X and R7 of Y form a bond                             No.                                                                               R.sup.17                                                                          R.sup.18                                                                          R.sup.19                                                                          n  R.sup.21                                                                          R.sup.22                                                                           R.sup.13                                                                          Y     L M                                             __________________________________________________________________________     5.1                                                                               H  H  H  0  H  H   H  COCH.sub.3                                                                           H H                                             5.2                                                                               H  H  H  2  H  H   H  COCH.sub.3                                                                           H H                                             5.3                                                                               H  H  H  0  H  H   H  COC.sub.2 H.sub.5                                                                    H H                                             5.4                                                                               H  H  H  2  H  H   H  COC.sub.2 H.sub.5                                                                    H H                                             5.5                                                                               H  H  H  0  H  H   H  COiPr H H                                             5.6                                                                               H  H  H  2  H  H   H  COiPr H H                                             5.7                                                                               CH.sub.3                                                                          H  H  0  H  H   H  COCH.sub.3                                                                           H H                                             5.8                                                                               CH.sub.3                                                                          H  H  2  H  H   H  COCH.sub.3                                                                           H H                                             5.9                                                                               CH.sub.3                                                                          H  H  0  H  H   H  COC.sub.2 H.sub.5                                                                    H H                                             5.10                                                                              CH.sub.3                                                                          H  H  2  H  H   H  COC.sub.2 H.sub.5                                                                    H H                                             5.11                                                                              CH.sub.3                                                                          H  H  0  H  H   H  COiPr H H                                             5.12                                                                              CH.sub.3                                                                          H  H  2  H  H   H  COiPr H H                                             5.13                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0  H  H   H  COCH.sub.3                                                                           H H                                             5.14                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2  H  H   H  COCH.sub.3                                                                           H H                                             5.15                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0  H  H   H  COC.sub.2 H.sub.5                                                                    H H                                             5.16                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2  H  H   H  COC.sub.2 H.sub.5                                                                    H H                                             5.17                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0  H  H   H  COiPr H H                                             S.18                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2  H  H   H  COiPr H H                                             5.19                                                                              H  H  H  0  H  H   H  COCH.sub.3                                                                           H CH.sub.3                                      5.20                                                                              H  H  H  2  H  H   H  COCH.sub.3                                                                           H CH.sub.3                                      5.21                                                                              H  H  H  0  H  H   H  COC.sub.2 H.sub.5                                                                    H CH.sub.3                                      5.22                                                                              H  H  H  2  H  H   H  COC.sub.2 H.sub.5                                                                    H CH.sub.3                                      5.23                                                                              H  H  H  0  H  H   H  COiPr H CH.sub.3                                      5.24                                                                              H  H  H  2  H  H   H  COiPr H CH.sub.3                                      5.25                                                                              CH.sub.3                                                                          H  H  0  H  H   H  COCH.sub.3                                                                           H CH.sub.3                                      5.26                                                                              CH.sub.3                                                                          H  H  2  H  H   H  COCH.sub.3                                                                           H CH.sub.3                                      5.27                                                                              CH.sub.3                                                                          H  H  0  H  H   H  COC.sub.2 H.sub.5                                                                    H CH.sub.3                                      5.28                                                                              CH.sub.3                                                                          H  H  2  H  H   H  COC.sub.2 H.sub.5                                                                    H CH.sub.3                                      5.29                                                                              CH.sub.3                                                                          H  H  0  H  H   H  COiPr H CH.sub.3                                      5.30                                                                              CH.sub.3                                                                          H  H  2  H  H   H  COiPr H CH.sub.3                                      5.31                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0  H  H   H  COCH.sub.3                                                                           H CH.sub.3                                      5.32                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2  H  H   H  COCH.sub.3                                                                           H CH.sub.3                                      5.33                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0  H  H   H  COC.sub.2 H.sub.5                                                                    H CH.sub.3                                      5.34                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2  H  H   H  COC.sub.2 H.sub.5                                                                    H CH.sub.3                                      5.35                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0  H  H   H  COiPr H CH.sub.3                                      5.36                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2  H  H   H  COiPr H CH.sub.3                                      5.37                                                                              H  H  H  0  H  H   H  COCH.sub.3                                                                           H Cl                                            5.38                                                                              H  H  H  2  H  H   H  COCH.sub.3                                                                           H Cl                                            5.39                                                                              H  H  H  0  H  H   H  COC.sub.2 H.sub.5                                                                    H Cl                                            5.40                                                                              H  H  H  2  H  H   H  COC.sub.2 H.sub.5                                                                    H Cl                                            5.41                                                                              H  H  H  0  H  H   H  COiPr H Cl                                            5.42                                                                              H  H  H  2  H  H   H  COiPr H Cl                                            5.43                                                                              CH.sub.3                                                                          H  H  0  H  H   H  COCH.sub.3                                                                           H Cl                                            5.44                                                                              CH.sub.3                                                                          H  H  2  H  H   H  COCH.sub.3                                                                           H Cl                                            5.45                                                                              CH.sub.3                                                                          H  H  0  H  H   H  COC.sub.2 H.sub.5                                                                    H Cl                                            5.46                                                                              CH.sub.3                                                                          H  H  2  H  H   H  COC.sub.2 H.sub.5                                                                    H Cl                                            5.47                                                                              CH.sub.3                                                                          H  H  0  H  H   H  COiPr H Cl                                            5.48                                                                              CH.sub.3                                                                          H  H  2  H  H   H  COiPr H Cl                                            5.49                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0  H  H   H  COCH.sub.3                                                                           H Cl                                            5.50                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2  H  H   H  COCH.sub.3                                                                           H Cl                                            5.51                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0  H  H   H  COC.sub.2 H.sub.5                                                                    H Cl                                            5.52                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2  H  H   H  COC.sub.2 H.sub.5                                                                    H Cl                                            5.53                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0  H  H   H  COiPr H Cl                                            5.54                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2  H  H   H  COiPr H Cl                                            __________________________________________________________________________

                                      TABLE 6                                      __________________________________________________________________________     Compounds of the formula                                                        ##STR235##                                                                    No.                                                                               R.sup.17                                                                          R.sup.18                                                                          R.sup.19                                                                          n R.sup.21                                                                          R.sup.22                                                                          R.sup.12                                                                          R.sup.13                                                                          Y          M L                                       __________________________________________________________________________     6.1                                                                               H  H  H  0 H  H  H  H  C═O    H CH.sub.3                                6.2                                                                               H  H  H  1 H  H  H  H  C═O    H CH.sub.3                                6.3                                                                               H  H  H  2 H  H  H  H  C═O    H CH.sub.3                                6.4                                                                               H  H  H  0 H  H  H  H  CH--OCH.sub.3                                                                             H CH.sub.3                                6.5                                                                               H  H  H  1 H  H  H  H  CH--OCH.sub.3                                                                             H CH.sub.3                                6.6                                                                               H  H  H  2 H  H  H  H  CH--OCH.sub.3                                                                             H CH.sub.3                                6.7                                                                               H  H  H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                6.8                                                                               H  H  H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                6.9                                                                               H  H  H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                6.10                                                                              H  H  H  0 H  H  H  H  CHOiPr     H CH.sub.3                                6.11                                                                              H  H  H  1 H  H  H  H  CHOiPr     H CH.sub.3                                6.12                                                                              H  H  H  2 H  H  H  H  CHOiPr     H CH.sub.3                                6.13                                                                              H  H  H  0 H  H  H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                6.14                                                                              H  H  H  1 H  H  H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                6.15                                                                              H  H  H  2 H  H  H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                6.16                                                                              H  H  H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                6.17                                                                              H  H  H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                6.18                                                                              H  H  H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                6.19                                                                              H  H  H  0 H  H  H  H  C═NOiPr                                                                               H CH.sub.3                                6.20                                                                              H  H  H  1 H  H  H  H  C═NOiPr                                                                               H CH.sub.3                                6.21                                                                              H  H  H  2 H  H  H  H  C═NOiPr                                                                               H CH.sub.3                                6.22                                                                              H  H  H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                6.23                                                                              H  H  H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                6.24                                                                              H  H  H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                6.25                                                                              H  H  H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                6.26                                                                              H  H  H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                6.27                                                                              H  H  H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                6.28                                                                              H  H  H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                6.29                                                                              H  H  H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                6.30                                                                              H  H  H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                6.31                                                                              H  H  H  0 H  H  H  H                                                                                  ##STR236##                                                                               H CH.sub.3                                6.32                                                                              H  H  H  1 H  H  H  H                                                                                  ##STR237##                                                                               H CH.sub.3                                6.33                                                                              H  H  H  2 H  H  H  H                                                                                  ##STR238##                                                                               H CH.sub.3                                6.34                                                                              H  H  H  0 H  H  H  H                                                                                  ##STR239##                                                                               H CH.sub.3                                6.35                                                                              H  H  H  1 H  H  H  H                                                                                  ##STR240##                                                                               H CH.sub.3                                6.36                                                                              H  H  H  2 H  H  H  H                                                                                  ##STR241##                                                                               H CH.sub.3                                6.37                                                                              H  H  H  0 H  H  H  H  C═N--CH.sub.3                                                                         H CH.sub.3                                6.38                                                                              H  H  H  1 H  H  H  H  C═N--CH.sub.3                                                                         H CH.sub.3                                6.39                                                                              H  H  H  2 H  H  H  H  C═N--CH.sub.3                                                                         H CH.sub.3                                6.40                                                                              H  H  H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.41                                                                              H  H  H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.42                                                                              H  H  H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.43                                                                              H  H  H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H CH.sub.3                                6.44                                                                              H  H  H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H CH.sub.3                                6.45                                                                              H  H  H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H CH.sub.3                                6.46                                                                              H  H  H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                6.47                                                                              H  H  H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                6.48                                                                              H  H  H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                6.49                                                                              H  H  H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                6.50                                                                              H  H  H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                6.51                                                                              H  H  H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                6.52                                                                              H  H  H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.53                                                                              H  H  H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.54                                                                              H  H  H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.55                                                                              H  H  H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                6.56                                                                              H  H  H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                6.57                                                                              H  H  H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                6.58                                                                              H  H  H  0 H  H  H  H  C═N--NH.sub.2                                                                         H CH.sub.3                                6.59                                                                              H  H  H  1 H  H  H  H  C═N--NH.sub.2                                                                         H CH.sub.3                                6.60                                                                              H  H  H  2 H  H  H  H  C═N--NH.sub.2                                                                         H CH.sub.3                                6.61                                                                              H  H  H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                6.62                                                                              H  H  H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                6.63                                                                              H  H  H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                6.64                                                                              H  H  H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                6.65                                                                              H  H  H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                6.66                                                                              H  H  H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                6.67                                                                              H  H  H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                6.68                                                                              H  H  H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                6.69                                                                              H  H  H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                6.70                                                                              H  H  H  0 H  H  H  H  O          H CH.sub.3                                6.71                                                                              H  H  H  1 H  H  H  H  O          H CH.sub.3                                6.72                                                                              H  H  H  2 H  H  H  H  O          H CH.sub.3                                6.73                                                                              CH.sub.3                                                                          H  H  0 H  H  H  H  C═O    H CH.sub.3                                6.74                                                                              CH.sub.3                                                                          H  H  1 H  H  H  H  C═O    H CH.sub.3                                6.75                                                                              CH.sub.3                                                                          H  H  2 H  H  H  H  C═O    H CH.sub.3                                6.76                                                                              CH.sub.3                                                                          H  H  0 H  H  H  H  CHOCH.sub.3                                                                               H CH.sub.3                                6.77                                                                              CH.sub.3                                                                          H  H  1 H  H  H  H  CHOCH.sub.3                                                                               H CH.sub.3                                6.78                                                                              CH.sub.3                                                                          H  H  2 H  H  H  H  CHOCH.sub.3                                                                               H CH.sub.3                                6.79                                                                              CH.sub.3                                                                          H  H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                6.80                                                                              CH.sub.3                                                                          H  H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                6.81                                                                              CH.sub.3                                                                          H  H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                6.82                                                                              CH.sub.3                                                                          H  H  0 H  H  H  H  CHOiPr     H CH.sub.3                                6.83                                                                              CH.sub.3                                                                          H  H  1 H  H  H  H  CHOiPr     H CH.sub.3                                6.84                                                                              CH.sub.3                                                                          H  H  2 H  H  H  H  CHOiPr     H CH.sub.3                                6.85                                                                              CH.sub.3                                                                          H  H  0 H  H  H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                6.86                                                                              CH.sub.3                                                                          H  H  1 H  H  H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                6.87                                                                              CH.sub.3                                                                          H  H  2 H  H  H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                6.88                                                                              CH.sub.3                                                                          H  H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                6.89                                                                              CH.sub.3                                                                          H  H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                6.90                                                                              CH.sub.3                                                                          H  H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                6.91                                                                              CH.sub.3                                                                          H  H  0 H  H  H  H  C═NOiPr                                                                               H CH.sub.3                                6.92                                                                              CH.sub.3                                                                          H  H  1 H  H  H  H  C═NOiPr                                                                               H CH.sub.3                                6.93                                                                              CH.sub.3                                                                          H  H  2 H  H  H  H  C═NOiPr                                                                               H CH.sub.3                                6.94                                                                              CH.sub.3                                                                          H  H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                6.95                                                                              CH.sub.3                                                                          H  H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                6.96                                                                              CH.sub.3                                                                          H  H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                6.97                                                                              CH.sub.3                                                                          H  H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                6.98                                                                              CH.sub.3                                                                          H  H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                6.99                                                                              CH.sub.3                                                                          H  H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                6.100                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                6.101                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                6.102                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                6.103                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H                                                                                  ##STR242##                                                                               H CH.sub.3                                6.104                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H                                                                                  ##STR243##                                                                               H CH.sub.3                                6.105                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H                                                                                  ##STR244##                                                                               H CH.sub.3                                6.106                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H                                                                                  ##STR245##                                                                               H CH.sub.3                                6.107                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H                                                                                  ##STR246##                                                                               H CH.sub.3                                6.108                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H                                                                                  ##STR247##                                                                               H CH.sub.3                                6.109                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═N--CH.sub.3                                                                         H CH.sub.3                                6.110                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═N--CH.sub.3                                                                         H CH.sub.3                                6.111                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═N--CH.sub.3                                                                         H CH.sub.3                                6.112                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.113                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.114                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.115                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H CH.sub.3                                6.116                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H CH.sub.3                                6.117                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H CH.sub.3                                6.118                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                6.119                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                6.120                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                6.121                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                6.122                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                6.123                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                6.124                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.125                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.126                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.127                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                6.128                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                6.129                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                6.130                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═N--NH.sub.2                                                                         H CH.sub.3                                6.131                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═N--NH.sub.2                                                                         H CH.sub.3                                6.132                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═N--NH.sub.2                                                                         H CH.sub.3                                6.133                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                6.134                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                6.135                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                6.136                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                6.137                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                6.138                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                6.139                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                6.140                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                6.141                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                6.142                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  O          H CH.sub.3                                6.143                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  O          H CH.sub.3                                6.144                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  O          H CH.sub.3                                6.145                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═O    H CH.sub.3                                6.146                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═O    H CH.sub.3                                6.147                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═O    H CH.sub.3                                6.148                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CHOCH.sub.3                                                                               H CH.sub.3                                6.149                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CHOCH.sub.3                                                                               H CH.sub.3                                6.150                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CHOCH.sub.3                                                                               H CH.sub.3                                6.151                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                6.152                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                6.153                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                6.154                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CHOiPr     H CH.sub.3                                6.155                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CHOiPr     H CH.sub.3                                6.156                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CHOiPr     H CH.sub.3                                6.157                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                6.158                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                6.159                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NOCH.sub.3                                                                          H CH.sub.3                                6.160                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                6.161                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                6.162                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                6.163                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NOiPr                                                                               H CH.sub.3                                6.164                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NOiPr                                                                               H CH.sub.3                                6.165                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NOiPr                                                                               H CH.sub.3                                6.166                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                6.167                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                6.168                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                6.169                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                6.170                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                6.171                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                6.172                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                6.173                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                6.174                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H CH.sub.3                                6.175                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H                                                                                  ##STR248##                                                                               H CH.sub.3                                6.176                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H                                                                                  ##STR249##                                                                               H CH.sub.3                                6.177                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H                                                                                  ##STR250##                                                                               H CH.sub.3                                6.178                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H                                                                                  ##STR251##                                                                               H CH.sub.3                                6.179                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H                                                                                  ##STR252##                                                                               H CH.sub.3                                6.180                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H                                                                                  ##STR253##                                                                               H CH.sub.3                                6.181                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═N--CH.sub.3                                                                         H CH.sub.3                                6.182                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═N--CH.sub.3                                                                         H CH.sub.3                                6.183                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═N--CH.sub.3                                                                         H CH.sub.3                                6.184                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.185                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.186                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.187                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H CH.sub.3                                6.188                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H CH.sub.3                                6.189                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H CH.sub.3                                6.190                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                6.191                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                6.192                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                6.193                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                6.194                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                6.195                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                6.196                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.197                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.198                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                6.199                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                6.200                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                6.201                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                6.202                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═N--NH.sub.2                                                                         H CH.sub.3                                6.203                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═N--NH.sub.2                                                                         H CH.sub.3                                6.204                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═N--NH.sub.2                                                                         H CH.sub.3                                6.205                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                6.206                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                6.207                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                6.208                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                6.209                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                6.210                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                6.211                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                6.212                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                6.213                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C(CH.sub.3)--OCh.sub.3                                                                    H CH.sub.3                                6.214                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  O          H CH.sub.3                                6.215                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  O          H CH.sub.3                                6.216                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  O          H CH.sub.3                                6.217                                                                             H  H  H  0 H  H  H  H  C═O    H Cl                                      6.218                                                                             H  H  H  1 H  H  H  H  C═O    H Cl                                      6.219                                                                             H  H  H  2 H  H  H  H  C═O    H Cl                                      6.220                                                                             H  H  H  0 H  H  H  H  CHOCH.sub.3                                                                               H Cl                                      6.221                                                                             H  H  H  1 H  H  H  H  CHOCH.sub.3                                                                               H Cl                                      6.222                                                                             H  H  H  2 H  H  H  H  CHOCH.sub.3                                                                               H Cl                                      6.223                                                                             H  H  H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                      6.224                                                                             H  H  H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                      6.225                                                                             H  H  H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                      6.226                                                                             H  H  H  0 H  H  H  H  CHOiPr     H Cl                                      6.227                                                                             H  H  H  1 H  H  H  H  CHOiPr     H Cl                                      6.228                                                                             H  H  H  2 H  H  H  H  CHOiPr     H Cl                                      6.229                                                                             H  H  H  0 H  H  H  H  C═NOCH.sub.3                                                                          H Cl                                      6.230                                                                             H  H  H  1 H  H  H  H  C═NOCH.sub.3                                                                          H Cl                                      6.231                                                                             H  H  H  2 H  H  H  H  C═NOCH.sub.3                                                                          H Cl                                      6.232                                                                             H  H  H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                      6.233                                                                             H  H  H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                      6.234                                                                             H  H  H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                      6.235                                                                             H  H  H  0 H  H  H  H  C═NOiPr                                                                               H Cl                                      6.236                                                                             H  H  H  1 H  H  H  H  C═NOiPr                                                                               H Cl                                      6.237                                                                             H  H  H  2 H  H  H  H  C═NOiPr                                                                               H Cl                                      6.238                                                                             H  H  H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                      6.239                                                                             H  H  H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                      6.240                                                                             H  H  H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                      6.241                                                                             H  H  H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                      6.242                                                                             H  H  H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                      6.243                                                                             H  H  H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                      6.244                                                                             H  H  H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H Cl                                      6.245                                                                             H  H  H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H Cl                                      6.246                                                                             H  H  H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H Cl                                      6.247                                                                             H  H  H  0 H  H  H  H                                                                                  ##STR254##                                                                               H Cl                                      6.248                                                                             H  H  H  1 H  H  H  H                                                                                  ##STR255##                                                                               H Cl                                      6.249                                                                             H  H  H  2 H  H  H  H                                                                                  ##STR256##                                                                               H Cl                                      6.250                                                                             H  H  H  0 H  H  H  H                                                                                  ##STR257##                                                                               H Cl                                      6.251                                                                             H  H  H  1 H  H  H  H                                                                                  ##STR258##                                                                               H Cl                                      6.252                                                                             H  H  H  2 H  H  H  H                                                                                  ##STR259##                                                                               H Cl                                      6.253                                                                             H  H  H  0 H  H  H  H  C═N--CH.sub.3                                                                         H Cl                                      6.254                                                                             H  H  H  1 H  H  H  H  C═N--CH.sub.3                                                                         H Cl                                      6.255                                                                             H  H  H  2 H  H  H  H  C═N--CH.sub.3                                                                         H Cl                                      6.256                                                                             H  H  H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H Cl                                      6.257                                                                             H  H  H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H Cl                                      6.258                                                                             H  H  H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H Cl                                      6.259                                                                             H  H  H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H Cl                                      6.260                                                                             H  H  H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H Cl                                      6.261                                                                             H  H  H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H Cl                                      6.262                                                                             H  H  H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H Cl                                      6.263                                                                             H  H  H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H Cl                                      6.264                                                                             H  H  H  2 H  H  H  H  CH--NHC.sub.2 H5                                                                          H Cl                                      6.265                                                                             H  H  H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H Cl                                      6.266                                                                             H  H  H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H Cl                                      6.267                                                                             H  H  H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H Cl                                      6.268                                                                             H  H  H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H Cl                                      6.269                                                                             H  H  H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H Cl                                      6.270                                                                             H  H  H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H Cl                                      6.271                                                                             H  H  H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H Cl                                      6.272                                                                             H  H  H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H Cl                                      6.273                                                                             H  H  H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H Cl                                      6.274                                                                             H  H  H  0 H  H  H  H  C═N--NH.sub.2                                                                         H Cl                                      6.275                                                                             H  H  H  1 H  H  H  H  C═N--NH.sub.2                                                                         H Cl                                      6.276                                                                             H  H  H  2 H  H  H  H  C═N--NH.sub.2                                                                         H Cl                                      6.277                                                                             H  H  H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H Cl                                      6.278                                                                             H  H  H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H Cl                                      6.279                                                                             H  H  H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H Cl                                      6.280                                                                             H  H  H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H Cl                                      6.281                                                                             H  H  H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H Cl                                      6.282                                                                             H  H  H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H Cl                                      6.283                                                                             H  H  H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H Cl                                      6.284                                                                             H  H  H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H Cl                                      6.285                                                                             H  H  H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H Cl                                      6.286                                                                             H  H  H  0 H  H  H  H  O          H Cl                                      6.287                                                                             H  H  H  1 H  H  H  H  O          H Cl                                      6.288                                                                             H  H  H  2 H  H  H  H  O          H Cl                                      6.289                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═O    H Cl                                      6.290                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═O    H Cl                                      6.291                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═O    H Cl                                      6.292                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CHOCH.sub.3                                                                               H Cl                                      6.293                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CHOCH.sub.3                                                                               H Cl                                      6.294                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CHOCH.sub.3                                                                               H Cl                                      6.295                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                      6.296                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                      6.297                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                      6.298                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CHOiPr     H Cl                                      6.299                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CHOiPr     H Cl                                      6.300                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CHOiPr     H Cl                                      6.301                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═NOCH.sub.3                                                                          H Cl                                      6.302                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═NOCH.sub.3                                                                          H Cl                                      6.303                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═NOCH.sub.3                                                                          H Cl                                      6.304                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                      6.305                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                      6.306                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                      6.307                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═NOiPr                                                                               H Cl                                      6.308                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═NOiPr                                                                               H Cl                                      6.309                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═NOiPr                                                                               H Cl                                      6.310                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                      6.311                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                      6.312                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                      6.313                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                      6.314                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                      6.315                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                      6.316                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H Cl                                      6.317                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H Cl                                      6.318                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H Cl                                      6.319                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H                                                                                  ##STR260##                                                                               H Cl                                      6.320                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H                                                                                  ##STR261##                                                                               H Cl                                      6.321                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H                                                                                  ##STR262##                                                                               H Cl                                      6.322                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H                                                                                  ##STR263##                                                                               H Cl                                      6.323                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H                                                                                  ##STR264##                                                                               H Cl                                      6.324                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H                                                                                  ##STR265##                                                                               H Cl                                      6.325                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═N--CH.sub.3                                                                         H Cl                                      6.326                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═N--CH.sub.3                                                                         H Cl                                      6.327                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═N--CH.sub.3                                                                         H Cl                                      6.328                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H Cl                                      6.329                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H Cl                                      6.330                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H Cl                                      6.331                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H Cl                                      6.332                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H Cl                                      6.333                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H Cl                                      6.334                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H Cl                                      6.335                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H Cl                                      6.336                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H Cl                                      6.337                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H Cl                                      6.338                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H Cl                                      6.339                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H Cl                                      6.340                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H Cl                                      6.341                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H Cl                                      6.342                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H Cl                                      6.343                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H Cl                                      6.344                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H Cl                                      6.345                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H Cl                                      6.346                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═N--NH.sub.2                                                                         H Cl                                      6.347                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═N--NH.sub.2                                                                         H Cl                                      6.348                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═N--NH.sub.2                                                                         H Cl                                      6.349                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H Cl                                      6.350                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H Cl                                      6.351                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H Cl                                      6.352                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H Cl                                      6.353                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H Cl                                      6.354                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H Cl                                      6.355                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H Cl                                      6.356                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H Cl                                      6.357                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H Cl                                      6.358                                                                             CH.sub.3                                                                          H  H  0 H  H  H  H  O          H Cl                                      6.359                                                                             CH.sub.3                                                                          H  H  1 H  H  H  H  O          H Cl                                      6.360                                                                             CH.sub.3                                                                          H  H  2 H  H  H  H  O          H Cl                                      6.361                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═O    H Cl                                      6.362                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═O    H Cl                                      6.363                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═O    H Cl                                      6.364                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CHOCH.sub.3                                                                               H Cl                                      6.365                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CHOCH.sub.3                                                                               H Cl                                      6.366                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CHOCH.sub.3                                                                               H Cl                                      6.367                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                      6.368                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                      6.369                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CHOC.sub.2 H.sub.5                                                                        H Cl                                      6.370                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CHOiPr     H Cl                                      6.371                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CHOiPr     H Cl                                      6.372                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CHOiPr     H Cl                                      6.373                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NOCH.sub.3                                                                          H Cl                                      6.374                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NOCH.sub.3                                                                          H Cl                                      6.375                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NOCH.sub.3                                                                          H Cl                                      6.376                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                      6.377                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                      6.378                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NOC.sub.2 H.sub.5                                                                   H Cl                                      6.379                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NOiPr                                                                               H Cl                                      6.380                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NOiPr                                                                               H Cl                                      6.381                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NOiPr                                                                               H Cl                                      6.382                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                      6.383                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                      6.384                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NOCH.sub.2 CH═CHCl                                                              H Cl                                      6.385                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                      6.386                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                      6.387                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H Cl                                      6.388                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C(CH.sub.3).sub.2                                                                         H Cl                                      6.389                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C(CH.sub.3).sub.2                                                                         H Cl                                      6.390                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C(CH.sub.3).sub.2                                                                         H Cl                                      6.391                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H                                                                                  ##STR266##                                                                               H Cl                                      6.392                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H                                                                                  ##STR267##                                                                               H Cl                                      6.393                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H                                                                                  ##STR268##                                                                               H Cl                                      6.394                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H                                                                                  ##STR269##                                                                               H Cl                                      6.395                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H                                                                                  ##STR270##                                                                               H Cl                                      6.396                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H                                                                                  ##STR271##                                                                               H Cl                                      6.397                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═N--CH.sub.3                                                                         H Cl                                      6.398                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═N--CH.sub.3                                                                         H Cl                                      6.399                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═N--CH.sub.3                                                                         H Cl                                      6.400                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H Cl                                      6.401                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H Cl                                      6.402                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═NC.sub.2 H.sub.5                                                                    H Cl                                      6.403                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--NHCH.sub.3                                                                            H Cl                                      6.404                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--NHCH.sub.3                                                                            H Cl                                      6.405                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--NHCH.sub.3                                                                            H Cl                                      6.406                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H Cl                                      6.407                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H Cl                                      6.408                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--NHC.sub.2 H.sub.5                                                                     H Cl                                      6.409                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H Cl                                      6.410                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--N(Cf3)2                                                                               H Cl                                      6.411                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--N(CH.sub.3).sub.2                                                                     H Cl                                      6.412                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H Cl                                      6.413                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H Cl                                      6.414                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--NHOC.sub.2 H.sub.5                                                                    H Cl                                      6.415                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H Cl                                      6.416                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H Cl                                      6.417                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H Cl                                      6.418                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═N--NH.sub.2                                                                         H Cl                                      6.419                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═N--NH.sub.2                                                                         H Cl                                      6.420                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═N--NH.sub.2                                                                         H Cl                                      6.421                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H Cl                                      6.422                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H Cl                                      6.423                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C═N--N(CH.sub.3).sub.2                                                                H Cl                                      6.424                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H Cl                                      6.425                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H Cl                                      6.426                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H Cl                                      6.427                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H Cl                                      6.428                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H Cl                                      6.429                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  C(CH.sub.3)--OCH.sub.3                                                                    H Cl                                      6.430                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H  H  H  O          H Cl                                      6.431                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H  H  H  O          H Cl                                      6.432                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H  H  H  O          H Cl                                      __________________________________________________________________________

                  TABLE 7                                                          ______________________________________                                         Compounds of the formula                                                        ##STR272##                                                                    The radicals R.sup.7 and R.sup.23 form a bond.                                 No.  R.sup.17                                                                               R.sup.18                                                                              R.sup.19                                                                             n    Y      L    M                                   ______________________________________                                         7.1  H       H      H     2    COCH.sub.3                                                                            H    H                                   7.2  H       H      H     2    COC.sub.2 H.sub.5                                                                     H    H                                   7.3  CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            H    H                                   7.4  CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     H    H                                   7.5  CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            H    H                                   7.6  CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     H    H                                   7.7  H       H      H     2    COCH.sub.3                                                                            H    CH.sub.3                            7.8  H       H      H     2    COC.sub.2 H.sub.5                                                                     H    CH.sub.3                            7.9  CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            H    CH.sub.3                            7.10 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     H    CH.sub.3                            7.11 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            H    CH.sub.3                            7.12 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     H    CH.sub.3                            7.13 H       H      H     2    COCH.sub.3                                                                            H    Cl                                  7.14 H       H      H     2    COC.sub.2 H.sub.5                                                                     H    Cl                                  7.15 CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            H    Cl                                  7.16 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     H    Cl                                  7.17 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            H    Cl                                  7.18 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     H    Cl                                  7.19 H       H      H     2    COCH.sub.3                                                                            H    NO.sub.2                            7.20 H       H      H     2    COC.sub.2 H.sub.5                                                                     H    NO.sub.2                            7.21 CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            H    NO.sub.2                            7.22 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     H    NO.sub.2                            7.23 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            H    NO.sub.2                            7.24 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     H    NO.sub.2                            7.25 H       H      H     2    COCH.sub.3                                                                            H    SO.sub.2 CH.sub.3                   7.26 H       H      H     2    COC.sub.2 H.sub.5                                                                     H    SO.sub.2 CH.sub.3                   7.27 CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            H    SO.sub.2 CH.sub.3                   7.28 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     H    SO.sub.2 CH.sub.3                   7.29 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            H    SO.sub.2 CH.sub.3                   7.30 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     H    SO.sub.2 CH.sub.3                   7.31 H       H      H     2    COCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                            7.32 H       H      H     2    COC.sub.2 H.sub.5                                                                     CH.sub.3                                                                            CH.sub.3                            7.33 CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                            7.34 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     CH.sub.3                                                                            CH.sub.3                            7.35 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                            7.36 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     CH.sub.3                                                                            CH.sub.3                            7.37 H       H      H     2    COCH.sub.3                                                                            Cl   Cl                                  7.38 H       H      H     2    COC.sub.2 H.sub.5                                                                     Cl   Cl                                  7.39 CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            Cl   Cl                                  7.40 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     Cl   Cl                                  7.41 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            Cl   Cl                                  7.42 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     Cl   Cl                                  ______________________________________                                    

                  TABLE 8                                                          ______________________________________                                         Compounds of the formula                                                        ##STR273##                                                                    No.  R.sup.17                                                                               R.sup.18                                                                              R.sup.19                                                                             n    Y      M    L                                   ______________________________________                                         8.1  H       H      H     2    COCH.sub.3                                                                            H    CH.sub.3                            8.2  H       H      H     2    COC.sub.2 H.sub.5                                                                     H    CH.sub.3                            8.3  CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            H    CH.sub.3                            8.4  CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     H    CH.sub.3                            8.5  CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            H    CH.sub.3                            8.6  CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     H    CH.sub.3                            8.7  H       H      H     2    COCH.sub.3                                                                            H    Cl                                  8.8  H       H      H     2    COC.sub.2 H.sub.5                                                                     H    Cl                                  8.9  CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            H    Cl                                  8.10 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     H    Cl                                  8.11 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            H    Cl                                  8.12 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     H    Cl                                  8.13 H       H      H     2    COCH.sub.3                                                                            H    NO.sub.2                            8.14 H       H      H     2    COC.sub.2 H.sub.5                                                                     H    NO.sub.2                            8.15 CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            H    NO.sub.2                            8.16 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     H    NO.sub.2                            8.17 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            H    NO.sub.2                            8.18 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     H    NO.sub.2                            8.19 H       H      H     2    COCH.sub.3                                                                            H    SO.sub.2 CH.sub.3                   8.20 H       H      H     2    COC.sub.2 H.sub.5                                                                     H    SO.sub.2 CH.sub.3                   8.21 CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            H    SO.sub.2 CH.sub.3                   8.22 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     H    SO.sub.2 CH.sub.3                   8.23 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            H    SO.sub.2 CH.sub.3                   8.24 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     H    SO.sub.2 CH.sub.3                   8.25 H       H      H     2    COCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                            8.26 H       H      H     2    COC.sub.2 H.sub.5                                                                     CH.sub.3                                                                            CH.sub.3                            8.27 CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                            8.28 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     CH.sub.3                                                                            CH.sub.3                            8.29 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                            8.30 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     CH.sub.3                                                                            CH.sub.3                            8.31 H       H      H     2    COCH.sub.3                                                                            Cl   Cl                                  8.32 H       H      H     2    COC.sub.2 H.sub.5                                                                     Cl   Cl                                  8.33 CH.sub.3                                                                               H      H     2    COCH.sub.3                                                                            Cl   Cl                                  8.34 CH.sub.3                                                                               H      H     2    COC.sub.2 H.sub.5                                                                     Cl   Cl                                  8.35 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COCH.sub.3                                                                            Cl   Cl                                  8.36 CH.sub.3                                                                               CH.sub.3                                                                              H     2    COC.sub.2 H.sub.5                                                                     Cl   Cl                                  ______________________________________                                    

                                      TABLE 9                                      __________________________________________________________________________     Compounds of the formula                                                        ##STR274##                                                                    No.                                                                               R.sup.15                                                                          R.sup.16                                                                           R.sup.19                                                                          n  X   Y           M L                                            __________________________________________________________________________     9.1                                                                               CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           C═O     H CH.sub.3                                     9.2                                                                               CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   C═O     H CH.sub.3                                     9.3                                                                               CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   C═O     H CH.sub.3                                     9.4                                                                               CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           CHOCH.sub.3 H CH.sub.3                                     9.5                                                                               CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   CHOCH.sub.3 H CH.sub.3                                     9.6                                                                               CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   CHOCH.sub.3 H CH.sub.3                                     9.7                                                                               CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           CHOC.sub.2 H.sub.5                                                                         H CH.sub.3                                     9.8                                                                               CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                         H CH.sub.3                                     9.9                                                                               CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                         H CH.sub.3                                     9.10                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           CHOiPr      H CH.sub.3                                     9.11                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   CHOiPr      H CH.sub.3                                     9.12                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   CHOiPr      H CH.sub.3                                     9.13                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           C═NOCH.sub.3                                                                           H CH.sub.3                                     9.14                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                           H CH.sub.3                                     9.15                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                           H CH.sub.3                                     9.16                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           C═NOC.sub.2 H.sub.5                                                                    H CH.sub.3                                     9.17                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                    H CH.sub.3                                     9.18                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                    H CH.sub.3                                     9.19                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           C═NOiPr H CH.sub.3                                     9.20                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   C═NOiPr H CH.sub.3                                     9.21                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   C═NOiPr H CH.sub.3                                     9.22                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           C═NOCH.sub.2 CH═CHCl                                                               H CH.sub.3                                     9.23                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   C═NOCH.sub.2 CH═CHCl                                                               H CH.sub.3                                     9.24                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   C═NOCH.sub.2 CH═CHCl                                                               H CH.sub.3                                     9.25                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           C═NOCH.sub.2 C.sub.6 H.sub.5                                                           H CH.sub.3                                     9.26                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   C═NOCH.sub.2 C.sub.6 H.sub.5                                                           H CH.sub.3                                     9.27                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   C═NOCH.sub.2 C.sub.6 H.sub.5                                                           H CH.sub.3                                     9.28                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           C(CH.sub.3).sub.2                                                                          H CH.sub.3                                     9.29                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   C(CH.sub.3).sub.2                                                                          H CH.sub.3                                     9.30                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   C(CH.sub.3).sub.2                                                                          H CH.sub.3                                     9.31                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                            ##STR275## H CH.sub.3                                     9.32                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                    ##STR276## H CH.sub.3                                     9.33                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                    ##STR277## H CH.sub.3                                     9.34                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                            ##STR278## H CH.sub.3                                     9.35                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                    ##STR279## H CH.sub.3                                     9.36                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                    ##STR280## H CH.sub.3                                     9.37                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           CH--NHCH.sub.3                                                                             H CH.sub.3                                     9.38                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   CH--NHCH.sub.3                                                                             H CH.sub.3                                     9.39                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   CH--NHCH.sub.3                                                                             H CH.sub.3                                     9.40                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           CH--NHC.sub.2 H.sub.5                                                                      H CH.sub.3                                     9.41                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   CH--NHC.sub.2 H.sub.5                                                                      H CH.sub.3                                     9.42                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   CH--NHC.sub.2 H.sub.5                                                                      H CH.sub.3                                     9.43                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           CH--N(CH.sub.3).sub.2                                                                      H CH.sub.3                                     9.44                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3).sub.2                                                                      H CH.sub.3                                     9.45                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3).sub.2                                                                      H CH.sub.3                                     9.46                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           CH--NHOC.sub.2 H.sub.5                                                                     H CH.sub.3                                     9.47                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   CH--NHOC.sub.2 H.sub.5                                                                     H CH.sub.3                                     9.48                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   CH--NHOC.sub.2 H.sub.5                                                                     H CH.sub.3                                     9.49                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                            H CH.sub.3                                     9.50                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                            H CH.sub.3                                     9.51                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                            H CH.sub.3                                     9.52                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           C═N--NH.sub.2                                                                          H CH.sub.3                                     9.53                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   C═N--NH.sub.2                                                                          H CH.sub.3                                     9.54                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   C═N--NH.sub.2                                                                          H CH.sub.3                                     9.55                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           C═N--N(CH.sub.3).sub.2                                                                 H CH.sub.3                                     9.56                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   C═N--N(CH.sub.3).sub.2                                                                 H CH.sub.3                                     9.57                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   C═N--N(CH.sub.3).sub.2                                                                 H CH.sub.3                                     9.58                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                   H CH.sub.3                                     9.59                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                   H CH.sub.3                                     9.60                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                   H CH.sub.3                                     9.61                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           C(CH.sub.3)--OCH.sub.3                                                                     H CH.sub.3                                     9.62                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   C(CH.sub.3)--OCH.sub.3                                                                     H CH.sub.3                                     9.63                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   C(CH.sub.3)--OCH.sub.3                                                                     H CH.sub.3                                     9.64                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  CH.sub.2                                                                           O           H CH.sub.3                                     9.65                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  2  (CH.sub.2).sub.2                                                                   O           H CH.sub.3                                     9.66                                                                              CH.sub.3                                                                          CH.sub.3                                                                           H  0  (CH.sub.2).sub.2                                                                   O           H CH.sub.3                                     9.67                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Br 2  CH.sub.2                                                                           CHOCH.sub.3 H CH.sub.3                                     9.68                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Br 2  (CH.sub.2).sub.2                                                                   CHOCH.sub.3 H CH.sub.3                                     9.69                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Br 0  (CH.sub.2).sub.2                                                                   CHOCH.sub.3 H CH.sub.3                                     9.70                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Br 2  CH.sub.2                                                                           CHOC.sub.2 H.sub.5                                                                         H CH.sub.3                                     9.71                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Br 2  (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                         H CH.sub.3                                     9.72                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Br 0  (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                         H CH.sub.3                                     9.73                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Br 2  CH.sub.2                                                                           CHOiPr      H CH.sub.3                                     9.74                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Brr                                                                               2  (CH.sub.2).sub.2                                                                   CHOiPr      H CH.sub.3                                               [sic]                                                                9.75                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Br 0  (CH.sub.2).sub.2                                                                   CHOiPr      H CH.sub.3                                     9.76                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Cl 2  CH.sub.2                                                                           CHOCH.sub.3 H CH.sub.3                                     9.77                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Cl 2  (CH.sub.2).sub.2                                                                   CHOCH.sub.3 H CH.sub.3                                     9.78                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Cl 0  (CH.sub.2).sub.2                                                                   CHOCH.sub.3 H CH.sub.3                                     9.79                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Cl 2  CH.sub.2                                                                           CHOC.sub.2 H.sub.5                                                                         H CH.sub.3                                     9.80                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Cl 2  (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                         H CH.sub.3                                     9.81                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Cl 0  (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                         H CH.sub.3                                     9.82                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Cl 2  CH.sub.2                                                                           CHOiPr      H CH.sub.3                                     9.83                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Cl 2  (CH.sub.2).sub.2                                                                   CHOiPr      H CH.sub.3                                     9.84                                                                              CH.sub.3                                                                          CH.sub.3                                                                           Cl 0  (CH.sub.2).sub.2                                                                   CHOiPr      H CH.sub.3                                     __________________________________________________________________________

                  TABLE 10                                                         ______________________________________                                         Compounds of the formula                                                        ##STR281##                                                                    No.  R.sup.17                                                                              R.sup.18                                                                              R.sup.19                                                                            n   R.sup.12                                                                            R.sup.13                                                                            Y      L   M                             ______________________________________                                         10.1 H      H      H    0   H    H    C═O                                                                               H   CH.sub.3                      10.2 CH.sub.3                                                                              H      H    0   H    H    C═O                                                                               H   CH.sub.3                      10.3 CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    H    C═O                                                                               H   CH.sub.3                      10.4 H      H      H    2   H    H    C═O                                                                               H   CH.sub.3                      10.5 CH.sub.3                                                                              H      H    2   H    H    C═O                                                                               H   CH.sub.3                      10.6 CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    H    C═O                                                                               H   CH.sub.3                      10.7 H      H      H    0   H    H    C═O                                                                               H   Cl                            10.8 CH.sub.3                                                                              H      H    0   H    H    C═O                                                                               H   Cl                            10.9 CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    H    C═O                                                                               H   Cl                            10.10                                                                               H      H      H    2   H    H    C═O                                                                               H   Cl                            10.11                                                                               CH.sub.3                                                                              H      H    2   H    H    C═O                                                                               H   Cl                            10.12                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    H    C═O                                                                               H   Cl                            10.13                                                                               H      H      H    0   H    H    CHOCH.sub.3                                                                           H   CH.sub.3                      10.14                                                                               CH.sub.3                                                                              H      H    0   H    H    CHOCH.sub.3                                                                           H   CH.sub.3                      10.15                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    H    CHOCH.sub.3                                                                           H   CH.sub.3                      10.16                                                                               H      H      H    2   H    H    CHOCH.sub.3                                                                           H   CH.sub.3                      10.17                                                                               CH.sub.3                                                                              H      H    2   H    H    CHOCH.sub.3                                                                           H   CH.sub.3                      10.18                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    H    CHOCH.sub.3                                                                           H   CH.sub.3                      10.19                                                                               H      H      H    0   H    H    CHOCH.sub.3                                                                           H   Cl                            10.20                                                                               CH.sub.3                                                                              H      H    0   H    H    CHOCH.sub.3                                                                           H   Cl                            10.21                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    H    CHOCH.sub.3                                                                           H   Cl                            10.22                                                                               H      H      H    2   H    H    CHOCH.sub.3                                                                           H   Cl                            10.23                                                                               CH.sub.3                                                                              H      H    2   H    H    CHOCH.sub.3                                                                           H   Cl                            10.24                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    H    CHOCH.sub.3                                                                           H   Cl                            10.25                                                                               H      H      H    0   H    CH.sub.3                                                                            C═O                                                                               H   CH.sub.3                      10.26                                                                               CH.sub.3                                                                              H      H    0   H    CH.sub.3                                                                            C═O                                                                               H   CH.sub.3                      10.27                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    CH.sub.3                                                                            C═O                                                                               H   CH.sub.3                      10.28                                                                               H      H      H    2   H    CH.sub.3                                                                            C═O                                                                               H   CH.sub.3                      10.29                                                                               CH.sub.3                                                                              H      H    2   H    CH.sub.3                                                                            C═O                                                                               H   CH.sub.3                      10.30                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    CH.sub.3                                                                            C═O                                                                               H   CH.sub.3                      10.31                                                                               H      H      H    0   H    CH.sub.3                                                                            C═O                                                                               H   Cl                            10.32                                                                               CH.sub.3                                                                              H      H    0   H    CH.sub.3                                                                            C═O                                                                               H   Cl                            10.33                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    CH.sub.3                                                                            C═O                                                                               H   Cl                            10.34                                                                               H      H      H    2   H    CH.sub.3                                                                            C═O                                                                               H   Cl                            10.35                                                                               CH.sub.3                                                                              H      H    2   H    CH.sub.3                                                                            C═O                                                                               H   Cl                            10.36                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    CH.sub.3                                                                            C═O                                                                               H   Cl                            10.37                                                                               H      H      H    0   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   CH.sub.3                      10.38                                                                               CH.sub.3                                                                              H      H    0   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   CH.sub.3                      10.39                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   CH.sub.3                      10.40                                                                               H      H      H    2   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   CH.sub.3                      10.41                                                                               CH.sub.3                                                                              H      H    2   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   CH.sub.3                      10.42                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   CH.sub.3                      10.43                                                                               H      H      H    0   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   Cl                            10.44                                                                               CH.sub.3                                                                              H      H    0   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   Cl                            10.45                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   Cl                            10.46                                                                               H      H      H    2   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   Cl                            10.47                                                                               CH.sub.3                                                                              H      H    2   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   Cl                            10.48                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    CH.sub.3                                                                            CHOCH.sub.3                                                                           H   Cl                            10.49                                                                               H      H      H    0   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   CH.sub.3                      10.50                                                                               CH.sub.3                                                                              H      H    0   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   CH.sub.3                      10.51                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   CH.sub.3                      10.52                                                                               H      H      H    2   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   CH.sub.3                      10.53                                                                               CH.sub.3                                                                              H      H    2   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   CH.sub.3                      10.54                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   CH.sub.3                      10.55                                                                               H      H      H    0   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   Cl                            10.56                                                                               CH.sub.3                                                                              H      H    0   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   Cl                            10.57                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   Cl                            10.58                                                                               H      H      H    2   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   Cl                            10.59                                                                               CH.sub.3                                                                              H      H    2   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   Cl                            10.60                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    C.sub.6 H.sub.5                                                                     C═O                                                                               H   Cl                            10.61                                                                               H      H      H    0   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   CH.sub.3                      10.62                                                                               CH.sub.3                                                                              H      H    0   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   CH.sub.3                      10.63                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   CH.sub.3                      10.64                                                                               H      H      H    2   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   CH.sub.3                      10.65                                                                               CH.sub.3                                                                              H      H    2   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   CH.sub.3                      10.66                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   CH.sub.3                      10.67                                                                               H      H      H    0   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   Cl                            10.68                                                                               CH.sub.3                                                                              H      H    0   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   Cl                            10.69                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   Cl                            10.70                                                                               H      H      H    2   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   Cl                            10.71                                                                               CH.sub.3                                                                              H      H    2   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   Cl                            10.72                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    C.sub.6 H.sub.5                                                                     CHOCH.sub.3                                                                           H   Cl                            10.73                                                                               H      H      H    0   H    H    CH.sub.2                                                                              H   CH.sub.3                      10.74                                                                               CH.sub.3                                                                              H      H    0   H    H    CH.sub.2                                                                              H   CH.sub.3                      10.75                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    H    CH.sub.2                                                                              H   CH.sub.3                      10.76                                                                               H      H      H    2   H    H    CH.sub.2                                                                              H   CH.sub.3                      10.77                                                                               CH.sub.3                                                                              H      H    2   H    H    CH.sub.2                                                                              H   CH.sub.3                      10.78                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    H    CH.sub.2                                                                              H   CH.sub.3                      10.79                                                                               H      H      H    0   H    H    CH.sub.2                                                                              H   Cl                            10.80                                                                               CH.sub.3                                                                              H      H    0   H    H    CH.sub.2                                                                              H   Cl                            10.81                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    0   H    H    CH.sub.2                                                                              H   Cl                            10.82                                                                               H      H      H    2   H    H    CH.sub.2                                                                              H   Cl                            10.83                                                                               CH.sub.3                                                                              H      H    2   H    H    CH.sub.2                                                                              H   Cl                            10.84                                                                               CH.sub.3                                                                              CH.sub.3                                                                              H    2   H    H    CH.sub.2                                                                              H   Cl                            ______________________________________                                    

                                      TABLE 11                                     __________________________________________________________________________     Compounds of the formula                                                        ##STR282##                                                                    No. R.sup.17   n X   Y          L M                                            __________________________________________________________________________     11.1                                                                               2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           C═O    H CH.sub.3                                     11.2                                                                               2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.3                                                                               2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.4                                                                               2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           CHOCH.sub.3                                                                               H CH.sub.3                                     11.5                                                                               2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.6                                                                               2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.7                                                                               2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.8                                                                               2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.9                                                                               2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.10                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           CHOiPr     H CH.sub.3                                     11.11                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.12                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.13                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           C═NOCH.sub.3                                                                          H CH.sub.3                                     11.14                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.15                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.16                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.17                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.18                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.19                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           C═NOiPr                                                                               H CH.sub.3                                     11.20                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.21                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.22                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                     11.23                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                     11.24                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                     11.25                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                     11.26                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                     11.27                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                     11.28                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           C(CH.sub.3).sub.2                                                                         H CH.sub.3                                     11.29                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   C(CH.sub.3).sub.2                                                                         H CH.sub.3                                     11.30                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   C(CH.sub.3).sub.2                                                                         H CH.sub.3                                     11.31                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           CH--NHCH.sub.3                                                                            H CH.sub.3                                     11.32                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   CH--NHCH.sub.3                                                                            H CH.sub.3                                     11.33                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   CH--NHCH.sub.3                                                                            H CH.sub.3                                     11.34                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                     11.35                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                     11.36                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   CH--NHC.sub.2 H.sub.5                                                                     H CH.sub.3                                     11.37                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                     11.38                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                     11.39                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3).sub.2                                                                     H CH.sub.3                                     11.40                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                     11.41                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                     11.42                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   CH--NHOC.sub.2 H.sub.5                                                                    H CH.sub.3                                     11.43                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                     11.44                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                     11.45                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3)OC.sub.2 H.sub.5                                                           H CH.sub.3                                     11.46                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           C═N--NH.sub.2                                                                         H CH.sub.3                                     11.47                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   C═N--NH.sub.2                                                                         H CH.sub.3                                     11.48                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   C═N--NH.sub.2                                                                         H CH.sub.3                                     11.49                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                     11.50                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                     11.51                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   C═N--N(CH.sub.3).sub.2                                                                H CH.sub.3                                     11.52                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                     11.53                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                     11.54                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   CH--N(CH.sub.3)OCH.sub.2 C.sub.6 H.sub.5                                                  H CH.sub.3                                     11.55                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                     11.56                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                     11.57                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   C(CH.sub.3)--OCH.sub.3                                                                    H CH.sub.3                                     11.58                                                                              2-Ethylthiopropyl                                                                         2 CH.sub.2                                                                           O          H CH.sub.3                                     11.59                                                                              2-Ethylthiopropyl                                                                         0 (CH.sub.2).sub.2                                                                   O          H CH.sub.3                                     11.60                                                                              2-Ethylthiopropyl                                                                         2 (CH.sub.2).sub.2                                                                   O          H CH.sub.3                                     11.61                                                                              Tetrahydropyran-3-yl                                                                      2 CH.sub.2                                                                           C═O    H CH.sub.3                                     11.62                                                                              Tetrahydropyran-3-yl                                                                      0 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.63                                                                              Tetrahydropyran-3-yl                                                                      2 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.64                                                                              Tetrahydropyran-3-yl                                                                      2 CH.sub.2                                                                           CHOCH.sub.3                                                                               H CH.sub.3                                     11.65                                                                              Tetrahydropyran-3-yl                                                                      0 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.66                                                                              Tetrahydropyran-3-yl                                                                      2 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.67                                                                              Tetrahydropyran-3-yl                                                                      2 CH.sub.2                                                                           CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.68                                                                              Tetrahydropyran-3-yl                                                                      0 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.69                                                                              Tetrahydropyran-3-yl                                                                      2 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.70                                                                              Tetrahydropyran-3-yl                                                                      2 CH.sub.2                                                                           CHOiPr     H CH.sub.3                                     11.71                                                                              Tetrahydropyran-3-yl                                                                      0 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.72                                                                              Tetrahydropyran-3-yl                                                                      2 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.73                                                                              Tetrahydropyran-3-yl                                                                      2 CH.sub.2                                                                           C═NOCH.sub.3                                                                          H CH.sub.3                                     11.74                                                                              Tetrahydropyran-3-yl                                                                      2 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.75                                                                              Tetrahydropyran-3-yl                                                                      0 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.76                                                                              Tetrahydropyran-3-yl                                                                      2 CH.sub.2                                                                           C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.77                                                                              Tetrahydropyran-3-yl                                                                      2 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.78                                                                              Tetrahydropyran-3-yl                                                                      0 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.79                                                                              Tetrahydropyran-3-yl                                                                      2 CH.sub.2                                                                           C═NOiPr                                                                               H CH.sub.3                                     11.80                                                                              Tetrahydropyran-3-yl                                                                      2 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.81                                                                              Tetrahydropyran-3-yl                                                                      0 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.82                                                                              Tetrahydropyran-4-yl                                                                      2 CH.sub.2                                                                           C═O    H CH.sub.3                                     11.83                                                                              Tetrahydropyran-4-yl                                                                      0 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.84                                                                              Tetrahydropyran-4-yl                                                                      2 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.85                                                                              Tetrahydropyran-4-yl                                                                      2 CH.sub.2                                                                           CHOCH.sub.3                                                                               H CH.sub.3                                     11.86                                                                              Tetrahydropyran-4-yl                                                                      0 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.87                                                                              Tetrahydropyran-4-yl                                                                      2 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.88                                                                              Tetrahydropyran-4-yl                                                                      2 CH.sub.2                                                                           CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.89                                                                              Tetrahydropyran-4-yl                                                                      0 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.90                                                                              Tetrahydropyran-4-yl                                                                      2 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.91                                                                              Tetrahydropyran-4-yl                                                                      2 CH.sub.2                                                                           CHOiPr     H CH.sub.3                                     11.92                                                                              Tetrahydropyran-4-yl                                                                      0 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.93                                                                              Tetrahydropyran-4-yl                                                                      2 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.94                                                                              Tetrahydropyran-4-yl                                                                      2 CH.sub.2                                                                           C═NOCH.sub.3                                                                          H CH.sub.3                                     11.95                                                                              Tetrahydropyran-4-yl                                                                      2 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.96                                                                              Tetrahydropyran-4-yl                                                                      0 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.97                                                                              Tetrahydropyran-4-yl                                                                      2 CH.sub.2                                                                           C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.98                                                                              Tetrahydropyran-4-yl                                                                      2 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.99                                                                              Tetrahydropyran-4-yl                                                                      0 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.100                                                                             Tetrahydropyran-4-yl                                                                      2 CH.sub.2                                                                           C═NOiPr                                                                               H CH.sub.3                                     11.101                                                                             Tetrahydropyran-4-yl                                                                      2 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.102                                                                             Tetrahydropyran-4-yl                                                                      0 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.103                                                                             Tetrahydrothiopyran-3-yl                                                                  2 CH.sub.2                                                                           C═O    H CH.sub.3                                     11.104                                                                             Tetrahydrothiopyran-3-yl                                                                  0 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.105                                                                             Tetrahydrothiopyran-3-yl                                                                  2 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.106                                                                             Tetrahydrothiopyran-3-yl                                                                  2 CH.sub.2                                                                           CHOCH.sub.3                                                                               H CH.sub.3                                     11.107                                                                             Tetrahydrothiopyran-3-yl                                                                  0 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.108                                                                             Tetrahydrothiopyran-3-yl                                                                  2 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.109                                                                             Tetrahydrothiopyran-3-yl                                                                  2 CH.sub.2                                                                           CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.110                                                                             Tetrahydrothiopyran-3-yl                                                                  0 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.111                                                                             Tetrahydrothiopyran-3-yl                                                                  2 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.112                                                                             Tetrahydrothiopyran-3-yl                                                                  2 CH.sub.2                                                                           CHOiPr     H CH.sub.3                                     11.113                                                                             Tetrahydrothiopyran-3-yl                                                                  0 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.114                                                                             Tetrahydrothiopyran-3-yl                                                                  2 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.115                                                                             Tetrahydrothiopyran-3-yl                                                                  2 CH.sub.2                                                                           C═NOCH.sub.3                                                                          H CH.sub.3                                     11.116                                                                             Tetrahydrothiopyran-3-yl                                                                  2 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.117                                                                             Tetrahydrothiopyran-3-yl                                                                  0 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.118                                                                             Tetrahydrothiopyran-3-yl                                                                  2 CH.sub.2                                                                           C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.119                                                                             Tetrahydrothiopyran-3-yl                                                                  2 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.120                                                                             Tetrahydrothiopyran-3-yl                                                                  0 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.121                                                                             Tetrahydrothiopyran-3-yl                                                                  2 CH.sub.2                                                                           C═NOiPr                                                                               H CH.sub.3                                     11.122                                                                             Tetrahydrothiopyran-3-yl                                                                  2 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.123                                                                             Tetrahydrothiopyran-3-yl                                                                  0 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.124                                                                             1-Methylthiocyclopropyl                                                                   2 CH.sub.2                                                                           C═O    H CH.sub.3                                     11.125                                                                             1-Methylthiocyclopropyl                                                                   0 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.126                                                                             1-Methylthiocyclopropyl                                                                   2 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.127                                                                             1-Methylthiocyclopropyl                                                                   2 CH.sub.2                                                                           CHOCH.sub.3                                                                               H CH.sub.3                                     11.128                                                                             1-Methylthiocyclopropyl                                                                   0 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.129                                                                             1-Methylthiocyclopropyl                                                                   2 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.130                                                                             1-Methylthiocyclopropyl                                                                   2 CH.sub.2                                                                           CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.131                                                                             1-Methylthiocyclopropyl                                                                   0 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.132                                                                             1-Methylthiocyclopropyl                                                                   2 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.133                                                                             1-Methylthiocyclopropyl                                                                   2 CH.sub.2                                                                           CHOiPr     H CH.sub.3                                     11.134                                                                             1-Methylthiocyclopropyl                                                                   0 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.135                                                                             1-Methylthiocyclopropyl                                                                   2 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.136                                                                             1-Methylthiocyclopropyl                                                                   2 CH.sub.2                                                                           C═NOCH.sub.3                                                                          H CH.sub.3                                     11.137                                                                             1-Methylthiocyclopropyl                                                                   2 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.138                                                                             1-Methylthiocyclopropyl                                                                   0 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.139                                                                             1-Methylthiocyclopropyl                                                                   2 CH.sub.2                                                                           C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.140                                                                             1-Methylthiocyclopropyl                                                                   2 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.141                                                                             1-Methylthiocyclopropyl                                                                   0 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.142                                                                             1-Methylthiocyclopropyl                                                                   2 CH.sub.2                                                                           C═NOiPr                                                                               H CH.sub.3                                     11.143                                                                             1-Methylthiocyclopropyl                                                                   2 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.144                                                                             1-Methylthiocyclopropyl                                                                   0 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.145                                                                             (Dimethoxy)methyl                                                                         2 CH.sub.2                                                                           C═O    H CH.sub.3                                     11.146                                                                             (Dimethoxy)methyl                                                                         0 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.147                                                                             (Dimethoxy)methyl                                                                         2 (CH.sub.2).sub.2                                                                   C═O    H CH.sub.3                                     11.148                                                                             (Dimethoxy)methyl                                                                         2 CH.sub.2                                                                           CHOCH.sub.3                                                                               H CH.sub.3                                     11.149                                                                             (Dimethoxy)methyl                                                                         0 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.150                                                                             (Dimethoxy)methyl                                                                         2 (CH.sub.2).sub.2                                                                   CHOCH.sub.3                                                                               H CH.sub.3                                     11.151                                                                             (Dimethoxy)methyl                                                                         2 CH.sub.2                                                                           CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.152                                                                             (Dimethoxy)methyl                                                                         0 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.153                                                                             (Dimethoxy)methyl                                                                         2 (CH.sub.2).sub.2                                                                   CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                     11.154                                                                             (Dimethoxy)methyl                                                                         2 CH.sub.2                                                                           CHOiPr     H CH.sub.3                                     11.155                                                                             (Dimethoxy)methyl                                                                         0 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.156                                                                             (Dimethoxy)methyl                                                                         2 (CH.sub.2).sub.2                                                                   CHOiPr     H CH.sub.3                                     11.157                                                                             (Dimethoxy)methyl                                                                         2 CH.sub.2                                                                           C═NOCH.sub.3                                                                          H CH.sub.3                                     11.158                                                                             (Dimethoxy)methyl                                                                         2 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.159                                                                             (Dimethoxy)methyl                                                                         0 (CH.sub.2).sub.2                                                                   C═NOCH.sub.3                                                                          H CH.sub.3                                     11.160                                                                             (Dimethoxy)methyl                                                                         2 CH.sub.2                                                                           C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.161                                                                             (Dimethoxy)methyl                                                                         2 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.162                                                                             (Dimethoxy)methyl                                                                         0 (CH.sub.2).sub.2                                                                   C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                     11.163                                                                             (Dimethoxy)methyl                                                                         2 CH.sub.2                                                                           C═NOiPr                                                                               H CH.sub.3                                     11.164                                                                             (Dimethoxy)methyl                                                                         2 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     11.165                                                                             (Dimethoxy)methyl                                                                         0 (CH.sub.2).sub.2                                                                   C═NOiPr                                                                               H CH.sub.3                                     __________________________________________________________________________

PREPARATION EXAMPLES

A) Preparation of the Starting Materials and Intermediates

1. 3-Thio-2-methylbenzoic Acid

100 g (0.66 mol) of 3-amino-2-methylbenzoic acid are initially introduced together with 270 g of ice and 127 ml of concentrated hydrochloric acid. 45.7 g (0.66 mol) of sodium nitrite in 270 ml of water are then added dropwise at 0-10° C.

In a second vessel, 84.2 g (0.79 mol) of sodium carbonate and 106 g (0.66 mol) of potassium methylxanthate are dissolved in 450 ml of water and heated to 60-70° C. The diazonium solution is cautiously added dropwise. The mixture is subsequently stirred for 1 hour. 106 g (2.65 mol) of sodium hydroxide in 270 ml of water are then added, the mixture is stirred for a further 2 hours, the solution is rendered acidic using hydrochloric acid and the resulting precipitate is filtered off with suction. The solid is washed with water and dried.

Yield: 110 g (100% of theory) of 3-thio-2-methylbenzoic acid; melting point 155° C. ¹ H-NMR (d⁶ -DMSO): δ [ppm]=13.0 (1H, bs), 7.7 (2H, m), 7.3 (1H, tr), 2.4 (3H, s).

2. Methyl 3-thio-2-methylbenzoate [sic]

110 g (0.66 mol) of 3-thio-2-methylbenzoic acid are dissolved in 1.6 l of methanol which contains 5% sulfuric acid and the mixture is refluxed for 5 hours. The alcohol is then distilled off, the residue is taken up in ethyl acetate, and the organic phase is washed with water and with sodium carbonate, dried using sodium sulfate and concentrated.

Yield: 104 g (87% of theory) of methyl 3-thio-2-methylbenzoate; ¹ H-NMR (CDCl₃):δ [ppm]=7.6 (1H, d), 7.4 (1H, d), 7.1 (1H, d), 3.9 (3H, s), 3.4 (1H, s), 2.5 (3H, s).

3. Methyl 3-thio(2'-propionic acid)-2-methylbenzoate ##STR283##

70 g (0.38 mol) of methyl 3-thio-2-methylbenzoate are dissolved in 400 ml of water and refluxed for 7 hours with 30.8 g (0.77 mol) of sodium hydroxide solution and 58.8 g (0.45 mol) of bromopropionic acid. After cooling, the aqueous phase is washed with methyl tert-butyl ether. The aqueous phase is then acidified with 2 N hydrochloric acid, the resulting precipitate is filtered off with suction and washed with water, and the product is dried.

Yield: 75.5 g (78% of theory) of methyl 3-thiopropionic acid-2-methylbenzoate; ¹ H-NMR (CDCl₃): δ [ppm]=7.66 (1H, d), 7.51 (1H, d), 7.20 (1H, tr), 3.96 (3H, s), 3.18 (2H, tr), 2.70 (2H, tr), 2.63 (3H, s).

4. Methyl 8-methylthiochroman-4-one-7-carboxylate ##STR284##

4 g (15.8 mmol) of methyl 3-thiopropionic acid-2-methylbenzoate are stirred at 70° C. for 15 minutes in 40 g of polyphosphoric acid. The reaction solution is then added to ice-water and the resulting precipitate is filtered off with suction. The product is washed with water and dried in a drying cabinet. As a by-product of the cyclization, methyl 8-methylthiochromen-4-one-carboxylate can be formed, which can be separated off by chromatography.

Yield: 3.1 g (83% of theory) of methyl 8-methylthiochroman-4-one-7-carboxylate; ¹ H-NMR (CDCl₃): δ [ppm]=8.00 (1H, d), 7.30 (1H, d), 3.94 (3H, s), 3.15 (2H, m), 2.98 (2H, m), 2.50 (3H, s);

Secondary component: methyl 8-methylthiochromen-4-one-carboxylate: ¹ H-NMR (CDCl₃): δ [ppm]=8.4 (1H, d), 7.9 (1H, d), 7.8 (1H, d), 7.0 (1H, d), 4.0 (3H, s), 2.7 (3H, s).

5. 8-Methylthiochroman-4-one-7-carboxylic acid

41.1 g (0.17 mol) of methyl 8-methylthiochroman-4-one-7-carboxylate are hydrolyzed under reflux with 10.3 g (0.26 mol) of NaOH in a mixture of 400 ml of water and methanol. The methanol is then distilled off and the residue is diluted with water and acidifed with 2N hydrochloric acid. The useful product precipitates out and is filtered off with suction, washed with water and dried.

Yield: 34.4 g (89% of theory) of 8-methylthiochroman-4-one-7-carboxylic acid; melting point: 243-246° C.

6. 8-Methyl-1,1-dioxothiochroman-4-one-7-carboxylic acid ##STR285##

20 g (0.09 mol) of 8-methylthiochroman-4-one-7-carboxylic acid are dissolved in 100 ml of acetic acid. A spatula tipful of sodium tungstate is added. 24.9 g (0.22 mol) of 30% strength hydrogen peroxide solution are then added dropwise at 50° C. The mixture is subsequently stirred at about 20° C. for 1 hour. The reaction solution is then added to water, a precipitate being formed which is filtered off with suction. After washing the product with water, it is dried.

Yield: 18.4 g (80% of theory) of 8-methyl-1,1-dioxothiochroman-4-one-7-carboxylic acid; melting point: 224-225° C.

7. Methyl 4-hydroxy-8-methylthiochroman-7-carboxylate ##STR286##

30 g (0.127 mol) of methyl 8-methylthiochroman-4-one-7-carboxylate are dissolved in a mixture of 120 ml of methylene chloride and 60 ml of methanol and cooled to 0-5° C. 2.4 g (0.064 mol) of sodium borohydride are then added in portions. The mixture is subsequently stirred at this temperature for 1 hour, and 200 ml of 2N hydrochloric acid are added to the reaction solution. Two phases are formed. The organic phase is separated off and dried, and the solvent is removed by distillation. The crude product is directly reacted further without further purification.

Yield: 27.6 g (91% of theory) of methyl 4-hydroxy-8-methylthiochroman-7-carboxylate.

8. Methyl 4-ethoxy-8-methylthiochroman-7-carboxylate

13.8 g (0.058 mol) of methyl 4-hydroxy-8-methylthiochroman-7-carboxylate are heated at boiling point for 4 hours in 60 ml of ethanol with addition of 1 g of sulfuric acid. The solvent is then distilled off and the residue is taken up with water. The aqueous phase is extracted with ethyl acetate. The organic phase is washed with sodium hydrogen carbonate solution, dried and concentrated. The product is purified by chromatography.

Yield: 10.1 g (60% of theory) of methyl 4-ethoxy-8-methylthiochroman-7-carboxylate; ¹ H-NMR (CDCl₃): δ [ppm]=7.44 (1H, d), 7.13 (1H, d), 4.40 (1H, m), 3.90 (3H, s), 3.60 (2H, m), 3.38 (1 H, dtr), 2.90 (1H, m), 2.50 (3H, g), 2.40 (1H, m), 1.98 (1H, m), 1.10 (3H, tr).

The reaction to give methyl 4-methoxy-8-methylthiochroman-4-one-7-carboxylate and methyl 4-isopropoxy-8-methylthiochroman-4-one-7-carboxylate is carried out analogously to the above procedure, in the case of methyl 4-methoxy-8-methylthiochroman-4-one-7-carboxylate ethanol being replaced by methanol and in the case of methyl 4-isopropoxy-8-methylthiochroman-4-one-7-carboxylate ethanol being replaced by isopropanol.

9. 4-Ethoxy-8-methylthiochroman-7-carboxylic acid

2.1 g of sodium hydroxide solution are dissolved in 20 ml of water. Methyl 4-ethoxy-8-methylthiochroman-4-one-7-carboxylate dissolved in 20 ml of methanol is added dropwise at about 20° C. The mixture is refluxed for 2 hours. The solvent is then distilled off and the residue is added to 2N hydrochloric acid. The aqueous phase is extracted with methylene chloride and the organic phase is dried and concentrated.

Yield: 9.3 g (100% of theory) of 4-ethoxy-8-methylthiochroman-7-carboxylic acid; melting point: 89-98° C.

Hydrolysis of the corresponding esters to 4-ethoxy-8-methylthiochroman-7-carboxylic acid and 4-isopropoxy-8-methylthiochroman-7-carboxylic acid proceeds in a similar manner. The same applies to the hydrolysis of the corresponding benzo[b]thiophene derivatives shown below.

10. 8-Methyl-4-ethoxy-1,1-dioxothiochroman-7-carboxylic acid

8.4 g (0.033 mol) of 4-ethoxy-8-methylthiochroman-7-carboxylic acid are initially introduced in 60 ml of acetic acid. A spatula tipful of sodium tungstate is added. 7.9 g (0.07 mol) is of 30% strength hydrogen peroxide solution are slowly added dropwise at 50° C. and the reaction mixture is subsequently stirred for 2 hours. It is then poured into water and the aqueous phase is extracted with ethyl acetate. The organic phase is washed with bisulfite solution, then dried and concentrated.

Yield: 9.5 g (100% of theory) of 8-methyl-4-ethoxy-1,1-dioxothiochroman-7-carboxylic acid; melting point: 150° C.

11. 8-Methylthiochroman-4-one-7-carboxylic acid O-ethyl oxime ##STR287##

0.88 g (9 mmol) of ethylhydroxylamine is initially introduced in 20 ml of methanol. 0.62 g (4.5 mmol) of potassium carbonate is then added, followed by 2.0 g (9 mmol) of 8-methylthiochroman-4-one-7-carboxylic acid. The reaction is stirred at about 20° C. for 10 days. It is worked up by addition of water and 2N hydrochloric acid, and the resulting precipitate is filtered of f with suction and dried.

Yield: 2.2 g (92% of theory) of 8-methylthiochroman-4-one-7-carboxylic acid O-ethyl oxime; melting point: 166° C.

12. 8-Methyl-1,1-dioxothiochroman-4-one-7-carboxylic acid O-ethyl oxime

3.0 g (0.011 mol) of 8-methylthiochroman-4-one-7-carboxylic acid O-ethyl oxime are initially introduced into 30 ml of acetic acid together with a spatula tipful of sodium tungstate. 2.8 g (0.024 mol) of 30% strength hydrogen peroxide solution are added dropwise at 50° C. After stirring for 1 hour, the reaction mixture is poured into ice-water and the resulting precipitate is filtered off with suction. The product is washed with water and dried.

Yield: 2.5 g (74% of theory) of 8-methyl-1,1-dioxothiochroman-4-one-7-carboxylic acid O-ethyl oxime; melting point 198° C.

13. 8-Methyl-1-oxothiochroman-4-one-7-carboxylic Acid

7.0 g (31.5 mmol) of 8-methylthiochroman-4-one-7-carboxylic acid are initially introduced into 70 ml of acetic acid together with a spatula tipful of sodium tungstate. 3.6 g (31.5 mmol) of 30% strength hydrogen peroxide solution are added dropwise at 50° C. and the reaction solution is subsequently stirred for 3 hours. It is then stirred into water and the product is extracted with ethyl acetate. The organic phase is dried and the solvent is removed. The product is purified by chromatography.

Yield: 5.4 g (72% of theory) of 8-methyl-1-oxothiochroman-4-one-7-carboxylic acid; ¹ H-NMR (d⁶ -DMSO): δ [ppm]=8.0 (2H, m), 3.5 (3H, m), 2.8 (1H, m), 2.7 (3H, s).

14. Methyl 3-carboxymethylthio-2-methylbenzoate ##STR288##

12.4 g (0.068 mmol) of methyl 3-mercapto-2-methylbenzoate in 80 ml of dimethylformamide are added dropwise to 1.6 g (0.068 mol) of sodium hydride in 40 ml of dimethylformamide and the mixture is stirred at about 20° C. for 60 min. 8 g (0.068 mol) of chloroacetic acid are then added and the mixture is stirred at about 20° C. for 4 hours.

The reaction mixture is worked up by stirring it into ice-water containing hydrochloric acid.

The resulting precipitate is filtered off with suction, washed with water and dried.

Yield: 14.6 g (89% of theory) of methyl 3-carboxymethylthio-2-methylbenzoate; ¹ H-NMR (d⁶ -DMSO): δ [ppm]=7.55 (1H, d), 7.45 (1H, d), 7.21 (1H, tr), 3.82 (2H, s), 2.50 (3H, s).

15. Methyl 7-methylbenzo[b]thiophene-3[2H]-one-6-carboxylate ##STR289##

14.3 g (0.06 mmol) of 3-carboxymethylthio-2-methylbenzoic acid are dissolved in 300 ml of methylene chloride and 13.1 g (0.11 mmol) of thionyl chloride are added dropwise. The mixture is refluxed for 1 hour and the solvent and excess thionyl chloride are then distilled off. The residue is taken up in 100 ml of methylene chloride and treated with 31.8 g (0.24 mmol) of aluminum trichloride. The reaction is stirred at about 20° C. for 1 hour. The mixture is then added to ice-water and the organic phase is separated off. After washing and drying the organic phase, the solvent is removed. The product is reacted further without purification.

Yield: 12.9 g (97% of theory) of methyl 7-methylbenzo[b]thiophene-3[2H]-one-6-carboxylate; ¹ H-NMR (CDCl₃): δ [ppm]=7.65 (2H, m), 3.93 (3H, s), 3.88 (2H, s), 2.50 (3H, s).

16. Methyl 7-methyl-3-hydroxybenzo[b]thiophene-[2H]-6-carboxylate ##STR290##

12.8 g (0.058 mol) of methyl 7-methylbenzo[b]thiophene-3[2H]-one-6-carboxylate are dissolved in 120 ml of methylene chloride and 60 ml of methanol and cooled to 0° C. 1.1 g (0.029 mol) of sodium borohydride is added in portions and the mixture is stirred for 3 hours. The reaction is terminated by adding water. The phases are separated and the aqueous phase is extracted with methylene chloride. The combined organic phases are dried and the solvent is distilled off. The crude product is reacted further.

Yield: 13.2 g (100% of theory) of methyl 7-methyl-3-hydroxybenzo[b]-thiophene-[2H]-6-carboxylate; ¹ H-NMR (CDCl₃): δ [ppm]=7.6 (2H, m), 5.3 (1H, m), 3.9 (3H, s), 3.7 (1H, m), 3.3 (1H, m), 2.4 (3H, s).

17. Methyl 7-methyl-3-methoxybenzo[b]thiophene-[2H]-6-carboxylate

2.4 g (0.059 mol) of NaH is dissolved in 50 ml of dimethylformamide. 13.2 g of methyl 7-methyl-3-hydroxybenzo[b]thiophene-[2H]-6-carboxylate dissolved in 50 ml are added dropwise and the mixture is subsequently stirred at about 20° C. for 2 hours. 8.4 g (0.059 mol) of iodomethane are then added and the mixture is stirred for a further 2 hours. The reaction solution is added to ice-water and extracted with ethyl acetate. The organic phase is dried and subsequently concentrated, and the product is purified by chromatography.

Yield: 3.5 g (25% of theory) of methyl 7-methyl-3-methoxybenzo[b]thiophene-[2H]-6-carboxylate; ¹ H-NMR (CDCl₃): δ [ppm]=7.60 (1H, d), 7.20 (1H, d), 5.04 (1H, m), 3.90 (3H, s),3.56 (1H, m), 3.40 (3H, s), 3.38 (1H, m), 2.50 (3H, s).

Similarly to the hydrolysis of the thiochromanone esters described above, the corresponding benzothiophene acids are also obtained.

The compounds shown in the following tables are obtained in a similar manner:

                                      TABLE 12                                     __________________________________________________________________________     Intermediates                                                                   ##STR291##                                                                    No.                                                                               T   n X    Y          L M  Physical data                                    __________________________________________________________________________     12.1                                                                              HO  0 (CH.sub.2).sub.2                                                                    C═O    H H  m.p. [° C.]: 226-231                      12.2                                                                              HO  2 (CH.sub.2).sub.2                                                                    C═O    H H  m.p. [° C.]: 217-220                      12.3                                                                              HO  0 (CH.sub.2).sub.2                                                                    C═O    H CH.sub.3                                                                          m.p. [° C.]: 243-246                      12.4                                                                              HO  2 (CH.sub.2).sub.2                                                                    C═O    H CH.sub.3                                                                          m.p. [° C.]: 224-225                      12.5                                                                              HO  0 (CH.sub.2).sub.2                                                                    CHOCH.sub.3                                                                               H CH.sub.3                                                                          m.p. [° C.]: 117-118                      12.6                                                                              HO  2 (CH.sub.2).sub.2                                                                    CHOCH.sub.3                                                                               H CH.sub.3                                                                          m.p. [° C.]: 167-172                      12.7                                                                              HO  0 (CH.sub.2).sub.2                                                                    CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                                                          m.p. [° C.]: 89-98                        12.8                                                                              HO  2 (CH.sub.2).sub.2                                                                    CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                                                          m.p. [° C.]: 150                          12.9                                                                              HO  0 (CH.sub.2).sub.2                                                                    CHOiPropyl H CH.sub.3                                                                          m.p. [° C.]: 138                          12.10                                                                             HO  2 (CH.sub.2).sub.2                                                                    CHOiPropyl H CH.sub.3                                                                          m.p. [° C.]: 142                          12.11                                                                             HO  0 (CH.sub.2).sub.2                                                                    C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                                                          m.p. [° C.]: 166                          12.12                                                                             HO  2 (CH.sub.2).sub.2                                                                    C═NOC.sub.2 H.sub.5                                                                   H CH.sub.3                                                                          m.p. [° C.]: 198                          12.13                                                                             HO  0 (CH.sub.2).sub.2                                                                    C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                                                          m.p. [° C.]: 163                          12.14                                                                             HO  2 (CH.sub.2).sub.2                                                                    C═NOCH.sub.2 CH═CHCl                                                              H CH.sub.3                                                                          m.p. [° C.]: 174                          12.15                                                                             HO  0 (CH.sub.2).sub.2                                                                    C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H CH.sub.3                                                                          m.p. [° C.]: 178                          12.16                                                                             HO  2 (CH.sub.2).sub.2                                                                    C═NO-tButyl                                                                           H CH.sub.3                                                                          m.p. [° C.]: 217                          12.17                                                                             H.sub.3 CO                                                                         0 (CH.sub.2).sub.2                                                                    C(CH.sub.3).sub.2                                                                         H CH.sub.3                                                                          m.p. [° C.]: 63-65                        12.18                                                                             HO  2 (CH.sub.2).sub.2                                                                    CHOCH.sub.3                                                                               H Cl m.p. [° C.]: 137-139                      12.19                                                                             HO  2 (CH.sub.2).sub.2                                                                    C═NOC.sub.2 H.sub.5                                                                   H Cl m.p. [° C.]: 205                          12.20                                                                             HO  0 (CH.sub.2)                                                                          CHOCH.sub.3                                                                               H CH.sub.3                                                                          .sup.1 H-NMR, 300 MHz                                                          (d.sup.6 -DMSO): δ [ppm] =                                               13.0 (1H, s), 7.55 (1H, d), 7.25                                               (1H, d), 5.10 (1H, s), 3.62 (1H,                                               m), 3.42 (1H, m), 3.41 (3H, s),                                                2.42 (3H, s)                                     12.21                                                                             HO  2 (CH.sub.2)                                                                          CHOCH.sub.3                                                                               H CH.sub.3                                                                          .sup.1 H-NMR, 300 MHz                                                          (d.sup.6 -DMSO): δ [ppm] =                                               13.5 (1H, bs), 8.10 (1H, d), 7.60                                              (1H, d), 5.18 (1H, m), 4.07 (1H,                                               m), 3.75 (1H, m), 3.40 (3H, s),                                                2.70 (3H, s)                                     12.22                                                                             HO  2 (CH.sub.2).sub.2                                                                    C═O    H Cl .sup.1 H-NMR, 300 MHz                                                          (d.sup.6 -DMSO): δ [ppm] =                                               14.2 (1H, bs), 8.10 (1H, d), 7.98                                              (1H, d), 4.13 (2H, m), 3.30 (2H,                                               m)                                               12.23                                                                             HO  0 (CH.sub.2).sub.2                                                                    C═O    H Cl .sup.1 H-NMR, 300 MHz                                                          (d.sup.6 -DMSO): δ [ppm] =                                               13.9 (1H, bs), 8.10 (1H, d), 7.52                                              (1H, d), 3.41 (2H, m), 2.90 (2H,                                               m)                                               12.24                                                                             H.sub.3 CO                                                                         0 (CH.sub.2).sub.2                                                                    CHOCH.sub.3                                                                               H CH.sub.3                                                                          .sup.1 H-NMR, 400 MHz (CDCl.sub.3):                                            δ [ppm] = 7.46, 7.13, 4.28, 3.87,                                        3.38, 3.30, 2.90, 2.48, 2.39, 1.91               12.25                                                                             H.sub.3 CO                                                                         0 (CH.sub.2).sub.2                                                                    CHOC.sub.2 H.sub.5                                                                        H CH.sub.3                                                                          m.p. [° C.]: 94-98                        12.26                                                                             H.sub.3 CO                                                                         0 (CH.sub.2).sub.2                                                                    CHOiPropyl H CH.sub.3                                                                          .sup.1 H-NMR, 250 MHz (CDCl.sub.3):                                            δ [ppm] = 7.47, 7.17, 4.48, 3.88,                                        3.79, 3.29, 2.90, 2.48, 2.29, 1.97,                                            1.21                                             12.27                                                                             HO  1 (CH.sub.2).sub.2                                                                    C═O    H CH.sub.3                                                                          m.p. [° C.]: 98 (decomp.)                 12.28                                                                             H.sub.3 CO                                                                         0 CH═CH                                                                           C═O    H CH.sub.3                                                                          m.p. [° C.]: 128-130                      12.29                                                                             HO  0 CH═CH                                                                           C═O    H CH.sub.3                                                                          .sup.1 H-NMR, 250 MHz                                                          (d.sup.6 -DMSO): δ [ppm] =                                               13.52, 8.48, 8.30, 7.87, 7.03, 2.66              12.30                                                                             HO  0 (CH.sub.2).sub.2                                                                    C═NO-tButyl                                                                           H CH.sub.3                                                                          m.p. [° C.]: 217                          12.31                                                                             HO  2 (CH.sub.2).sub.2                                                                    C═NOC.sub.2 H.sub.5                                                                   H Cl m.p. [° C.]: 205                          12.32                                                                             HO  0 (CH.sub.2).sub.2                                                                    C(CH.sub.3).sub.2                                                                         H CH.sub.3                                                                          m.p. [° C.]: 212                          12.33                                                                             HO  0 (CH.sub.2).sub.2                                                                    CH.sub.2   H CH.sub.3                                                                          m.p. [° C.]: 155                          12.34                                                                             HO  0 (CH.sub.2).sub.2                                                                    CH(C.sub.6 H.sub.5)                                                                       H CH.sub.3                                                                          m.p. [° C.]: 175                          12.35                                                                             HO  2 (CH.sub.2).sub.2                                                                    CH.sub.2   H CH.sub.3                                                                          m.p. [° C.]: 204                          12.36                                                                             H.sub.3 CO                                                                         0 (CH.sub.2).sub.2                                                                    CH(C.sub.6 H.sub.5)                                                                       H CH.sub.3                                                                          m.p. [° C.]: 103                          12.37                                                                             HO  2 (CH.sub.2).sub.2                                                                    CH(C.sub.6 H.sub.5)                                                                       H CH.sub.3                                                                          m.p. [° C.]: 145                          12.38                                                                             HO  0 (CH.sub.2).sub.2                                                                    CHSC.sub.6 H.sub.5                                                                        H CH.sub.3                                                                          m.p. [° C.]: 77                           12.39                                                                             HO  2 (CH.sub.2).sub.2                                                                    CHSO2C.sub.6 H.sub.5                                                                      H CH.sub.3                                                                          m.p. [° C.]: 239                          12.40                                                                             HO  0 (CH.sub.2).sub.2                                                                    C═O    Cl                                                                               Cl .sup.1 H-NMR, 250 MHz (CDCl.sub.3):                                            δ [ppm] = 7.69, 3.31, 3.01                 12.41                                                                             HO  2 (CH.sub.2).sub.2                                                                    C═O    Cl                                                                               Cl .sup.1 H-NMR, 250 MHz                                                          (d.sup.6 -DMSO): δ [ppm]=                                                8.04, 4.16, 3.31                                 12.42                                                                             H.sub.3 CO                                                                         0 (CH.sub.2).sub.2                                                                    CHOH       Cl                                                                               Cl .sup.1 H-NMR, 250 MHz (CDCl.sub.3):                                            δ [ppm] = 7.50, 5.20, 4.92, 3.36,                                        2.89, 2.53, 1.85                                 12.43                                                                             HO  2 (CH.sub.2).sub.2                                                                    CHOI       Cl                                                                               Cl .sup.1 H-NMR, 250 MHz                                                          (d.sup.6 -DMSO): δ [ppm] = 8.03,                                         6.96, 5.08, 3.87, 3.62, 2.54, 2.37               12.44                                                                             HO  0 (CH.sub.2).sub.2                                                                    CHOH       H CH.sub.3                                                                          m.p. [° C.]: 209                          __________________________________________________________________________

                                      TABLE 12a                                    __________________________________________________________________________     Intermediates                                                                   ##STR292##                                                                    No.                                                                               T   n R.sup.12                                                                          R.sup.13                                                                          R.sup.21                                                                          R.sup.22                                                                          Y    L M  Physical data                                   __________________________________________________________________________     12.45                                                                             H.sub.3 CO                                                                         0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  C═O                                                                             H CH.sub.3                                                                          .sup.1 H-NMR, 270 MHz (CDCl.sub.3):                                            δ [ppm] = 8.02, 7.50, 3.92, 3.09,                                        2.50, 1.33                                      12.46                                                                             H.sub.3 CO                                                                         0 H  CH.sub.3                                                                          H  H  C═O                                                                             H CH.sub.3                                                                          m.p. [° C.]: 79                          12.47                                                                             H.sub.3 CO                                                                         0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                         H CH.sub.3                                                                          .sup.1 H-NMR, 270 MHz (CDCl.sub.3):                                            δ [ppm] = 7.44, 7.02, 3.89, 3.59,                                        3.33, 3.28, 2.50, 2.48, 1.21, 0.88              12.48                                                                             H.sub.3 CO                                                                         0 H  H  CH.sub.3                                                                          H  C═O                                                                             H CH.sub.3                                                                          m.p. [° C.]: 83                          12.49                                                                             H.sub.3 CO                                                                         0 H  H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                         H CH.sub.3                                                                          .sup.1 H-NMR, 270 MHz (CDCl.sub.3):                                            δ [ppm] = 7.46, 7.11, 4.31, 3.89,                                        3.65, 3.37, 2.48, 2.44, 1.64, 1.44              12.50                                                                             HO  0 H  CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                         H CH.sub.3                                                                          m.p. [° C.]: 124                         12.51                                                                             HO  0 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                         H CH.sub.3                                                                          m.p. [° C.]: 168                         12.52                                                                             HO  0 H  H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                         H CH.sub.3                                                                          m.p. [° C.]: 145                         12.53                                                                             HO  2 H  CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                         H CH.sub.3                                                                          m.p. [° C.]: 184                                              (trans)                                                   12.54                                                                             HO  2 CH.sub.3                                                                          CH.sub.3                                                                          H  H  CHOCH.sub.3                                                                         H CH.sub.3                                                                          m.p. [° C.]: 161                         12.55                                                                             HO  2 H  H  CH.sub.3                                                                          H  CHOCH.sub.3                                                                         H CH.sub.3                                                                          m.p. [° C.]: 182                         __________________________________________________________________________

Preparation of the Final Products

1. 2-(8-Methyl-1,1-dioxothiochroman-4-one-7-carbonyl)-1,3-cyclohexanedione ##STR293## a) 17.4 g (0.0685 mol) of 8-methyl-1,1-dioxothiochroman-4-one-7-carboxylic acid are dissolved in 170 ml of toluene and treated with one drop of dimethylformamide, and 8.96 g (0.0753 mol) of thionyl chloride are added. After refluxing for 4 hours, the reaction mixture is concentrated. The reaction product is directly reacted further.

Yield: 18.6 g (99% of theory) of 8-methyl-1,1-dioxothiochroman-4-one-7-carbonyl chloride;

b) 0.62 g (5.5 mmol) of cyclohexane-1,3-dione is initially introduced into 10 ml of acetonitrile together with 0.56 g (5.5 mol) of triethylamine. 1.5 (5.5 mmol) of 8-methyl-1,1-dioxothiochroman-4-one-7-carbonyl chloride dissolved in 20 ml of acetonitrile are then added dropwise.

The mixture is subsequently stirred at about 20° C. for one hour. 0.31 g (3.7 mmol) of acetone cyanohydrin and 2.8 g (22.5 mmol) of triethylamine are then added and the mixture is stirred for 1 hour. For working-up, the reaction solution is stirred into 2N hydrochloric acid and the aqueous phase is extracted with ethyl acetate. The organic phase is then extracted with Na₂ CO₃ solution and the alkaline aqueous phase is rendered acidic with cooling. The resulting precipitate is filtered off with suction, washed with water and dried.

Yield: 1.0 g (52% of theory) of 2-(8-methyl-1,1-dioxothiochroman-4-one-7-carbonyl)-1,3-cyclohexanedione melting point: 173-178° C.

2. 2-(8-Methyl-1,1-dioxothiochroman-4-one-7-carbonyl O-ethyl oxime)cyclohexane-1,3-dione ##STR294##

1.0 g (3.4 mmol) of 8-methyl-1,1-dioxochroman-4-one-7-carboxylic acid O-ethyl oxime is initially introduced into 10 ml of acetonitrile together with 0.39 g (3.5 mmol) of cyclohexane-1,3-dione, 0.75 g (3.6 mmol) of dicyclocarbodiimide (DCC) is added and the mixture is stirred for 2 hours. 0.1 ml of acetone cyanohydrin and 0.51 g (5.1 mmol) of triethylamine are then added and the reaction mixture is stirred for a further 2 hours. It is then stirred into sodium carbonate solution and extracted with ethyl acetate, and the organic phase is discarded. The aqueous phase is rendered acidic using hydrochloric acid and extracted again with ethyl acetate, the organic phase is dried and the solvent is distilled off. The product is purified by chromatography.

Yield: 600 mg (45% of theory) of 2-(8-methyl-1,1-dioxothiochroman-4-one-7-carbonyl O-ethyl oxime)cylohexane-1,3-dione; melting point: 143° C.

3. 2-(8-Methyl-4-ethoxy-1,1-dioxothiochroman-7-carbonyl)cyclohexane-1,3-dione ##STR295## a) 8.8 g (0.031 mmol) of 8-methyl-4-ethoxy-1,1-dioxothiochroman-7-carboxylic acid are dissolved in 50 ml of toluene, the solution is treated with 2 drops of dimethylformamide and 4.4 g (0.04 mmol) of thionyl chloride are added. After refluxing for 4 hours, the reaction mixture is concentrated. The acid chloride is directly employed further.

b) 0.56 g of cyclohexane-1,3-dione is initially introduced into 10 ml of methylene chloride together with 0.47 g (6 mmol) of pyridine. 1.5 g (5 mmol) of the acid chloride from 3a) in 20 ml of methylene chloride are then added dropwise and the mixture is stirred for one hour. The reaction solution is added to water and rendered acidic with hydrochloric acid. The aqueous phase is extracted with ethyl acetate, the organic phase is dried and the solvent is removed.

Yield: 1.88 g (99% of theory) of O-acylated product.

c) 1.3 g (3.4 mmol) of the product from 3b are dissolved in 20 ml of acetonitrile. The reaction mixture is then treated with 0.19 g (2.3 mmol) of acetone cyanohydrin and 1.7 g (17.2 mmol) of triethylamine and stirred for 2 hours. It is then added to 2N hydrochloric acid and extracted with ethyl acetate. The organic phase is then washed with sodium carbonate solution and discarded. Finally, the alkaline aqueous phase is rendered acidic using hydrochloric acid. The resulting precipitate is filtered off with suction and dried.

Yield: 0.6 g (46% of theory) of 2-(8-methyl-4-ethoxy-1,1-dioxothiochroman-7-carbonyl)cyclohexane-1,3-dione; ¹ H-NMR (CDCl₃): δ ppm]=17.5 (1H, s), 7.30 (1H, d), 7.18 (1H, d), 4.47 (1H, m), 3.95-3.83 (1H, m), 3.70-3.50 (2H, m), 3.28 (1H, m), 2.81 (2H, tr), 2.71-2.50 (2H, m), 2.64 (3H,s), 2.43 (2H, tr), 2.05 (2H, m), 1.24 (3H, tr).

The compounds shown in the following tables are obtained in a similar manner:

                                      TABLE 13                                     __________________________________________________________________________     Compounds of the formula                                                        ##STR296##                                                                    No.                                                                               R.sup.17                                                                          R.sup.18                                                                          R.sup.19                                                                          n R.sup.12                                                                          R.sup.13                                                                           R.sup.21                                                                          R.sup.22                                                                           Y          L  M  Physical data                     __________________________________________________________________________     13.1                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   C═O    H  H  m.p. [° C.]: 110           13.2                                                                              CH.sub.3                                                                          H  H  2 H  H   H  H   C═O    H  CH.sub.3                                                                          m.p. [° C.]: 84-86         13.3                                                                              H  H  H  2 H  H   H  H   C═O    H  CH.sub.3                                                                          m.p. [° C.]: 173-178       13.4                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   C═O    H  CH.sub.3                                                                          m.p. [° C.]: 84-85         13.5                                                                              H  H  H  0 H  H   H  H   C═O    H  CH.sub.3                                                                          m.p. [° C.]: 148-150       13.6                                                                              CH.sub.3                                                                          H  H  0 H  H   H  H   C═O    H  CH.sub.3                                                                          m.p. [° C.]: 128-130       13.7                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H   H  H   C═O    H  CH.sub.3                                                                          NMR (CDCl.sub.3), 300 MHz:                                                     δ [ppm] =                                                                17.5 (1H, s), 8.06 (1H, d),                                                    6.89 (1H, d),                                                                  3.25 (2H, m), 2.97 (2H, m),                                                    2.68                                                                           (2H, s), 2.31 (2H, s), 2.19                                                    (3H, s),                                                                       1.12 (6H, s)                      13.8                                                                              H  H  H  2 H  H   H  H   C═O    H  H  m.p. [° C.]: 159-162       13.9                                                                              CH.sub.3                                                                          H  H  2 H  H   H  H   C═O    H  H  m.p. [° C.]: 161-163       13.10                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   CHOCH.sub.3                                                                               H  CH.sub.3                                                                          NMR (CDCl.sub.3), 300 MHz:                                                     δ [ppm] =                                                                17.5 (1H, s), 7.30 (1H, d),                                                    7.19 (1H, d),                                                                  4.36 (1H, m), 3.41 (3H, s),                                                    3.28                                                                           (1H, m), 2.70-2.59 (4H, m),                                                    2.61                                                                           (3H, s), 2.30 (2H, m), 1.14                                                    (6H, s)                           13.11                                                                             H  H  H  2 H  H   H  H   CHOCH.sub.3                                                                               H  CH.sub.3                                                                          m.p. [° C.]: 80-84         13.12                                                                             CH.sub.3                                                                          H  H  2 H  H   H  H   CHOCH.sub.3                                                                               H  CH.sub.3                                                                          m.p. [° C.]: 73            13.13                                                                             H  H  H  2 H  H   H  H   CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                                                                          NMR (CDCl.sub.3), 300 MHz:                                                     δ [ppm] =                                                                17.5 (1H, s), 7.30 (1H, d),                                                    7.18 (1H, d),                                                                  4.47 (1H, m), 3.95-3.83 (1H,                                                   m),                                                                            3.70-3.50 (2H, m), 3.28 (1H,                                                   m),                                                                            2.81 (2H, tr), 2.71-2.50                                                       (2H, m), 2.64                                                                  (3H, s), 2.43 (2H, tr), 2.05                                                   (2H, m),                                                                       1.24 (3H, tr)                     13.14                                                                             CH.sub.3                                                                          H  H  2 H  H   H  H   CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                                                                          m.p. [° C.]: 68-72         13.15                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   CHOC.sub.2 H.sub.5                                                                        H  CH.sub.3                                                                          NMR (CDCl.sub.3), 300 MHz:                                                     δ [ppm] =                                                                17.5 (1H, s), 7.31 (1H, d),                                                    7.18 (1H, d),                                                                  4.47 (1H, m), 3.96-3.82 (1H,                                                   m),                                                                            3.69-3.50 (2H, m), 3.28 (1H,                                                   m), 2.81                                                                       (2H, tr), 2.72-2.49 (2H, m),                                                   2.68                                                                           (2H, s), 2.60 (3H, s), 2.31                                                    (2H, s), 1.24                                                                  (3H, tr), 1.11 (6H, s)            13.16                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   CHOiPropyl H  CH.sub.3                                                                          m.p. [° C.]: 80-83         13.17                                                                             H  H  H  2 H  H   H  H   CHOiPropyl H  CH.sub.3                                                                          m.p. [° C.]: 144-146       13.18                                                                             CH.sub.3                                                                          H  H  2 H  H   H  H   CHOiPropyl H  CH.sub.3                                                                          m.p. [° C.]: 85            13.19                                                                             H  H  H  1 H  H   H  H   C═O    H  CH.sub.3                                                                          NMR (CDCl.sub.3), 300 MHz:                                                     δ [ppm] =                                                                17.25 (1H, s), 8.14 (1H, d),                                                   7.33                                                                           (1H, d), 3.90-3.57 (1H, m),                                                    3.39-3.26                                                                      (1H, m), 2.99-2.79 (3H, m),                                                    3.63                                                                           (3H, m), 2.44 (2H, tr),                                                        2.13-2.03                                                                      (2H, m)                           13.20                                                                             CH.sub.3                                                                          H  H  1 H  H   H  H   C═O    H  CH.sub.3                                                                          NMR (CDCl.sub.3), 300 MHz:                                                     δ [ppm] =                                                                17.25 (1H, s), 8.14 (1H, d),                                                   7.33                                                                           (1H, d), 3.87 (1H, m),                                                         3.69-3.58                                                                      (1H, m), 3.28 (1H, m),                                                         2.96-2.79 (2H,                                                                 m), 2.62 (3H, s), 2.57-2.44                                                    (2H, m),                                                                       2.40-2.13 (2H, m), 1.15 (3H,                                                   d)                                13.21                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  1 H  H   H  H   C═O    H  CH.sub.3                                                                          NMR (CDCl.sub.3), 300 MHz:                                                     δ [ppm] =                                                                17.30 (1H, m), 8.13 (1H, d),                                                   7.34                                                                           (1H, d), 3.82 (1H, m), 3.64                                                    (1H, m),                                                                       3.40-3.25 (1H, m), 2.91 (1H,                                                   m), 2.70                                                                       (2H, s), 2.64 (3H, s), 2.31                                                    (2H, s), 1.15                                                                  (6H, s)                           13.22                                                                             H  H  H  2 H  H   H  H   C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                                                                          m.p. [° C.]: 143           13.23                                                                             CH.sub.3                                                                          H  H  2 H  H   H  H   C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                                                                          m.p. [° C.]: 62            13.24                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                                                                          m.p. [° C.]: 75            13.25                                                                             H  H  H  2 H  H   H  H   C═NOCH.sub.2 CH═CHCl                                                              H  CH.sub.3                                                                          m.p. [° C.]: 75            13.26                                                                             H  H  H  2 H  H   H  H   C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                                                                          m.p. [° C.]: 192           13.27                                                                             CH.sub.3                                                                          H  H  2 H  H   H  H   C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                                                                          m.p. [° C.]: 143           13.28                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   C═NOCH.sub.2 C.sub.6 H.sub.5                                                          H  CH.sub.3                                                                          m.p. [° C.]: 126           13.29                                                                             H  H  H  2 H  H   H  H   C═NO-tButyl                                                                           H  CH.sub.3                                                                          m.p. [° C.]: 98            13.30                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   C═NO-tButyl                                                                           H  CH.sub.3                                                                          m.p. [° C.]: 91            13.31                                                                             H  H  H  2 H  H   H  H   C═O    H  Cl NMR (d.sup.6 -DMSO), 300                                                       MHz: δ [ppm] =                                                           8.05 (1H, d), 7.69 (1H, d),                                                    4.18                                                                           (2H, m), 3.31 (2H, m), 2.62                                                    (4H, m), 1.96 (2H, m)             13.32                                                                             CH.sub.3                                                                          H  H  2 H  H   H  H   C═O    H  Cl m.p. [° C.]: 66            13.33                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   C═O    H  Cl m.p. [° C.]: 104           13.34                                                                             H  H  H  2 H  H   H  H   CHOCH.sub.3                                                                               H  Cl m.p. [° C.]: 97            13.35                                                                             CH.sub.3                                                                          H  H  2 H  H   H  H   CHOCH.sub.3                                                                               H  Cl m.p. [° C.]: 86            13.36                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   CHOCH.sub.3                                                                               H  Cl m.p. [° C.]: 92            13.37                                                                             H  H  H  2 H  H   H  H   C(CH.sub.3).sub.2                                                                         H  CH.sub.3                                                                          m.p. [° C.]: 165           13.38                                                                             CH.sub.3                                                                          H  H  2 H  H   H  H   C(CH.sub.3).sub.2                                                                         H  CH.sub.3                                                                          m.p. [° C.]: 92            13.39                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   C(CH.sub.3).sub.2                                                                         H  CH.sub.3                                                                          m.p. [° C.]: 107           13.40                                                                             H  H  H  2 H  H   H  H   C═NOC.sub.2 H.sub.5                                                                   H  CH.sub.3                                                                          .sup.1 H-NMR (CDCl.sub.3),                                                     250 MHz:                                                                       δ [ppm] = 16.8, 8.20,                                                    7.32, 4.33, 3.37,                                                              2.82, 2.45, 2.08, 1.35            13.41                                                                             H  H  H  2 H  H   H  H   CH.sub.2   H  CH.sub.3                                                                          m.p. [° C.]: 199           13.42                                                                             H  H  H  2 H  CH.sub.3                                                                           H  H   CHOCH.sub.3 (trans)                                                                       H  CH.sub.3                                                                          m.p. [° C.]: 95                                                         (decomp.)                         13.43                                                                             CH.sub.3                                                                          H  H  2 H  CH.sub.3                                                                           H  H   CHOCH.sub.3 (trans)                                                                       H  CH.sub.3                                                                          m.p. [° C.]: 79-82         13.44                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  CH.sub.3                                                                           H  H   CHOCH.sub.3 (trans)                                                                       H  CH.sub.3                                                                          m.p. [° C.]: 136-137       13.45                                                                             H  H  H  2 CH.sub.3                                                                          CH.sub.3                                                                           H  H   CHOCH.sub.3                                                                               H  CH.sub.3                                                                          m.p. [° C.]: 118           13.46                                                                             CH.sub.3                                                                          H  H  2 CH.sub.3                                                                          CH.sub.3                                                                           H  H   CHOCH.sub.3                                                                               H  CH.sub.3                                                                          m.p. [° C.]: 110           13.47                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 CH.sub.3                                                                          CH.sub.3                                                                           H  H   CHOCH.sub.3                                                                               H  CH.sub.3                                                                          m.p. [° C.]: 95                                                         (decomp.)                         13.48                                                                             H  H  H  0 H  H   H  H   CH(C.sub.6 H.sub.5)                                                                       H  CH.sub.3                                                                          m.p. [° C.]: 81            13.49                                                                             H  H  H  2 H  H   CH.sub.3                                                                          H   CHOCH.sub.3                                                                               H  CH.sub.3                                                                          m.p. [° C.]: 100           13.50                                                                             CH.sub.3                                                                          H  H  2 H  H   CH.sub.3                                                                          H   CHOCH.sub.3                                                                               H  CH.sub.3                                                                          m.p. [° C.]: 86            13.51                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   CH.sub.3                                                                          H   CHOCH.sub.3                                                                               H  CH.sub.3                                                                          m.p. [° C.]: 149           13.52                                                                             H  H  H  2 H  H   H  H   CH(C.sub.6 H.sub.5)                                                                       H  CH.sub.3                                                                          m.p. [° C.]: 124           13.53                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   CH(C.sub.6 H.sub.5)                                                                       H  CH.sub.3                                                                          m.p. [° C.]: 115           13.54                                                                             H  H  H  2 H  H   H  H   CHNHOC.sub.2 H.sub.5                                                                      H  CH.sub.3                                                                          m.p. [° C.]: 98            13.55                                                                             H  H  H  2 H  CH.sub.3                                                                           H  H   CHOCH.sub.3 (cis)                                                                         H  CH.sub.3                                                                          m.p. [° C.]: 108           13.56                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   CHSO.sub.2 C.sub.6 H.sub.5                                                                H  CH.sub.3                                                                          m.p. [° C.]: 140           13.57                                                                             H  H  H  2 H  H   H  H   CHSO.sub.2 C.sub.6 H.sub.5                                                                H  CH.sub.3                                                                          m.p. [° C.]: 125           13.58                                                                             CH.sub.3                                                                          CH.sub.3                                                                          H  2 H  H   H  H   CHOH       Cl Cl m.p. [° C.]: 88            13.59                                                                             H  H  H  2 H  H   H  H   C(CH.sub.3).sub.2                                                                         Cl Cl m.p. [° C.]: 200                                                        (decomp.)                         __________________________________________________________________________

                                      TABLE 14                                     __________________________________________________________________________     Compounds of the formula                                                        ##STR297##                                                                                                   Physical data                                   No. R.sup.17                                                                          R.sup.18                                                                          R.sup.19                                                                          n R.sup.12                                                                          R.sup.13                                                                          Y    L M  m.p. [° C.]                              __________________________________________________________________________     14.001                                                                             H  H  H  2 H  H  CHOCH.sub.3                                                                         H CH.sub.3                                                                          70                                              __________________________________________________________________________

                                      TABLE 15                                     __________________________________________________________________________     Compounds of the formula                                                        ##STR298##                                                                                                  Physical data                                    No.                                                                               R.sup.17                                                                          R.sup.18                                                                          R.sup.19                                                                          n R.sup.12                                                                          R.sup.13                                                                           Y  L  M  m.p. [° C.]                               __________________________________________________________________________     15.1                                                                              H  H  H  0 H  H   C═O                                                                           H  CH.sub.3                                                                          184                                              15.2                                                                              CH.sub.3                                                                          H  H  0 H  H   C═O                                                                           H  CH.sub.3                                                                          178-180                                          15.3                                                                              CH.sub.3                                                                          CH.sub.3                                                                          H  0 H  H   C═O                                                                           H  CH.sub.3                                                                          198                                              __________________________________________________________________________

                                      TABLE 16                                     __________________________________________________________________________     Compounds of the formula                                                        ##STR299##                                                                                                  Physical data                                    No.                                                                               R.sup.3    n X    Y  L  M  m.p. [° C.]                               __________________________________________________________________________     16.1                                                                              1-Methylthiocyclopropyl                                                                   0 (CH.sub.2).sub.2                                                                    C═O                                                                           H  CH.sub.3                                                                          151-153                                          16.2                                                                              1-Methylthiocyclopropyl                                                                   2 (CH.sub.2).sub.2                                                                    C═O                                                                           H  CH.sub.3                                                                          133-135                                          __________________________________________________________________________

The compounds I and their agriculturally utilizable salts are suitable as herbicides, both in the form of isomer mixtures and in pure isomer form. The isomer-containing herbicidal compositions provide highly effective control of plant growth on uncultivated areas, in particular at high application rates. They act against broad-leaved weeds and grass weeds in crops such as wheat, rice, maize, soybeans and cotton without significantly harming the crop plants. This effect occurs especially at low application rates.

In consideration of the versatility of the application methods, the compounds I or compositions containing them can additionally be employed in a further number of crop plants for the elimination of undesired plants. Suitable crops, for example, are the following:

Allium cepa, Ananas comosus, Arachis hypogaea, Asparagus officinalis, Beta vulgaris spec. altissima, Beta vulgaris spec. rapa, Brassica napus var. napus, Brassica napus var. napobrassica, Brassica rapa var. silvestris, Camellia sinensis, Carthamus tinctorius, Carya illinoinensis, Citrus limon, Citrus sinensis, Coffea arabica (Coffea canephora, Coffea liberica), Cucumis sativus, Cynodon dactylon, Daucus carota, Elaeis guineensis, Fragaria vesca, Glycine max, Gossypium hirsutum (Gossypium arboreum, Gossypium herbaceum, Gossypium vitifolium), Helianthus annuus, Hevea brasiliensis, Hordeum vulgare, Humulus lupulus, Ipomoea batatas, Juglans regia, Lens culinaris, Linum usitatissimum, Lycopersicon lycopersicum, Malus spec., Manihot esculenta, Medicago sativa, Musa spec., Nicotiana tabacum (N. rustica), Olea europaea, Oryza sativa, Phaseolus lunatus, Phaseolus vulgaris, Picea abies, Pinus spec., Pisum sativum, Prunus avium, Prunus persica, Pyrus communis, Ribes sylvestre, Ricinus communis, Saccharum officinarum, Secale cereale, Solanum tuberosum, Sorghum bicolor (s. vulgare), Theobroma cacao, Trifolium pratense, Triticum aestivum, Triticum durum, Vicia faba, Vitis vinifera, Zea mays.

Moreover, the compounds I can also be used in crops which are tolerant to the action of herbicides as a result of breeding, including genetic engineering methods.

The compounds I and the herbicidal compositions containing them can be applied by spraying, atomizing, dusting, scattering or watering, for example in the form of directly sprayable aqueous solutions, powders, suspensions, even high-percentage aqueous, oily or other suspensions, or dispersions, emulsions, oil dispersions, pastes, dusting compositions, scattering compositions or granules. The application forms depend on the intended uses; in each case they should if possible ensure the finest dispersion of the active compounds according to the invention.

Suitable inert additives are mineral oil fractions of medium to high boiling point, such as kerosene or diesel oil, further coal tar oils and oils of vegetable or animal origin, aliphatic, cyclic and aromatic hydrocarbons, e.g. paraffin, tetrahydronaphthalene, alkylated naphthalenes or their derivatives, alkylated benzenes or their derivatives, methanol, ethanol, propanol, butanol, cyclohexanol, cyclohexanone or strongly polar solvents, such as N-methylpyrrolidone or water.

Aqueous application forms can be prepared from emulsion concentrates, dispersions, pastes, wettable powders or water-dispersible granules by addition of water. To prepare emulsions, pastes or oil dispersions, the substrates can be homogenized in water as such or dissolved in an oil or solvent, by means of wetting agents, adhesives, dispersants or emulsifiers. However, concentrates consisting of active substance, wetting agent, adhesive, dispersant or emulsifier and possibly solvent or oil can also be prepared which are suitable for dilution with water.

Suitable surface-active substances (adjuvants) are the alkali metal, alkaline earth metal or ammonium salts of aromatic sulfonic acids, e.g. lignosulfonic, phenolsulfonic, naphthalenesulfonic and dibutylnaphthalenesulfonic acid, and also of fatty acids, alkyl and alkylarylsulfonates, alkyl, lauryl ether and fatty alcohol sulfates, as well as salts of sulfated hexa-, hepta- and octadecanols, and also of fatty alcohol glycol ether, condensation products of sulfonated naphthalene and its derivatives with formaldehyde, condensation products of naphthalene or of the naphthalenesulfonic acids with phenol and formaldehyde, polyoxyethylene octylphenol ethers, ethoxylated isooctyl-, octyl- or nonylphenol, alkylphenyl or tributylphenyl polyglycol ethers, alkyl-aryl polyether alcohols, isotridecyl alcohol, fatty alcohol-ethylene oxide condensates, ethoxylated castor oil, polyoxyethylene alkyl ethers or polyoxypropylene alkyl ethers, lauryl alcohol polyglycol ether acetate, sorbitol esters, lignin-sulfite waste liquors or methylcellulose.

Powder, scattering and dusting compositions can be prepared by mixing or joint grinding of the active substances with a solid carrier.

Granules, e.g. coated, impregnated and homogeneous granules, can be prepared by binding the active compounds to solid carriers. Solid carriers are mineral earths such as silicic acids, silica gels, silicates, talc, kaolin, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate and magnesium sulfate, magnesium oxide, ground synthetic materials, fertilizers, such as ammonium sulfate, ammonium phosphate, ammonium nitrate, ureas and vegetable products, such as grain flour, tree bark, wood and nutshell meal, cellulose powder or other solid carriers.

The concentrations of the active compounds I in the ready-to-use preparations can be varied within wide ranges. The formulations in general contain from 0.001 to 98% by weight, preferably from 0.01 to 95% by weight, of at least one active compound. The active compounds are employed here in a purity of from 90 to 100%, preferably 95 to 100% (according to NMR spectrum).

The compounds I according to the invention can be formulated, for example, as follows

I. 20 parts by weight of the compound No. 13.1 are dissolved in a mixture which consists of 80 parts by weight of alkylated benzene, 10 parts by weight of the addition product of from 8 to 10 mol of ethylene oxide to 1 mol of oleic acid N-monoethanolamide, 5 parts by weight of calcium dodecylbenzenesulfonate and 5 parts by weight of the addition product of 40 mol of ethylene oxide to 1 mol of castor oil. By pouring out the solution and finely dispersing it in 100,000 parts by weight of water, an aqueous dispersion is obtained which contains 0.02% by weight of the active compound.

II. 20 parts by weight of the compound No. 13.3 are dissolved in a mixture which consists of 40 parts by weight of cyclohexanone, 30 parts by weight of isobutanol, 20 parts by weight of the addition product of 40 mol of isooctylphenol and 10 parts by weight of the addition product of 40 mol of ethylene oxide to 1 mol of castor oil. By pouring the solution into and finely dispersing it in 100,000 parts by weight of water, an aqueous dispersion is obtained which contains 0.02% by weight of the active compound.

III. 20 parts by weight of the active compound No. 13.8 are dissolved in a mixture which consists of 25 parts by weight of cyclohexanone, 65 parts by weight of a mineral oil fraction of boiling point from 210 to 280° C. and 10 parts by weight of the addition product of 40 mol of ethylene oxide to 1 mol of castor oil. By pouring the solution into and finely dispersing it in 100,000 parts by weight of water, an aqueous dispersion is obtained which contains 0.02% by weight of the active compound.

IV. 20 parts by weight of the active compound No. 13.9 are well mixed with 3 parts by weight of the sodium salt of diisobutylnaphthalene-α-sulfonic acid, 17 parts by weight of the sodium salt of a lignosulfonic acid from a sulfite waste liquor and 60 parts by weight of powdered silica gel and the mixture is ground in a hammer mill. By finely dispersing the mixture in 20,000 parts by weight of water, a spray mixture is contained obtained which contains 0.1% by weight of the active compound.

V. 3 parts by weight of the active compound No. 13.5 are mixed with 97 parts by weight of finely divided kaolin. In this manner, a dusting composition is obtained which contains 3% by weight of the active compound.

VI. 20 parts by weight of the active compound No. 13.15 are intimately mixed with 2 parts by weight of calcium salt of dodecylbenzenesulfonic acid, 8 parts by weight of fatty alcohol polyglycol ether, 2 parts by weight of sodium salt of a phenol/urea/formaldehyde condensate and 68 parts by weight of a paraffinic mineral oil. A stable oily dispersion is obtained.

VII. 1 part by weight of the active compound No. 13.16 is dissolved in a mixture which consists of 70 parts by weight of cyclohexanone, 20 parts by weight of ethoxylated isooctylphenol and 10 parts by weight of ethoxylated castor oil. A stable emulsion concentrate is obtained.

VIII. 1 part by weight of the active compound No. 13.17 is dissolved in a mixture which consists of 80 parts by weight of cyclohexanone and 20 parts by weight of Wettol® EM 31 (=nonionic emulsifier based on ethoxylated castor oil). A stable emulsion concentrate is obtained.

The application of the active compounds I or of the herbicidal compositions can be carried out pre-emergence or post-emergence. If the active compounds are less tolerable for certain crop plants, application techniques can be used in which the herbicidal compositions are sprayed with the aid of the spray equipment such that the leaves of the sensitive crop plants are not affected if possible, while the active compounds reach the leaves of undesired plants growing under them or the uncovered soil surface (post-directed, lay-by).

Depending on the aim of control, time of year, target plants and stage of growth, the application rates of active compound are from 0.001 to 3.0, preferably from 0.01 to 1.0, kg/ha of active substance (a.s.).

To widen the spectrum of action and to achieve synergistic effects, the benzoyl derivatives I can be mixed and applied together with numerous representatives of other herbicidal or growth-regulating active compound groups. For example, suitable mixture components are 1,2,4-thiadiazoles, 1,3,4-thiadiazoles, amides, aminophosphoric acid and its derivatives, aminotriazoles, anilides, aryloxy-/heteroaryloxyalkanoic acids and their derivatives, benzoic acid and its derivatives, benzothiadiazinones, 2-(heteroaryl/aroyl)-1,3-cyclohexadiones, heteroaryl aryl ketones, benzylisoxazolidinones, meta-CF₃ -phenyl derivatives, carbamates, quinolinecarboxylic acid and its derivatives, chloroacetanilides, cyclohexane-1,3-dione derivatives, diazines, dichloropropionic acid and its derivatives, dihydrobenzofurans, dihydrofuran-3-ones, dinitroanilines, dinitrophenols, diphenyl ethers, dipyridyls, halocarboxylic acids and their derivatives, ureas, 3-phenyluracils, imidazoles, imidazolinones, N-phenyl-3,4,5,6-tetrahydrophthalimides, oxadiazoles, oxiranes, phenols, aryloxy- and heteroaryloxyphenoxypropionic acid esters, phenylacetic acid and its derivatives, 2-phenylpropionic acid and its derivatives, pyrazoles, phenylpyrazoles, pyridazines, pyridinecarboxylic acid and its derivatives, pyrimidyl ethers, sulfonamides, sulfonylureas, triazines, triazinones, triazolinones, tirazolecarboxamides and uracils.

Additionally, it may be useful to apply the compounds I on their own or in combination with other herbicides additionally mixed with further crop protection agents, for example with agents for controlling pests or phytopathogenic fungi or bacteria. Further of interest is the miscibility with mineral salt solutions, which are employed for the elimination of nutritional and trace element deficiencies. Nonphytotoxic oils and oil concentrates can also be added.

Use Examples

It was possible to show the herbicidal action of the benzoyl derivatives of the formula I by greenhouse tests:

The cultivation containers used were plastic flowerpots containing loamy sand with about 3.0% humus as a substrate. The seeds of the test plants were sown separately according to species.

In the case of pre-emergence treatment, the active compounds suspended or emulsified in water were applied directly after sowing by means of finely dispersing nozzles. The containers were lightly watered to promote germination and growth and then covered with transparent plastic hoods until the plants had taken root. This covering causes uniform germination of the test plants if this has not been adversely affected by the active compounds.

For the purposes of post-emergence application, the test plants, depending on growth form, were first raised to a height growth of from 3 to 15 cm and only then treated with the active compounds suspended or emulsified in water. For this purpose, the test plants were either sown directly and grown in the same containers or they were first raised separately as seedlings and transplanted into the test containers a few days before treatment.

The application rate for post-emergence treatment was from 0.5 to 0.25 kg/ha of a.s.

The plants were kept species-specifically at from 10-25° C. or 20-35° C. The test period extended over 2 to 4 weeks. During this time, the plants were tended and their reaction to the individual treatments was assessed.

Assessment was carried out on a scale of from 0 to 100. 100 here means no emergence of the plants or complete destruction of at least the above-ground parts and 0 means no damage or normal course of growth.

The plants used in the greenhouse tests were made up of the following species:

    ______________________________________                                         Botanical Name  English Name                                                   ______________________________________                                         Chenopodium album                                                                              lambs-quarters                                                 (CHEAL)         (goosefoot)                                                    Ipomoea subspecies                                                                             morning glory                                                  (IPOSS)                                                                        Sinapis alba    white mustard                                                  (SINAL)                                                                        Solanum nigrum  black nightshade                                               (SOLNI)                                                                        Triticum aestivum                                                                              summer wheat                                                   (TRZAS)                                                                        Zea mays        Indian corn                                                    (ZEAMX)                                                                        ______________________________________                                    

                  TABLE 17                                                         ______________________________________                                         Herbicidal activity in the case of post-emergence application in               the greenhouse                                                                  ##STR300##                                                                               Ex. No.                                                                        13.3                                                                           Application rate (kg/ha of a.s.)                                               0.5      0.25                                                       Test plants  Damage in %                                                       ______________________________________                                         TRZAS         0          0                                                     CHEAL        95         95                                                     SINAL        95         95                                                     SOLNI        100        95                                                     ______________________________________                                    

                  TABLE 18                                                         ______________________________________                                         Herbicidal activity in the case of post-emergence application in               the greenhouse                                                                  ##STR301##                                                                               Ex. No.                                                                        13.13                                                                          Application rate (kg/ha of a.s.)                                               0.5      0.25                                                       Test plants  Damage in %                                                       ______________________________________                                         ZEAMX         10         0                                                     CHEAL         95         95                                                    IPOSS        100        100                                                    SOLNI        100        100                                                    ______________________________________                                     

We claim:
 1. A benzoyl compound of the formula I ##STR302## where the substituents have the following meanings: L and M are hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, where these groups may carry one to five halogen atoms or C₁ -C₄ -alkoxy; halogen, cyano, nitro, a group --(A)_(m) --S(O)_(n) R¹ or a group --(A)_(m) --CO--R² ;Y is CR¹⁰ R¹¹ ; X is --CR¹² R¹³ --CR²¹ R²² -- or --CR¹² ═CR¹³ --; the bond between X and Y can be saturated or unsaturated; A is O or NR¹⁴ ; m is zero or one; n is zero, one or two; R¹ is C₁ -C₄ -alkyl, C₁ -C₄ -haloalkyl or NR¹⁴ ; R² is C₁ -C₄ -alkyl, C₁ -C₄ -haloalkyl, C₁ -C₄ -alkoxy or NR¹⁴ ; R¹⁰, R¹¹ independently of one another are hydrogen, C₁ -C₆ -alkyl; unsubstituted or substituted phenyl, wherein the substituents are selected from the group consisting of one to three halogens, C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy and nitro; R¹⁰ and R¹² or R¹⁰ and R²¹ can form a bond; R¹² and R¹³ independently of one another are hydrogen, C₁ -C₆ -alkyl, C₁ -C₆ -haloalkyl, C₁ -C₆ -alkoxy, C₁ -C₆ -haloalkoxy; unsubstituted or substituted phenyl, wherein the substituents are selected from the group consisting of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano and nitro; R¹⁴ is C₁ -C₄ -alkyl; R²¹ is hydrogen, C₁ -C₆ -alkyl, C₁ -C₆ -haloalkyl, C₁ -C₆ -alkoxy, C₁ -C₆ -haloalkoxy; unsubstituted or substituted phenyl, wherein the substituents are selected from the group consisting of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano and nitro; R²² is hydrogen, C₁ -C₆ -alkyl, C₁ -C₆ -haloalkyl, C₁ -C₆ -alkoxy, C₁ -C₆ -haloalkoxy; unsubstituted or substituted phenyl, wherein the substituents are selected from the group consisting of C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkyl, halogen, cyano and nitro; Q is a cyclohexane-1,3-dione ring, which is linked in the 2-position, of the formula II ##STR303## where R¹⁵, R¹⁶, R¹⁸ and R²⁰ are hydrogen or C₁ -C₄ -alkyl, R¹⁹ is hydrogen, C₁ -C₄ -alkyl or a group --COOR¹⁴, R¹⁷ is hydrogen, C₁ -C₄ -alkyl, C₃ -C₄ -cycloalkyl, where these groups may carry one to three of the following substituents: halogen, C₁ -C₄ -alkylthio or C₁ -C₄ -alkoxy, or R¹⁷ is tetrahydropyran-3-yl, tetrahydropyran-4-yl or tetrahydrothiopyran-3-yl, or R¹⁷ and R²⁰ together form a bond or a three to six-membered carbocyclic ring,or an agriculturally utilizable salt thereof.
 2. A benzoyl compound of the formula Ia ##STR304## where L is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -alkylthio, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkylthio, C₁ -C₄ -alkylsulfonyl, halogen, nitro or cyano,M is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -alkylthio, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, C₁ -C₄ -haloalkylthio, C₁ -C₄ -alkylsulfonyl, halogen, nitro or cyano, and Q, X, n and Y have the meanings given in claim
 1. 3. A benzoyl compound of the formula Ib ##STR305## where L is C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano,M is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano, and Q, X, n and Y have the meanings given in claim
 1. 4. The benzoyl compound of the formula I as defined in claim 1 where the radicals L and M are hydrogen, methyl, methoxy, chlorine, cyano, nitro or trifluoromethyl.
 5. A benzoyl compound of the formula Ic ##STR306## where L is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano,M is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano, and Q, n, Y and R²², R²¹, R¹² and R¹³ have the meanings given in claim
 1. 6. A benzoyl compound of the formula Ie ##STR307## where L is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano,M is hydrogen, C₁ -C-C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, halogen, nitro or cyano, and Q, n, Y and R¹² and R¹³ have the meanings given in claim
 1. 7. A herbicidal composition comprising at least one benzoyl compound of the formula I as defined in claim 1 and customary inert additives.
 8. A method of controlling undesirable vegetation, which comprises allowing a herbicidally active amount of a benzoyl compound of the formula I as defined in claim 1 to act on the plants or their environment.
 9. A process for preparing a compound of the formula I as defined in claim 1, which comprises acylating a 1,3-cyclohexanedione of the formula II ##STR308## with an acid chloride of the formula IIIa or an acid IIIb, ##STR309## and rearranging the acylation product in the presence of a catalyst to give the compound I.
 10. A benzoyl compound of the formula IIIc ##STR310## where T, L, M, X, n and Y have the following meanings: T is chlorine, OH or C₁ -C₄ -alkoxy;L is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, C₁ -C₄ -alkylthio, C₁ -C₄ -halothioalkyl, C₁ -C₄ -alkylsulfonyl, halogen, nitro or cyano; M is C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, C₁ -C₄ -alkylthio, C₁ -C₄ -halothioalkyl, C₁ -C₄ -alkylsulfonyl, halogen, nitro or cyano; X is --CR¹² R¹³ --CR²¹ R²² -- or --CR¹² ═CR¹³ --; Y is CR¹⁰ R¹¹ ; n is zero, one or two.
 11. A benzoyl compound of the formula IIId ##STR311## where T, L, M, X, n and Y have the following meanings: T is chlorine, OH or C₁ -C₄ -alkoxy;L is C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, C₁ -C₄ -alkylthio, C₁ -C₄ -halothioalkyl, C₁ -C₄ -alkylsulfonyl, halogen or cyano; M is hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₄ -alkoxy, C₁ -C₄ -haloalkyl, C₁ -C₄ -haloalkoxy, C₁ -C₄ -alkylthio, C₁ -C₄ -halothioalkyl, C₁ -C₄ -alkylsulfonyl, halogen, nitro or cyano; X is --CR¹² R¹³ --CR²¹ R²² -- or --CR¹² ═CR¹³ --; Y is CR¹⁰ R¹¹ ; n is zero, one or two. 